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1VXG
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NATIVE SPERM WHALE MYOGLOBIN
分子名称: MYOGLOBIN, PROTOPORPHYRIN IX CONTAINING FE, SULFATE ION
著者Yang, F, Phillips Jr, G.N.
登録日1996-01-09
公開日1996-08-01
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structures of CO-, deoxy- and met-myoglobins at various pH values.
J.Mol.Biol., 256, 1996
1VXF
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NATIVE SPERM WHALE MYOGLOBIN
分子名称: CARBON MONOXIDE, MYOGLOBIN, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Yang, F, Phillips Jr, G.N.
登録日1996-01-09
公開日1996-08-01
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structures of CO-, deoxy- and met-myoglobins at various pH values.
J.Mol.Biol., 256, 1996
1VXH
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BU of 1vxh by Molmil
NATIVE SPERM WHALE MYOGLOBIN
分子名称: MYOGLOBIN, PROTOPORPHYRIN IX CONTAINING FE, SULFATE ION
著者Yang, F, Phillips Jr, G.N.
登録日1996-01-09
公開日1996-08-01
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structures of CO-, deoxy- and met-myoglobins at various pH values.
J.Mol.Biol., 256, 1996
1JEA
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BU of 1jea by Molmil
ALTERED TOPOLOGY AND FLEXIBILITY IN ENGINEERED SUBTILISIN
分子名称: CALCIUM ION, SUBTILISIN, SULFATE ION
著者Bott, R.
登録日1997-05-20
公開日1997-11-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Engineered Bacillus lentus subtilisins having altered flexibility.
J.Mol.Biol., 292, 1999
3HV3
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BU of 3hv3 by Molmil
Human p38 MAP Kinase in Complex with RL49
分子名称: 1-{4-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1H-pyrazol-5-yl]urea, GLYCEROL, Mitogen-activated protein kinase 14, ...
著者Gruetter, C, Simard, J.R, Getlik, M, Rauh, D.
登録日2009-06-15
公開日2009-11-17
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Displacement assay for the detection of stabilizers of inactive kinase conformations.
J.Med.Chem., 53, 2010
1JGG
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Even-skipped Homeodomain Complexed to AT-rich DNA
分子名称: 5'-D(P*AP*AP*TP*TP*CP*AP*AP*TP*TP*A)-3', 5'-D(P*TP*AP*AP*TP*TP*GP*AP*AP*TP*T)-3', Segmentation Protein Even-Skipped
著者Hirsch, J.A, Aggarwal, A.K.
登録日2001-06-25
公開日2001-07-06
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure of the even-skipped homeodomain complexed to AT-rich DNA: new perspectives on homeodomain specificity.
EMBO J., 14, 1995
1WBK
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BU of 1wbk by Molmil
HIV-1 protease in complex with asymmetric inhibitor, BEA568
分子名称: N,N-[2,5-O-DIBENZYL-GLUCARYL]-DI-[1-AMINO-INDAN-2-OL], POL PROTEIN (FRAGMENT)
著者Lindberg, J, Unge, T.
登録日2004-11-02
公開日2004-11-04
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献HIV-1 Protease in Complex with Asymmetric Inhibitor, Bea568
To be Published
1JC6
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BU of 1jc6 by Molmil
SOLUTION STRUCTURE OF BUNGARUS FACIATUS IX, A KUNITZ-TYPE CHYMOTRYPSIN INHIBITOR
分子名称: VENOM BASIC PROTEASE INHIBITORS IX AND VIIIB
著者Chen, C, Hsu, C.H, Su, N.Y, Chiou, S.H, Wu, S.H.
登録日2001-06-08
公開日2003-06-17
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献Solution structure of a Kunitz-type chymotrypsin inhibitor isolated from the elapid snake Bungarus fasciatus
J.BIOL.CHEM., 276, 2001
1VXC
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NATIVE SPERM WHALE MYOGLOBIN
分子名称: CARBON MONOXIDE, MYOGLOBIN, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Yang, F, Phillips Jr, G.N.
登録日1996-01-09
公開日1996-08-01
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structures of CO-, deoxy- and met-myoglobins at various pH values.
J.Mol.Biol., 256, 1996
2DNM
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BU of 2dnm by Molmil
Solution structure of RNA binding domain in SRp46 splicing factor
分子名称: SRp46 splicing factor
著者Tsuda, K, Muto, Y, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-04-26
公開日2006-10-26
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of RNA binding domain in SRp46 splicing factor
To be Published
2DO2
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BU of 2do2 by Molmil
Design of specific inhibitors of phospholipase A2: Crystal structure of the complex formed between a group II Cys 49 phospholipase A2 and a designed pentapeptide Ala-Leu-Ala-Ser-Lys at 2.6A resolution
分子名称: Ala-Leu-Ala-Ser-Lys, Phospholipase A2 VRV-PL-VIIIa, SULFATE ION
著者Singh, N, Sharma, S, Somvanshi, R.K, Dey, S, Singh, T.P.
登録日2006-04-27
公開日2006-05-16
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Design of specific inhibitors of phospholipase A2: Crystal structure of the complex formed between a group II Cys 49 phospholipase A2 and a designed pentapeptide Ala-Leu-Ala-Ser-Lys at 2.6A resolution
To be Published
1W6X
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BU of 1w6x by Molmil
SH3 domain of p40phox, component of the NADPH oxidase
分子名称: NEUTROPHIL CYTOSOL FACTOR 4
著者Massenet, C, Chenavas, S, Cohen-Addad, C, Dagher, M.-C, Brandolin, G, Pebay-Peyroula, E, Fieschi, F.
登録日2004-08-24
公開日2005-01-18
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Effects of P47Phox C-Terminus Phosphorylation on Binding Interactions with P40Phox and P67Phox: Structural and Functional Comparison of P40Phox P67Phox SH3 Domains
J.Biol.Chem., 280, 2005
1JCO
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BU of 1jco by Molmil
Solution structure of the monomeric [Thr(B27)->Pro,Pro(B28)->Thr] insulin mutant (PT insulin)
分子名称: Insulin A chain, Insulin B chain
著者Keller, D, Clausen, R, Josefsen, K, Led, J.J.
登録日2001-06-11
公開日2001-10-03
最終更新日2021-10-27
実験手法SOLUTION NMR
主引用文献Flexibility and bioactivity of insulin: an NMR investigation of the solution structure and folding of an unusually flexible human insulin mutant with increased biological activity.
Biochemistry, 40, 2001
2DQK
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Crystal structure of the complex of proteinase K with a specific lactoferrin peptide Val-Leu-Leu-His at 1.93 A resolution
分子名称: CALCIUM ION, NITRATE ION, Proteinase K, ...
著者Singh, A.K, Singh, N, Sharma, S, Dey, S, Bhushan, A, Singh, T.P.
登録日2006-05-29
公開日2006-06-20
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献Crystal structure of the complex of proteinase K with a specific lactoferrin peptide Val-Leu-Leu-His at 1.93 resolution
To be Published
1JEF
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BU of 1jef by Molmil
TURKEY LYSOZYME COMPLEX WITH (GLCNAC)3
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, LYSOZYME, SULFATE ION
著者Harata, K, Muraki, M.
登録日1997-04-23
公開日1997-10-15
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献X-ray structure of turkey-egg lysozyme complex with tri-N-acetylchitotriose. Lack of binding ability at subsite A.
Acta Crystallogr.,Sect.D, 53, 1997
2DDI
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BU of 2ddi by Molmil
NMR structure of the second Kunitz domain of human WFIKKN1
分子名称: WAP, follistatin/kazal, immunoglobulin, ...
著者Liepinsh, E, Otting, G.
登録日2006-01-30
公開日2006-12-19
最終更新日2022-03-09
実験手法SOLUTION NMR
主引用文献Second Kunitz-type protease inhibitor domain of the human WFIKKN1 protein
J.Biomol.Nmr, 35, 2006
1W8C
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BU of 1w8c by Molmil
CO-CRYSTAL STRUCTURE OF 6-CYCLOHEXYLMETHOXY-8-ISOPROPYL-9H-PURIN-2- YLAMINE AND MONOMERIC CDK2
分子名称: 6-(CYCLOHEXYLMETHOXY)-8-ISOPROPYL-9H-PURIN-2-AMINE, CELL DIVISION PROTEIN KINASE 2
著者Pratt, D.J, Endicott, J.A, Noble, M.E.M.
登録日2004-09-20
公開日2006-08-30
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献8-Substituted O6-Cyclohexylmethylguanine Cdk2 Inhibitors; Using Structure-Based Inhibitor Design to Optimise an Alternative Binding Mode.
J.Med.Chem., 57, 2014
1JF3
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BU of 1jf3 by Molmil
Crystal Structure Of Component III Glycera Dibranchiata Monomeric Hemoglobin
分子名称: PROTOPORPHYRIN IX CONTAINING FE, monomer hemoglobin component III
著者Park, H.J, Yang, C, Treff, N, Satterlee, J.D, Kang, C.H.
登録日2001-06-20
公開日2002-06-20
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Crystal Structures of Unligated and CN-Ligated Glycera dibranchiata Monomer Ferric Hemoglobin Components III and IV
Proteins, 49, 2002
3HUB
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BU of 3hub by Molmil
Human p38 MAP Kinase in Complex with Scios-469
分子名称: 2-(6-chloro-5-{[(2R,5S)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1H-indol-3-yl)-N,N-dimethyl-2-oxoacetamide, Mitogen-activated protein kinase 14, octyl beta-D-glucopyranoside
著者Gruetter, C, Simard, J.R, Rauh, D.
登録日2009-06-13
公開日2010-03-09
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Fluorophore labeling of the glycine-rich loop as a method of identifying inhibitors that bind to active and inactive kinase conformations.
J.Am.Chem.Soc., 132, 2010
1VYZ
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BU of 1vyz by Molmil
Structure of CDK2 complexed with PNU-181227
分子名称: CELL DIVISION PROTEIN KINASE 2, N-(5-CYCLOPROPYL-1H-PYRAZOL-3-YL)BENZAMIDE
著者Pevarello, P, Brasca, M.G, Amici, R, Orsini, P, Traquandi, G, Corti, L, Piutti, C, Sansonna, P, Villa, M, Pierce, B.S, Pulici, M, Giordano, G, Martina, K, Lfritzen, E, Nugent, R.A, Casale, E, Cameron, A, Ciomei, M, Roletto, F, Isacchi, A, Fogliatto, G, Pesenti, E, Pastori, W, Marsiglio, W, Leach, K.L, Clare, P.M, Fiorentini, F, Varasi, M, Vulpetti, A, Warpehoski, M.A.
登録日2004-05-07
公開日2004-06-17
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.21 Å)
主引用文献3-Aminopyrazole Inhibitors of Cdk2/Cyclin a as Antitumor Agents. 1. Lead Finding
J.Med.Chem., 47, 2004
1JFB
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X-ray structure of nitric oxide reductase (cytochrome P450nor) in the ferric resting state at atomic resolution
分子名称: GLYCEROL, PROTOPORPHYRIN IX CONTAINING FE, nitric-oxide reductase cytochrome P450 55A1
著者Shimizu, H, Adachi, S, Park, S.Y, Shiro, Y, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2001-06-20
公開日2001-12-20
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1 Å)
主引用文献X-ray structure of nitric oxide reductase (cytochrome P450nor) at atomic resolution.
Acta Crystallogr.,Sect.D, 58, 2002
2DGQ
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Solution structure of the N-terminal RNA binding domain in Bruno-like 6 RNA-binding protein
分子名称: bruno-like 6, RNA binding protein
著者Abe, C, Muto, Y, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-03-15
公開日2006-09-15
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the N-terminal RNA binding domain in Bruno-like 6 RNA-binding protein
To be Published
1W5W
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HIV-1 protease in complex with fluoro substituted diol-based C2- symmetric inhibitor
分子名称: (2R,3R,4R,5R)-2,5-BIS[(2,4-DIFLUOROBENZYL)OXY]-3,4-DIHYDROXY-N,N'-BIS[(1R,2S)-2-HYDROXY-2,3-DIHYDRO-1H-INDEN-1-YL]HEXAN EDIAMIDE, POL POLYPROTEIN
著者Lindberg, J, Pyring, D, Loewgren, S, Rosenquist, A, Zuccarello, G, Kvarnstroem, I, Zhang, H, Vrang, L, Claesson, B, Hallberg, A, Samuelsson, B, Unge, T.
登録日2004-08-10
公開日2004-12-22
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Symmetric Fluoro-Substituted Diol-Based HIV Protease Inhibitors. Ortho-Fluorinated and Meta-Fluorinated P1/P1'-Benzyloxy Side Groups Significantly Improve the Antiviral Activity and Preserve Binding Efficacy
Eur.J.Biochem., 271, 2004
2DIZ
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The solution structure of the third thioredoxin domain of human Thioredoxin domain-containing protein 5
分子名称: Thioredoxin domain-containing protein 5
著者Tochio, N, Koshiba, S, Inoue, M, Kigawa, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-03-30
公開日2006-09-30
最終更新日2022-03-09
実験手法SOLUTION NMR
主引用文献The solution structure of the third thioredoxin domain of human Thioredoxin domain-containing protein 5
To be Published
1JI0
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Crystal Structure Analysis of the ABC transporter from Thermotoga maritima
分子名称: ABC transporter, ADENOSINE-5'-TRIPHOSPHATE
著者Zhang, R, Joachimiak, A, Edwards, A, Savchenko, A, Beasley, S, Midwest Center for Structural Genomics (MCSG)
登録日2001-06-28
公開日2002-08-14
最終更新日2017-10-04
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The 2.0 A Crystal Structure of ABC Transporter from Thermotoga maritima
TO BE PUBLISHED

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