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3HV3

Human p38 MAP Kinase in Complex with RL49

Summary for 3HV3
Entry DOI10.2210/pdb3hv3/pdb
Related3GCP 3GCQ 3GCS 3GCU 3GCV 3HV4 3HV5 3HV6 3HV7
DescriptorMitogen-activated protein kinase 14, 1-{4-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1H-pyrazol-5-yl]urea, octyl beta-D-glucopyranoside, ... (5 entities in total)
Functional Keywordsdfg-out, type ii, rl49, quinoline-pyrazolourea, hybrid, atp-binding, kinase, nucleotide-binding, nucleus, phosphoprotein, serine/threonine-protein kinase, transferase
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight42125.05
Authors
Gruetter, C.,Simard, J.R.,Getlik, M.,Rauh, D. (deposition date: 2009-06-15, release date: 2009-11-17, Last modification date: 2023-09-06)
Primary citationKluter, S.,Grutter, C.,Naqvi, T.,Rabiller, M.,Simard, J.R.,Pawar, V.,Getlik, M.,Rauh, D.
Displacement assay for the detection of stabilizers of inactive kinase conformations.
J.Med.Chem., 53:357-367, 2010
Cited by
PubMed: 19928858
DOI: 10.1021/jm901297e
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2 Å)
Structure validation

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