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4ES0
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X-ray structure of WDR5-SETd1b Win motif peptide binary complex
分子名称: Histone-lysine N-methyltransferase SETD1B, WD repeat-containing protein 5
著者Dharmarajan, V, Lee, J.-H, Patel, A, Skalnik, D.G, Cosgrove, M.S.
登録日2012-04-21
公開日2012-05-30
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.817 Å)
主引用文献Structural basis for WDR5 interaction (Win) motif recognition in human SET1 family histone methyltransferases.
J.Biol.Chem., 287, 2012
2JUP
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BU of 2jup by Molmil
FBP28WW2 domain in complex with the PPLIPPPP peptide
分子名称: Formin-1, Transcription elongation regulator 1
著者Ramirez-Espain, X, Ruiz, L, Martin-Malpartida, P, Oschkinat, H, Macias, M.J.
登録日2007-09-01
公開日2007-11-06
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献Structural Characterization of a New Binding Motif and a Novel Binding Mode in Group 2 WW Domains
J.Mol.Biol., 373, 2007
2K2F
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BU of 2k2f by Molmil
Solution structure of Ca2+-S100A1-RyRP12
分子名称: CALCIUM ION, Protein S100-A1, Ryanodine receptor 1 peptide
著者Wright, N.T, Varney, K.M, Weber, D.J.
登録日2008-04-01
公開日2008-07-29
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献S100A1 and Calmodulin Compete for the Same Binding Site on Ryanodine Receptor.
J.Biol.Chem., 283, 2008
1FJL
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BU of 1fjl by Molmil
HOMEODOMAIN FROM THE DROSOPHILA PAIRED PROTEIN BOUND TO A DNA OLIGONUCLEOTIDE
分子名称: DNA (5'-D(*AP*AP*TP*AP*AP*TP*CP*TP*GP*AP*TP*TP*AP*C)-3'), DNA (5'-D(*TP*GP*TP*AP*AP*TP*CP*AP*GP*AP*TP*TP*AP*T)-3'), DNA (5'-D(*TP*GP*TP*AP*AP*TP*CP*TP*GP*AP*TP*TP*AP*C)-3'), ...
著者Wilson, D.S, Guenther, B, Desplan, C, Kuriyan, J.
登録日1995-12-17
公開日1996-06-20
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献High resolution crystal structure of a paired (Pax) class cooperative homeodomain dimer on DNA.
Cell(Cambridge,Mass.), 82, 1995
2KZ5
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Solution NMR Structure of Transcription factor NF-E2 subunit's DNA binding domain from Homo sapiens, Northeast Structural Genomics Consortium Target HR4653B
分子名称: Transcription factor NF-E2 45 kDa subunit
著者Liu, G, Janjua, H, Xiao, R, Ciccosanti, C, Shastry, R, Acton, T.B, Tong, S, Everett, J.K, Montelione, G.T, Northeast Structural Genomics Consortium (NESG)
登録日2010-06-11
公開日2010-07-07
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Northeast Structural Genomics Consortium Target HR4653B
To be Published
1QRJ
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BU of 1qrj by Molmil
Solution structure of htlv-i capsid protein
分子名称: HTLV-I CAPSID PROTEIN
著者Khorasanizadeh, S, Campos-Olivas, R, Clark, C.A, Summers, M.F.
登録日1999-06-14
公開日1999-07-13
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献Sequence-specific 1H, 13C and 15N chemical shift assignment and secondary structure of the HTLV-I capsid protein.
J.Biomol.NMR, 14, 1999
1RO4
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BU of 1ro4 by Molmil
RDC-derived models of the zinc ribbon domain of human general transcription factor TFIIB (zinc free structures)
分子名称: Transcription initiation factor IIB
著者Ghosh, M, Ikura, M.
登録日2003-12-01
公開日2004-05-25
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Probing Zn2+-binding effects on the zinc-ribbon domain of human general transcription factor TFIIB.
Biochem.J., 378, 2004
1J7V
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BU of 1j7v by Molmil
HUMAN IL-10 / IL-10R1 COMPLEX
分子名称: INTERLEUKIN-10, INTERLEUKIN-10 RECEPTOR ALPHA CHAIN
著者Josephson, K, Logsdon, N, Walter, M.R.
登録日2001-05-18
公開日2001-09-19
最終更新日2021-10-27
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal structure of the IL-10/IL-10R1 complex reveals a shared receptor binding site.
Immunity, 15, 2001
8T0E
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TRPV1 in Nanodisc not bound with lysophosphatidic acid (apo)
分子名称: (2R)-3-{[(R)-hydroxy{[(1S,2R,3R,4S,5S,6R)-2,3,4,5,6-pentahydroxycyclohexyl]oxy}phosphoryl]oxy}propane-1,2-diyl dioctadecanoate, SODIUM ION, Transient receptor potential cation channel subfamily V member 1
著者Arnold, W.R, Cheng, Y.
登録日2023-05-31
公開日2024-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Structural basis of TRPV1 modulation by endogenous bioactive lipids.
Nat.Struct.Mol.Biol., 2024
8T0C
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TRPV1 in Nanodisc bound with lysophosphatidic acid in all four monomers
分子名称: (2R)-2-hydroxy-3-(phosphonooxy)propyl tetradecanoate, SODIUM ION, Transient receptor potential cation channel subfamily V member 1
著者Arnold, W.R, Cheng, Y.
登録日2023-05-31
公開日2024-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Structural basis of TRPV1 modulation by endogenous bioactive lipids.
Nat.Struct.Mol.Biol., 2024
8T10
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TRPV1 in nanodisc bound with two LPA molecules in opposite monomers
分子名称: (2R)-2-hydroxy-3-(phosphonooxy)propyl tetradecanoate, (2R)-3-{[(R)-hydroxy{[(1S,2R,3R,4S,5S,6R)-2,3,4,5,6-pentahydroxycyclohexyl]oxy}phosphoryl]oxy}propane-1,2-diyl dioctadecanoate, SODIUM ION, ...
著者Arnold, W.R, Julius, D, Cheng, Y.
登録日2023-06-01
公開日2024-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献Structural basis of TRPV1 modulation by endogenous bioactive lipids.
Nat.Struct.Mol.Biol., 2024
8T0Y
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BU of 8t0y by Molmil
TRPV1 in nanodisc bound with one LPA in one monomer
分子名称: (2R)-2-hydroxy-3-(phosphonooxy)propyl tetradecanoate, (2R)-3-{[(R)-hydroxy{[(1S,2R,3R,4S,5S,6R)-2,3,4,5,6-pentahydroxycyclohexyl]oxy}phosphoryl]oxy}propane-1,2-diyl dioctadecanoate, SODIUM ION, ...
著者Arnold, W.R, Cheng, Y.
登録日2023-06-01
公開日2024-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Structural basis of TRPV1 modulation by endogenous bioactive lipids.
Nat.Struct.Mol.Biol., 2024
2MBH
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BU of 2mbh by Molmil
NMR structure of EKLF(22-40)/Ubiquitin Complex
分子名称: Krueppel-like factor 1, Ubiquitin
著者Raiola, L, Omichinski, J.G.
登録日2013-07-31
公開日2013-10-09
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Structural Characterization of a Noncovalent Complex between Ubiquitin and the Transactivation Domain of the Erythroid-Specific Factor EKLF.
Structure, 21, 2013
1PY2
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BU of 1py2 by Molmil
Structure of a 60 nM Small Molecule Bound to a Hot Spot on IL-2
分子名称: 5-[2,3-DICHLORO-4-(5-{1-[2-(2-GUANIDINO-4-METHYL-PENTANOYLAMINO)-ACETYL]-PIPERIDIN-4-YL}-1-METHYL-1H-PYRAZOL-3-YL)-PHENOXYMETHYL]-FURAN-2-CARBOXYLIC ACID, Interleukin-2, ZINC ION
著者Thanos, C.D, Randal, M, Wells, J.A.
登録日2003-07-07
公開日2004-01-13
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Potent small-molecule binding to a dynamic hot spot on IL-2.
J.Am.Chem.Soc., 125, 2003
2LZ1
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BU of 2lz1 by Molmil
Solution NMR Structure of the DNA-Binding Domain of Human NF-E2-Related Factor 2, Northeast Structural Genomics Consortium (NESG) Target HR3520O
分子名称: Nuclear factor erythroid 2-related factor 2
著者Eletsky, A, Pulavarti, S.V.S.R.K, Lee, D, Kohan, E, Janjua, H, Xiao, R, Acton, T.B, Everett, J.K, Montelione, G.T, Szyperski, T, Northeast Structural Genomics Consortium (NESG)
登録日2012-09-22
公開日2012-11-28
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Solution NMR Structure of the DNA-Binding Domain of Human NF-E2-Related Factor 2, Northeast Structural Genomics Consortium (NESG) Target HR3520O
To be Published
1SKN
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BU of 1skn by Molmil
THE BINDING DOMAIN OF SKN-1 IN COMPLEX WITH DNA: A NEW DNA-BINDING MOTIF
分子名称: DNA (5'-D(*CP*AP*GP*GP*GP*AP*TP*GP*AP*CP*AP*TP*TP*GP*T)-3'), DNA (5'-D(*TP*GP*AP*CP*AP*AP*TP*GP*TP*CP*AP*TP*CP*CP*C)-3'), DNA-BINDING DOMAIN OF SKN-1, ...
著者Rupert, P.B, Daughdrill, G.W, Bowerman, B, Matthews, B.W.
登録日1998-03-30
公開日1998-06-24
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献A new DNA-binding motif in the Skn-1 binding domain-DNA complex.
Nat.Struct.Biol., 5, 1998
7BRP
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BU of 7brp by Molmil
Crystal structure of the 2019-nCoV main protease complexed with Boceprevir
分子名称: 3C-like proteinase, boceprevir (bound form)
著者Fu, L.F.
登録日2020-03-29
公開日2020-05-13
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Both Boceprevir and GC376 efficaciously inhibit SARS-CoV-2 by targeting its main protease.
Nat Commun, 11, 2020
1QB3
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BU of 1qb3 by Molmil
CRYSTAL STRUCTURE OF THE CELL CYCLE REGULATORY PROTEIN CKS1
分子名称: CYCLIN-DEPENDENT KINASES REGULATORY SUBUNIT
著者Bourne, Y, Watson, M.H, Arvai, A.S, Bernstein, S.L, Reed, S.I, Tainer, J.A.
登録日1999-04-30
公開日2000-08-31
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Crystal structure and mutational analysis of the Saccharomyces cerevisiae cell cycle regulatory protein Cks1: implications for domain swapping, anion binding and protein interactions.
Structure Fold.Des., 8, 2000
1QQP
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FOOT-AND-MOUTH DISEASE VIRUS/ OLIGOSACCHARIDE RECEPTOR COMPLEX.
分子名称: 2-O-sulfo-alpha-L-gulopyranuronic acid-(1-4)-2-deoxy-6-O-sulfo-2-(sulfoamino)-alpha-D-glucopyranose-(1-4)-2-O-sulfo-alpha-L-idopyranuronic acid-(1-4)-2-deoxy-6-O-sulfo-2-(sulfoamino)-alpha-D-glucopyranose-(1-4)-2-O-sulfo-alpha-L-gulopyranuronic acid, PROTEIN (GENOME POLYPROTEIN)
著者Fry, E.E, Lea, S.M, Jackson, T, Newman, J.W.I, Ellard, F.M, Blakemore, W.E, Abu-Ghazaleh, R, Samuel, A, King, A.M.Q, Stuart, D.I.
登録日1999-05-20
公開日1999-06-18
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献The structure and function of a foot-and-mouth disease virus-oligosaccharide receptor complex.
EMBO J., 18, 1999
3Q33
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BU of 3q33 by Molmil
Structure of the Rtt109-AcCoA/Vps75 Complex and Implications for Chaperone-Mediated Histone Acetylation
分子名称: 1,2-ETHANEDIOL, ACETYL COENZYME *A, HISTONE H3, ...
著者Tang, Y, Yuan, H, Meeth, K, Marmorstein, R.
登録日2010-12-21
公開日2011-02-02
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure of the Rtt109-AcCoA/Vps75 Complex and Implications for Chaperone-Mediated Histone Acetylation.
Structure, 19, 2011
7BRO
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BU of 7bro by Molmil
Crystal structure of the 2019-nCoV main protease
分子名称: 3C-like proteinase
著者Fu, L.F.
登録日2020-03-29
公開日2020-05-13
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Both Boceprevir and GC376 efficaciously inhibit SARS-CoV-2 by targeting its main protease.
Nat Commun, 11, 2020
8U30
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BU of 8u30 by Molmil
TRPV1 in nanodisc bound with diC8-PIP2 in the closed state
分子名称: SODIUM ION, Transient receptor potential cation channel subfamily V member 1, [(2R)-2-octanoyloxy-3-[oxidanyl-[(1R,2R,3S,4R,5R,6S)-2,3,6-tris(oxidanyl)-4,5-diphosphonooxy-cyclohexyl]oxy-phosphoryl]oxy-propyl] octanoate
著者Arnold, W.R, Julius, D, Cheng, Y.
登録日2023-09-06
公開日2024-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3 Å)
主引用文献Structural basis of TRPV1 modulation by endogenous bioactive lipids.
Nat.Struct.Mol.Biol., 2024
8U3C
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TRPV1 in nanodisc bound with PI-Br4 bound in Conformation 2 (monomer)
分子名称: (2S)-2-[(9,10-dibromooctadecanoyl)oxy]-3-{[(S)-hydroxy{[(1S,2R,3R,4S,5S,6R)-2,3,4,5,6-pentahydroxycyclohexyl]oxy}phosphoryl]oxy}propyl (9R,10S)-9,10-dibromooctadecanoate, 1,2-DIACYL-GLYCEROL-3-SN-PHOSPHATE, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, ...
著者Arnold, W.R, Julius, D, Cheng, Y.
登録日2023-09-07
公開日2024-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (2.3 Å)
主引用文献Structural basis of TRPV1 modulation by endogenous bioactive lipids.
Nat.Struct.Mol.Biol., 2024
6ZZ6
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Cryo-EM structure of S.cerevisiae cohesin-Scc2-DNA complex
分子名称: ADENOSINE-5'-TRIPHOSPHATE, DNA (34-MER), MAGNESIUM ION, ...
著者Lee, B.-G, Gonzalez Llamazares, A, Collier, J, Nasmyth, K.A, Lowe, J.
登録日2020-08-04
公開日2020-09-30
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Transport of DNA within cohesin involves clamping on top of engaged heads by Scc2 and entrapment within the ring by Scc3.
Elife, 9, 2020
8U3L
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TRPV1 in nanodisc bound with empty vanilloid binding pocket at 25C
分子名称: 1,2-DIACYL-GLYCEROL-3-SN-PHOSPHATE, SODIUM ION, Transient receptor potential cation channel subfamily V member 1
著者Arnold, W.R, Julius, D, Cheng, Y.
登録日2023-09-07
公開日2024-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献Structural basis of TRPV1 modulation by endogenous bioactive lipids.
Nat.Struct.Mol.Biol., 2024

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