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8RQR
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In meso structure of apolipoprotein N-acyltransferase, Lnt, from Escherichia coli in 7.10 monoacylglycerol
分子名称: 7.10 monoacylglycerol (S-form), Apolipoprotein N-acyltransferase, GLYCEROL
著者Smithers, L, Boland, C, Krawinski, P, Caffrey, M.
登録日2024-01-19
公開日2024-04-03
最終更新日2024-04-17
実験手法X-RAY DIFFRACTION (2.19 Å)
主引用文献7.10 MAG. A Novel Host Monoacylglyceride for In Meso (Lipid Cubic Phase) Crystallization of Membrane Proteins.
Cryst.Growth Des., 24, 2024
8SNZ
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BU of 8snz by Molmil
X-ray Crystal Structure of FMN-bound long-chain flavodoxin from Rhodopseudomonas palustris
分子名称: FLAVIN MONONUCLEOTIDE, Flavodoxin
著者Ansari, A, Khan, S.A, Miller, A.F.
登録日2023-04-28
公開日2024-03-13
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.17 Å)
主引用文献Structure, dynamics, and redox reactivity of an all-purpose flavodoxin.
J.Biol.Chem., 300, 2024
8SEI
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BU of 8sei by Molmil
SF Tau from Down Syndrome
分子名称: Microtubule-associated protein tau
著者Hoq, M.R, Bharath, S.R, Jiang, W, Vago, F.S, Bharath, S.R.
登録日2023-04-10
公開日2024-04-03
最終更新日2024-06-26
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献Cryo-EM structures of amyloid-beta and tau filaments in Down syndrome.
Nat.Struct.Mol.Biol., 31, 2024
8SAG
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BU of 8sag by Molmil
Carbonic anhydrase II in complex with the coumarin benzene sulfonamide SG1-57
分子名称: 2-[(2-oxo-2H-1-benzopyran-7-yl)oxy]-N-[(4-sulfamoylphenyl)methyl]acetamide, Carbonic anhydrase 2, GLYCEROL, ...
著者Combs, J.E, Mckenna, R.
登録日2023-03-31
公開日2024-04-03
実験手法X-RAY DIFFRACTION (1.52 Å)
主引用文献Carbonic anhydrase II in complex with novel coumarin benzene sulfonamides
To Be Published
8SAJ
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BU of 8saj by Molmil
Mycobacterium phage Adjutor
分子名称: HNH endonuclease, Major capsid protein, gp_16 (Minor Capsid Protein)
著者Podgorski, J.M, White, S.J.
登録日2023-04-01
公開日2024-04-03
実験手法ELECTRON MICROSCOPY (2.66 Å)
主引用文献A novel accessory protein stabilizes the capsid of two actinobacteriophages
To Be Published
5D3X
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BU of 5d3x by Molmil
Crystal Structure of the P-Rex1 PH domain with Inositol-(1,3,4,5)-Tetrakisphosphate Bound
分子名称: INOSITOL-(1,3,4,5)-TETRAKISPHOSPHATE, Phosphatidylinositol 3,4,5-trisphosphate-dependent Rac exchanger 1 protein
著者Cash, J.N, Tesmer, J.J.G.
登録日2015-08-06
公開日2016-04-20
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.69 Å)
主引用文献Structural and Biochemical Characterization of the Catalytic Core of the Metastatic Factor P-Rex1 and Its Regulation by PtdIns(3,4,5)P3.
Structure, 24, 2016
8SL4
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BU of 8sl4 by Molmil
Dimeric form of human adenylyl cyclase 5
分子名称: Adenylate cyclase type 5
著者Yen, Y.C, Tesmer, J.J.G.
登録日2023-04-20
公開日2024-04-03
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (7 Å)
主引用文献Structure of adenylyl cyclase 5 in complex with G beta gamma offers insights into ADCY5-related dyskinesia.
Nat.Struct.Mol.Biol., 2024
8SM8
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Air-oxidized A. ca TruffO expressed from M9 minimal medium supplemented with Fe
分子名称: FE (III) ION, MAGNESIUM ION, Putative amidohydrolase, ...
著者Liu, C, Rittle, J.
登録日2023-04-25
公開日2024-03-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Bioinformatic Discovery of a Cambialistic Monooxygenase.
J.Am.Chem.Soc., 146, 2024
5D4A
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Crystal Structure of FABP4 in complex with 3-(2-phenyl-1H-indol-1-yl)propanoic acid
分子名称: 3-(2-phenyl-1H-indol-1-yl)propanoic acid, Fatty acid-binding protein, adipocyte
著者Tagami, U, Takahashi, K, Igarashi, S, Ejima, C, Yoshida, T, Takeshita, S, Miyanaga, W, Sugiki, M, Tokumasu, M, Hatanaka, T, Kashiwagi, T, Ishikawa, K, Miyano, H, Mizukoshi, T.
登録日2015-08-07
公開日2016-06-22
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Interaction Analysis of FABP4 Inhibitors by X-ray Crystallography and Fragment Molecular Orbital Analysis
Acs Med.Chem.Lett., 7, 2016
8SO9
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BU of 8so9 by Molmil
Phosphoinositide phosphate 3 kinase gamma
分子名称: Phosphoinositide 3-kinase regulatory subunit 5, phosphatidylinositol-4,5-bisphosphate 3-kinase
著者Chen, C.-L, Tesmer, J.J.G.
登録日2023-04-28
公開日2024-04-03
最終更新日2024-04-17
実験手法ELECTRON MICROSCOPY (3.03 Å)
主引用文献Molecular basis for G beta gamma-mediated activation of phosphoinositide 3-kinase gamma.
Nat.Struct.Mol.Biol., 2024
8SAF
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CA II in complex with the coumarin benzene sulfonamide SG1-51
分子名称: 2-[(2-oxo-3,4-dihydro-2H-1-benzopyran-7-yl)oxy]-N-(4-sulfamoylphenyl)acetamide, Carbonic anhydrase 2, ZINC ION
著者Combs, J.E, Mckenna, R.
登録日2023-03-31
公開日2024-04-03
実験手法X-RAY DIFFRACTION (1.23 Å)
主引用文献CA in complex with novel coumarin benzene sulfonamides
To Be Published
8SEJ
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BU of 8sej by Molmil
Type I beta-amyloid 42 Filaments from Down syndrome
分子名称: Amyloid-beta protein 42
著者Hoq, M.R, Bharath, S.R, Vago, F.S, Jiang, W.
登録日2023-04-10
公開日2024-04-03
最終更新日2024-06-26
実験手法ELECTRON MICROSCOPY (3.17 Å)
主引用文献Cryo-EM structures of amyloid-beta and tau filaments in Down syndrome.
Nat.Struct.Mol.Biol., 31, 2024
8SOA
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BU of 8soa by Molmil
Phosphoinositide phosphate 3 kinase gamma bound with ATP
分子名称: ADENOSINE-5'-TRIPHOSPHATE, Phosphoinositide 3-kinase regulatory subunit 5, phosphatidylinositol-4,5-bisphosphate 3-kinase
著者Chen, C.-L, Tesmer, J.J.G.
登録日2023-04-28
公開日2024-04-03
最終更新日2024-04-17
実験手法ELECTRON MICROSCOPY (3.32 Å)
主引用文献Molecular basis for G beta gamma-mediated activation of phosphoinositide 3-kinase gamma.
Nat.Struct.Mol.Biol., 2024
2FU5
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BU of 2fu5 by Molmil
structure of Rab8 in complex with MSS4
分子名称: BETA-MERCAPTOETHANOL, Guanine nucleotide exchange factor MSS4, Ras-related protein Rab-8A, ...
著者Itzen, A, Pylypenko, O, Goody, R.S, Rak, A.
登録日2006-01-26
公開日2006-04-04
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Nucleotide exchange via local protein unfolding-structure of Rab8 in complex with MSS4
Embo J., 25, 2006
8S03
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BU of 8s03 by Molmil
NMR solution structure of the CysD2 domain of MUC2
分子名称: CALCIUM ION, Mucin-2
著者Recktenwald, C, Karlsson, B.G, Garcia-Bonnete, M.-J, Katona, G, Jensen, M, Lymer, R, Baeckstroem, M, Johansson, M.E.V, Hansson, G.C, Trillo-Muyo, S.
登録日2024-02-13
公開日2024-04-17
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献The structure of the second CysD domain of MUC2 and role in mucin organization by transglutaminase-based cross-linking.
Cell Rep, 43, 2024
8S5I
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BU of 8s5i by Molmil
Full-length human cystathionine beta-synthase with C-terminal 6xHis-tag, basal state, single particle reconstruction
分子名称: Cystathionine beta-synthase, PROTOPORPHYRIN IX CONTAINING FE
著者McCorvie, T.J, Yue, W.W.
登録日2024-02-23
公開日2024-04-17
実験手法ELECTRON MICROSCOPY (3.1 Å)
主引用文献Architecture and regulation of filamentous human cystathionine beta-synthase.
Nat Commun, 15, 2024
2FT9
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BU of 2ft9 by Molmil
Crystal structure of axolotl (Ambystoma mexicanum) liver bile acid-binding protein bound to cholic acid
分子名称: CHOLIC ACID, Fatty acid-binding protein 2, liver
著者Capaldi, S, Guariento, M, Perduca, M, Di Pietro, S.M, Santome, J.A, Monaco, H.L.
登録日2006-01-24
公開日2006-04-11
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of axolotl (Ambystoma mexicanum) liver bile acid-binding protein bound to cholic and oleic acid
Proteins, 64, 2006
8SBQ
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BU of 8sbq by Molmil
FphE, Staphylococcus aureus fluorophosphonate-binding serine hydrolases E, fluorophosphonate JB101 bound
分子名称: Fluorophosphonate-binding serine hydrolases E, MAGNESIUM ION, ethyl (R)-(10-{[(but-3-yn-1-yl)carbamoyl]oxy}decyl)phosphonofluoridate
著者Fellner, M.
登録日2023-04-04
公開日2024-04-17
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献FphE, Staphylococcus aureus fluorophosphonate-binding serine hydrolases E, fluorophosphonate JB101 bound
To Be Published
2FW8
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BU of 2fw8 by Molmil
Structure of PurE (N5-carboxyaminoimidazole ribonucleotide mutase) H89G from the acidophilic bacterium Acetobacter aceti, at pH 8
分子名称: N5-carboxyaminoimidazole ribonucleotide mutase
著者Starks, C.M, Kappock, T.J.
登録日2006-02-01
公開日2006-06-13
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Biochemical and Structural Studies of N(5)-Carboxyaminoimidazole Ribonucleotide Mutase from the Acidophilic Bacterium Acetobacter aceti.
Biochemistry, 45, 2006
5DGD
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BU of 5dgd by Molmil
Benzoylformate decarboxylase F464I and A460V mutant from Pseudomonas putida
分子名称: Benzoylformate decarboxylase, CALCIUM ION, MAGNESIUM ION, ...
著者Bera, A.K, Hasson, M.S.
登録日2015-08-27
公開日2015-09-16
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.13 Å)
主引用文献Benzoylformate decarboxylase F464I and A460V mutant from Pseudomonas putida
to be published
8SBF
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BU of 8sbf by Molmil
Full-length structure of the LysR-type transcriptional regulator, ACIAD0746, from Acinetobacter baylyi
分子名称: GLYCEROL, MAGNESIUM ION, Putative transcriptional regulator (LysR family), ...
著者Momany, C, Nune, M, Brondani, J.C, Afful, D, Neidle, E, Galloway, N.R.
登録日2023-04-03
公開日2024-04-17
実験手法X-RAY DIFFRACTION (2.29 Å)
主引用文献FinR, a LysR-type transcriptional regulator involved in sulfur homeostasis with homologs in diverse microorganisms
To Be Published
8S4G
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BU of 8s4g by Molmil
Cryo-EM structure of the Anaphase-promoting complex/cyclosome (APC/C) bound to co-activator Cdh1 at 3.2 Angstrom resolution
分子名称: Anaphase-promoting complex subunit 1, Anaphase-promoting complex subunit 10, Anaphase-promoting complex subunit 11, ...
著者Hoefler, A, Yu, J, Chang, L, Zhang, Z, Yang, J, Boland, A, Barford, D.
登録日2024-02-21
公開日2024-03-13
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献New structural features of the APC/C revealed by high resolution cryo-EM structures of apo-APC/C and the APC/C-CDH1-EMI1 complex
To Be Published
8SFT
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BU of 8sft by Molmil
Crystal structure of TuUGT202A2 (Tetur22g00270) in complex with kaempferol
分子名称: 3,5,7-TRIHYDROXY-2-(4-HYDROXYPHENYL)-4H-CHROMEN-4-ONE, SULFATE ION, UDP-glycosyltransferase 202A2, ...
著者Arriaza, R.H, Dermauw, W, Wybouw, N, Van Leeuwen, T, Chruszcz, M.
登録日2023-04-11
公開日2024-04-17
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Crystal structure of TuUGT202A2 (Tetur22g00270) in complex with kaempferol
To Be Published
5DGZ
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BU of 5dgz by Molmil
Discovery of 3,5-substituted 6-azaindazoles as potent pan-Pim inhibitors
分子名称: (2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE, PHOSPHATE ION, Serine/threonine-protein kinase pim-1
著者Murray, J.M, Wallweber, H, Steffek, M.
登録日2015-08-29
公開日2015-10-28
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.502 Å)
主引用文献Discovery of 3,5-substituted 6-azaindazoles as potent pan-Pim inhibitors.
Bioorg.Med.Chem.Lett., 25, 2015
2FY1
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A dual mode of RNA recognition by the RBMY protein
分子名称: RNA-binding motif protein, Y chromosome, family 1 member A1, ...
著者Skrisovska, L, Bourgois, C, Stefl, R, Kister, L, Wenter, P, Elliot, D, Stevenin, J, Allain, F.H.T.
登録日2006-02-07
公開日2007-02-06
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献The testis-specific human protein RBMY recognizes RNA through a novel mode of interaction.
EMBO Rep., 8, 2007

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件を2024-07-10に公開中

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