3I29
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![BU of 3i29 by Molmil](/molmil-images/mine/3i29) | Crystal structure of a binary complex between an mutant trypsin inhibitor with bovine trypsin | 分子名称: | CALCIUM ION, Cationic trypsin, Chymotrypsin inhibitor 3 | 著者 | Khamrui, S, Majumder, S, Dasgupta, J, Dattagupta, J.K, Sen, U. | 登録日 | 2009-06-29 | 公開日 | 2010-06-16 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Role of remote scaffolding residues in the inhibitory loop pre-organization, flexibility, rigidification and enzyme inhibition of serine protease inhibitors Biochim.Biophys.Acta, 1824, 2012
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4NCY
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![BU of 4ncy by Molmil](/molmil-images/mine/4ncy) | In situ trypsin crystallized on a MiTeGen micromesh with imidazole ligand | 分子名称: | 1,2-ETHANEDIOL, BENZAMIDINE, CALCIUM ION, ... | 著者 | Yin, X, Scalia, A, Leroy, L, Cuttitta, C.M, Polizzo, G.M, Ericson, D.L, Roessler, C.G, Campos, O, Agarwal, R, Allaire, M, Orville, A.M, Jackimowicz, R, Ma, M.Y, Sweet, R.M, Soares, A.S. | 登録日 | 2013-10-25 | 公開日 | 2014-04-09 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.42 Å) | 主引用文献 | Hitting the target: fragment screening with acoustic in situ co-crystallization of proteins plus fragment libraries on pin-mounted data-collection micromeshes. Acta Crystallogr.,Sect.D, 70, 2014
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3GY3
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![BU of 3gy3 by Molmil](/molmil-images/mine/3gy3) | A comparative study on the inhibition of bovine beta-trypsin by bis-benzamidines diminazene and pentamidine by X-ray crystallography and ITC | 分子名称: | 1,2-ETHANEDIOL, 1,5-BIS(4-AMIDINOPHENOXY)PENTANE, CALCIUM ION, ... | 著者 | Perilo, C.S, Pereira, M.T, Santoro, M.M, Nagem, R.A.P. | 登録日 | 2009-04-03 | 公開日 | 2010-03-23 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structural binding evidence of the trypanocidal drugs Berenil and Pentacarinate active principles to a serine protease model. Int.J.Biol.Macromol., 46, 2010
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3GY8
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![BU of 3gy8 by Molmil](/molmil-images/mine/3gy8) | A comparative study on the inhibition of bovine beta-trypsin by bis-benzamidines diminazene and pentamidine by X-ray crystallography and ITC | 分子名称: | 1,2-ETHANEDIOL, BERENIL, CALCIUM ION, ... | 著者 | Perilo, C.S, Pereira, M.T, Santoro, M.M, Nagem, R.A.P. | 登録日 | 2009-04-03 | 公開日 | 2010-03-23 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Structural binding evidence of the trypanocidal drugs Berenil and Pentacarinate active principles to a serine protease model. Int.J.Biol.Macromol., 46, 2010
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3GY6
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![BU of 3gy6 by Molmil](/molmil-images/mine/3gy6) | A comparative study on the inhibition of bovine beta-trypsin by the bis-benzamidines diminazene and pentamidine | 分子名称: | 1,2-ETHANEDIOL, BERENIL, CALCIUM ION, ... | 著者 | Perilo, C.S, Pereira, M.T, Santoro, M.M, Nagem, R.A.P. | 登録日 | 2009-04-03 | 公開日 | 2010-03-23 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structural binding evidence of the trypanocidal drugs Berenil and Pentacarinate active principles to a serine protease model. Int.J.Biol.Macromol., 46, 2010
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3GY4
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![BU of 3gy4 by Molmil](/molmil-images/mine/3gy4) | A comparative study on the inhibition of bovine beta-trypsin by bis-benzamidines diminazene and pentamidine by X-ray crystallography and ITC | 分子名称: | 1,2-ETHANEDIOL, CALCIUM ION, Cationic trypsin, ... | 著者 | Perilo, C.S, Pereira, M.T, Santoro, M.M, Nagem, R.A.P. | 登録日 | 2009-04-03 | 公開日 | 2010-03-23 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Structural binding evidence of the trypanocidal drugs Berenil and Pentacarinate active principles to a serine protease model. Int.J.Biol.Macromol., 46, 2010
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3GY5
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![BU of 3gy5 by Molmil](/molmil-images/mine/3gy5) | A comparative study on the inhibition of bovine beta-trypsin by bis-benzamidines diminazene and pentamidine by X-ray crystallography and ITC | 分子名称: | 1,2-ETHANEDIOL, BERENIL, CALCIUM ION, ... | 著者 | Perilo, C.S, Pereira, M.T, Santoro, M.M, Nagem, R.A.P. | 登録日 | 2009-04-03 | 公開日 | 2010-03-23 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.57 Å) | 主引用文献 | Structural binding evidence of the trypanocidal drugs Berenil and Pentacarinate active principles to a serine protease model. Int.J.Biol.Macromol., 46, 2010
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3GY2
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![BU of 3gy2 by Molmil](/molmil-images/mine/3gy2) | A comparative study on the inhibition of bovine beta-trypsin by bis-benzamidines diminazene and pentamidine by X-ray crystallography and ITC | 分子名称: | 1,2-ETHANEDIOL, BERENIL, CALCIUM ION, ... | 著者 | Perilo, C.S, Pereira, M.T, Santoro, M.M, Nagem, R.A.P. | 登録日 | 2009-04-03 | 公開日 | 2010-03-23 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.57 Å) | 主引用文献 | Structural binding evidence of the trypanocidal drugs Berenil and Pentacarinate active principles to a serine protease model. Int.J.Biol.Macromol., 46, 2010
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3GY7
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![BU of 3gy7 by Molmil](/molmil-images/mine/3gy7) | A comparative study on the inhibition of bovine beta-trypsin by bis-benzamidines diminazene and pentamidine by X-ray crystallography and ITC | 分子名称: | 1,2-ETHANEDIOL, BENZAMIDINE, CALCIUM ION, ... | 著者 | Perilo, C.S, Pereira, M.T, Santoro, M.M, Nagem, R.A.P. | 登録日 | 2009-04-03 | 公開日 | 2010-03-23 | 最終更新日 | 2017-11-15 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Structural binding evidence of the trypanocidal drugs Berenil and Pentacarinate active principles to a serine protease model. Int.J.Biol.Macromol., 46, 2010
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4NIX
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![BU of 4nix by Molmil](/molmil-images/mine/4nix) | Crystal structure of trypsiligase (K60E/N143H/Y151H/D189K trypsin) orthorhombic form, zinc-bound | 分子名称: | CALCIUM ION, Cationic trypsin, GLYCEROL, ... | 著者 | Schoepfel, M, Parthier, C, Stubbs, M.T. | 登録日 | 2013-11-08 | 公開日 | 2014-02-19 | 最終更新日 | 2014-03-19 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | N-terminal protein modification by substrate-activated reverse proteolysis. Angew.Chem.Int.Ed.Engl., 53, 2014
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4NIW
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![BU of 4niw by Molmil](/molmil-images/mine/4niw) | |
4NIV
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![BU of 4niv by Molmil](/molmil-images/mine/4niv) | |
4KTU
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![BU of 4ktu by Molmil](/molmil-images/mine/4ktu) | Bovine trypsin in complex with microviridin J at pH 6.5 | 分子名称: | CALCIUM ION, Cationic trypsin, microviridin j | 著者 | Quitterer, F, Groll, M, Hertweck, C, Dittmann, E. | 登録日 | 2013-05-21 | 公開日 | 2014-04-02 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | Harnessing the evolvability of tricyclic microviridins to dissect protease-inhibitor interactions. Angew.Chem.Int.Ed.Engl., 53, 2014
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4NIY
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![BU of 4niy by Molmil](/molmil-images/mine/4niy) | Crystal structure of trypsiligase (K60E/N143H/Y151H/D189K trypsin) complexed to YRH-ecotin (M84Y/M85R/A86H ecotin) | 分子名称: | CALCIUM ION, Cationic trypsin, Ecotin, ... | 著者 | Schoepfel, M, Parthier, C, Stubbs, M.T. | 登録日 | 2013-11-08 | 公開日 | 2014-02-19 | 最終更新日 | 2014-03-19 | 実験手法 | X-RAY DIFFRACTION (2.84 Å) | 主引用文献 | N-terminal protein modification by substrate-activated reverse proteolysis. Angew.Chem.Int.Ed.Engl., 53, 2014
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4KTS
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![BU of 4kts by Molmil](/molmil-images/mine/4kts) | Bovine trypsin in complex with microviridin J at pH 8.5 | 分子名称: | CALCIUM ION, Cationic trypsin, DI(HYDROXYETHYL)ETHER, ... | 著者 | Quitterer, F, Groll, M, Hertweck, C, Dittmann, E. | 登録日 | 2013-05-21 | 公開日 | 2014-04-02 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Harnessing the evolvability of tricyclic microviridins to dissect protease-inhibitor interactions. Angew.Chem.Int.Ed.Engl., 53, 2014
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3FP6
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![BU of 3fp6 by Molmil](/molmil-images/mine/3fp6) | Anionic trypsin in complex with bovine pancreatic trypsin inhibitor (BPTI) determined to the 1.49 A resolution limit | 分子名称: | 1,2-ETHANEDIOL, Anionic trypsin-2, CALCIUM ION, ... | 著者 | Zakharova, E, Horvath, M.P, Goldenberg, D.P. | 登録日 | 2009-01-04 | 公開日 | 2009-02-17 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.49 Å) | 主引用文献 | Structure of a serine protease poised to resynthesize a peptide bond. Proc.Natl.Acad.Sci.USA, 106, 2009
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8I0X
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![BU of 8i0x by Molmil](/molmil-images/mine/8i0x) | Beta-Xylosidase JB13GH39P28 showing salt/ethanol/trypsin tolerance, low-pH/low-Temperature activity, and transformation of notoginsenosides | 分子名称: | Glycoside hydrolase family 39 beta-xylosidase | 著者 | Zhou, J.P, Cao, L.J, Lin, M.Y, Zhang, R, Huang, Z.X. | 登録日 | 2023-01-11 | 公開日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | beta-Xylosidase JB13GH39P28(D41G)showing salt/ethanol/trypsin tolerance and transformation of notoginsenosides To Be Published
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1AKS
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![BU of 1aks by Molmil](/molmil-images/mine/1aks) | CRYSTAL STRUCTURE OF THE FIRST ACTIVE AUTOLYSATE FORM OF THE PORCINE ALPHA TRYPSIN | 分子名称: | ALPHA TRYPSIN, CALCIUM ION | 著者 | Johnson, A, Krishnaswamy, S, Sundaram, P.V, Pattabhi, V. | 登録日 | 1996-07-24 | 公開日 | 1997-02-12 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | The first structure at 1.8 A resolution of an active autolysate form of porcine alpha-trysoin. Acta Crystallogr.,Sect.D, 53, 1997
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3FP7
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![BU of 3fp7 by Molmil](/molmil-images/mine/3fp7) | Anionic trypsin variant S195A in complex with bovine pancreatic trypsin inhibitor (BPTI) cleaved at the scissile bond (LYS15-ALA16) determined to the 1.46 A resolution limit | 分子名称: | 1,2-ETHANEDIOL, Anionic trypsin-2, CALCIUM ION, ... | 著者 | Zakharova, E, Horvath, M.P, Goldenberg, D.P. | 登録日 | 2009-01-04 | 公開日 | 2009-02-17 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.46 Å) | 主引用文献 | Structure of a serine protease poised to resynthesize a peptide bond. Proc.Natl.Acad.Sci.USA, 106, 2009
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2PKA
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![BU of 2pka by Molmil](/molmil-images/mine/2pka) | REFINED 2 ANGSTROMS X-RAY CRYSTAL STRUCTURE OF PORCINE PANCREATIC KALLIKREIN A, A SPECIFIC TRYPSIN-LIKE SERINE PROTEINASE. CRYSTALLIZATION, STRUCTURE DETERMINATION, CRYSTALLOGRAPHIC REFINEMENT, STRUCTURE AND ITS COMPARISON WITH BOVINE TRYPSIN | 分子名称: | BENZAMIDINE, KALLIKREIN A | 著者 | Bode, W, Chen, Z. | 登録日 | 1984-05-21 | 公開日 | 1984-07-19 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Refined 2 A X-ray crystal structure of porcine pancreatic kallikrein A, a specific trypsin-like serine proteinase. Crystallization, structure determination, crystallographic refinement, structure and its comparison with bovine trypsin. J.Mol.Biol., 164, 1983
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5XWA
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![BU of 5xwa by Molmil](/molmil-images/mine/5xwa) | Crystal Structure of Porcine pancreatic trypsin with tripeptide inhibitor, PRY, at pH 10 | 分子名称: | Acetylated-Pro-Arg-Tyr Inhibitor, CALCIUM ION, Trypsin | 著者 | Saikhedkar, N.S, Bhoite, A.S, Giri, A.P, Kulkarni, K.A. | 登録日 | 2017-06-29 | 公開日 | 2018-03-28 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Tripeptides derived from reactive centre loop of potato type II protease inhibitors preferentially inhibit midgut proteases of Helicoverpa armigera. Insect Biochem. Mol. Biol., 95, 2018
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5XW9
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![BU of 5xw9 by Molmil](/molmil-images/mine/5xw9) | Crystal Structure of Porcine pancreatic trypsin with tripeptide inhibitor, PRY, at pH 7 | 分子名称: | Acetylated-Pro-Arg-Tyr Inhibitor, CALCIUM ION, Trypsin | 著者 | Saikhedkar, N.S, Bhoite, A.S, Giri, A.P, Kulkarni, K.A. | 登録日 | 2017-06-29 | 公開日 | 2018-03-28 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Tripeptides derived from reactive centre loop of potato type II protease inhibitors preferentially inhibit midgut proteases of Helicoverpa armigera. Insect Biochem. Mol. Biol., 95, 2018
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5XW8
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![BU of 5xw8 by Molmil](/molmil-images/mine/5xw8) | Crystal Structure of Porcine pancreatic trypsin with tripeptide inhibitor, PRN, at pH 7 | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, Acetylated-Pro-Arg-Asn Inhibitor, CALCIUM ION, ... | 著者 | Saikhedkar, N.S, Bhoite, A.S, Giri, A.P, Kulkarni, K.A. | 登録日 | 2017-06-29 | 公開日 | 2018-03-28 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.002 Å) | 主引用文献 | Tripeptides derived from reactive centre loop of potato type II protease inhibitors preferentially inhibit midgut proteases of Helicoverpa armigera. Insect Biochem. Mol. Biol., 95, 2018
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3FP8
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![BU of 3fp8 by Molmil](/molmil-images/mine/3fp8) | Anionic trypsin variant S195A in complex with bovine pancreatic trypsin inhibitor (BPTI) determined to the 1.46 A resolution limit | 分子名称: | 1,2-ETHANEDIOL, Anionic trypsin-2, CALCIUM ION, ... | 著者 | Zakharova, E, Horvath, M.P, Goldenberg, D.P, Curtice, K. | 登録日 | 2009-01-04 | 公開日 | 2009-02-17 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.46 Å) | 主引用文献 | Structure of a serine protease poised to resynthesize a peptide bond. Proc.Natl.Acad.Sci.USA, 106, 2009
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1BA8
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![BU of 1ba8 by Molmil](/molmil-images/mine/1ba8) | THROMBIN INHIBITOR WITH A RIGID TRIPEPTIDYL ALDEHYDES | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, HIRUGEN, THROMBIN, ... | 著者 | Krishnan, R, Zhang, E, Hakansson, K, Arni, R.K, Tulinsky, A, Lim-Wilby, M.S.L, Levy, O.E, Semple, J.E, Brunck, T.K. | 登録日 | 1998-04-23 | 公開日 | 1999-04-27 | 最終更新日 | 2023-08-02 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Highly selective mechanism-based thrombin inhibitors: structures of thrombin and trypsin inhibited with rigid peptidyl aldehydes. Biochemistry, 37, 1998
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