7UGJ
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![BU of 7ugj by Molmil](/molmil-images/mine/7ugj) | TBOA-bound GltPh RSMR mutant in OFS state | 分子名称: | (3S)-3-(BENZYLOXY)-L-ASPARTIC ACID, Glutamate transporter homolog, SODIUM ION | 著者 | Huang, Y, Boudker, O. | 登録日 | 2022-03-24 | 公開日 | 2023-03-29 | 最終更新日 | 2023-05-10 | 実験手法 | ELECTRON MICROSCOPY (2.81 Å) | 主引用文献 | Environmentally Ultrasensitive Fluorine Probe to Resolve Protein Conformational Ensembles by 19F NMR and Cryo-EM J.Am.Chem.Soc., 145, 2023
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4GMM
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4GMW
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7ULD
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4FLI
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![BU of 4fli by Molmil](/molmil-images/mine/4fli) | Human MetAP1 with bengamide analog Y16, in Mn form | 分子名称: | (E,2R,3R,4S,5R)-N-(2-azanyl-2-oxidanylidene-ethyl)-2-methoxy-8,8-dimethyl-3,4,5-tris(oxidanyl)non-6-enamide, MANGANESE (II) ION, Methionine aminopeptidase 1, ... | 著者 | Ye, Q.Z, Xu, W. | 登録日 | 2012-06-14 | 公開日 | 2012-09-19 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Structural analysis of bengamide derivatives as inhibitors of methionine aminopeptidases. J.Med.Chem., 55, 2012
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4FM6
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4FLJ
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![BU of 4flj by Molmil](/molmil-images/mine/4flj) | Human MetAP1 with bengamide analog Y08, in Mn form | 分子名称: | (E,2R,3R,4S,5R)-N-[[(3S)-1-cyclopropylcarbonylpiperidin-3-yl]methyl]-2-methoxy-8,8-dimethyl-3,4,5-tris(oxidanyl)non-6-enamide, MANGANESE (II) ION, Methionine aminopeptidase 1, ... | 著者 | Ye, Q.Z, Xu, W. | 登録日 | 2012-06-14 | 公開日 | 2012-09-19 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Structural analysis of bengamide derivatives as inhibitors of methionine aminopeptidases. J.Med.Chem., 55, 2012
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4GNO
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4GPE
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![BU of 4gpe by Molmil](/molmil-images/mine/4gpe) | Crystal Structure of Benzoylformate Decarboxylase Mutant L403M | 分子名称: | 2-{3-[(4-AMINO-2-METHYLPYRIMIDIN-5-YL)METHYL]-4-METHYL-2-OXO-2,3-DIHYDRO-1,3-THIAZOL-5-YL}ETHYL TRIHYDROGEN DIPHOSPHATE, Benzoylformate decarboxylase, CALCIUM ION, ... | 著者 | Novak, W.R.P, Andrews, F.H, Tom, A.R, Gunderman, P.R, McLeish, M.J. | 登録日 | 2012-08-20 | 公開日 | 2013-05-22 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.39 Å) | 主引用文献 | A bulky hydrophobic residue is not required to maintain the v-conformation of enzyme-bound thiamin diphosphate. Biochemistry, 52, 2013
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4H3O
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![BU of 4h3o by Molmil](/molmil-images/mine/4h3o) | Crystal structure of a new form of lectin from Allium sativum at 2.17 A resolution | 分子名称: | CADMIUM ION, Lectin, SODIUM ION | 著者 | Kumar, S, Yamini, S, Kumar, J, Kaur, P, Singh, T.P, Dey, S. | 登録日 | 2012-09-14 | 公開日 | 2012-09-26 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.17 Å) | 主引用文献 | Crystal structure of a new form of lectin from Allium sativum at 2.17 A resolution To be Published
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4GNP
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4H7O
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4HE9
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![BU of 4he9 by Molmil](/molmil-images/mine/4he9) | Crystal Structure of HIV-1 protease mutants I54M complexed with inhibitor GRL-0519 | 分子名称: | (3R,3aS,3bR,6aS,7aS)-octahydrodifuro[2,3-b:3',2'-d]furan-3-yl [(1S,2R)-1-benzyl-2-hydroxy-3-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}propyl]carbamate, CHLORIDE ION, HIV-1 protease, ... | 著者 | Shen, C.H, Zhang, H, Weber, I.T. | 登録日 | 2012-10-03 | 公開日 | 2013-08-21 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.06 Å) | 主引用文献 | Novel P2 tris-tetrahydrofuran group in antiviral compound 1 (GRL-0519) fills the S2 binding pocket of selected mutants of HIV-1 protease. J.Med.Chem., 56, 2013
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4IMQ
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![BU of 4imq by Molmil](/molmil-images/mine/4imq) | Structural Basis of Substrate Specificity and Protease Inhibition in Norwalk Virus | 分子名称: | 3C-like protease, PEPTIDE INHIBITOR, syc8, ... | 著者 | Prasad, B.V.V, Muhaxhiri, Z, Deng, L, Shanker, S, Sankaran, B, Estes, M.K, Palzkill, T, Song, Y. | 登録日 | 2013-01-03 | 公開日 | 2013-02-20 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structural basis of substrate specificity and protease inhibition in norwalk virus. J.Virol., 87, 2013
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4IHS
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![BU of 4ihs by Molmil](/molmil-images/mine/4ihs) | Crystal Structure of BenM_DBD/catB site 1 DNA Complex | 分子名称: | HTH-type transcriptional regulator BenM, MALONATE ION, SODIUM ION, ... | 著者 | Alanazi, A, Momany, C, Neidle, E.L. | 登録日 | 2012-12-19 | 公開日 | 2013-07-10 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | The DNA-binding domain of BenM reveals the structural basis for the recognition of a T-N11-A sequence motif by LysR-type transcriptional regulators. Acta Crystallogr.,Sect.D, 69, 2013
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4IN9
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![BU of 4in9 by Molmil](/molmil-images/mine/4in9) | Structure of karilysin MMP-like catalytic domain in complex with inhibitory tetrapeptide SWFP | 分子名称: | GLYCEROL, Karilysin protease, POTASSIUM ION, ... | 著者 | Guevara, T, Ksiazek, M, Skottrup, P.D, Cerda-Costa, N, Trillo-Muyo, S, de Diego, I, Riise, E, Potempa, J, Gomis-Ruth, F.X. | 登録日 | 2013-01-04 | 公開日 | 2013-05-15 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Structure of the catalytic domain of the Tannerella forsythia matrix metallopeptidase karilysin in complex with a tetrapeptidic inhibitor. Acta Crystallogr.,Sect.F, 69, 2013
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4HA4
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![BU of 4ha4 by Molmil](/molmil-images/mine/4ha4) | Structure of beta-glycosidase from Acidilobus saccharovorans in complex with glycerol | 分子名称: | 1-(2-METHOXY-ETHOXY)-2-{2-[2-(2-METHOXY-ETHOXY]-ETHOXY}-ETHANE, Beta-galactosidase, GLYCEROL, ... | 著者 | Trofimov, A.A, Polyakov, K.M, Tikhonov, A.V, Bezsudnova, E.Y, Dorovatovskii, P.V, Gumerov, V.M, Ravin, N.V, Skryabin, K.G, Popov, V.O. | 登録日 | 2012-09-25 | 公開日 | 2012-10-10 | 最終更新日 | 2013-09-04 | 実験手法 | X-RAY DIFFRACTION (1.37 Å) | 主引用文献 | Structures of beta-glycosidase from Acidilobus saccharovorans in complexes with tris and glycerol. Dokl.Biochem.Biophys., 449
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1F7Y
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![BU of 1f7y by Molmil](/molmil-images/mine/1f7y) | THE CRYSTAL STRUCTURE OF TWO UUCG LOOPS HIGHLIGHTS THE ROLE PLAYED BY 2'-HYDROXYL GROUPS IN ITS UNUSUAL STABILITY | 分子名称: | 16S RIBOSOMAL RNA FRAGMENT, 30S RIBOSOMAL PROTEIN S15, MAGNESIUM ION, ... | 著者 | Ennifar, E, Nikouline, A, Serganov, A, Tishchenko, S, Nevskaya, N, Garber, M, Ehresmann, B, Ehresmann, C, Nikonov, S, Dumas, P. | 登録日 | 2000-06-28 | 公開日 | 2000-11-22 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | The crystal structure of UUCG tetraloop. J.Mol.Biol., 304, 2000
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4GPJ
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![BU of 4gpj by Molmil](/molmil-images/mine/4gpj) | Crystal Structure of the first bromodomain of human BRD4 in complex with a isoxazolylbenzimidazole ligand | 分子名称: | (1R)-6-(3,5-dimethyl-1,2-oxazol-4-yl)-1-phenyl-2,3-dihydro-1H-inden-1-ol, 1,2-ETHANEDIOL, Bromodomain-containing protein 4, ... | 著者 | Filippakopoulos, P, Picaud, S, Qi, J, Felletar, I, Heightman, T.D, Brennan, P, von Delft, F, Bountra, C, Arrowsmith, C.H, Edwards, A, Knapp, S, Structural Genomics Consortium (SGC) | 登録日 | 2012-08-21 | 公開日 | 2012-10-17 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | The design and synthesis of 5- and 6-isoxazolylbenzimidazoles as selective inhibitors of the BET bromodomains. Medchemcomm, 4, 2013
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1NVJ
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![BU of 1nvj by Molmil](/molmil-images/mine/1nvj) | Deletion Mutant (Delta 141) of Molybdopterin Synthase | 分子名称: | FORMIC ACID, GLYCEROL, Molybdopterin converting factor subunit 2, ... | 著者 | Rudolph, M.J, Wuebbens, M.M, Turque, O, Rajagopalan, K.V, Schindelin, H. | 登録日 | 2003-02-03 | 公開日 | 2003-05-06 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Structural Studies of Molybdopterin Synthase Provide Insights into its Catalytic Mechanism J.Biol.Chem., 278, 2003
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4GYF
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![BU of 4gyf by Molmil](/molmil-images/mine/4gyf) | Crystal structure of histidinol phosphate phosphatase (HISK) from Lactococcus lactis subsp. lactis Il1403 complexed with ZN, L-histidinol and phosphate | 分子名称: | CHLORIDE ION, DI(HYDROXYETHYL)ETHER, Histidinol-phosphatase, ... | 著者 | Fedorov, A.A, Fedorov, E.V, Ghodge, S, Raushel, F.M, Almo, S.C. | 登録日 | 2012-09-05 | 公開日 | 2013-02-06 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (1.647 Å) | 主引用文献 | Crystal structure of histidinol phosphate phosphatase (HISK) from Lactococcus lactis subsp. lactis Il1403 complexed with ZN, L-histidinol and phosphate To be Published
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4GYM
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![BU of 4gym by Molmil](/molmil-images/mine/4gym) | Crystal structure of Glyoxalase/bleomycin resistance protein/dioxygenase from Conexibacter woesei DSM 14684 | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Glyoxalase/bleomycin resistance protein/dioxygenase, POTASSIUM ION, ... | 著者 | Chang, C, Tesar, C, Clancy, S, Joachimiak, A, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2012-09-05 | 公開日 | 2012-09-26 | 実験手法 | X-RAY DIFFRACTION (1.56 Å) | 主引用文献 | Crystal structure of Glyoxalase/bleomycin resistance protein/dioxygenase from Conexibacter woesei DSM 14684 To be Published
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1O9I
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![BU of 1o9i by Molmil](/molmil-images/mine/1o9i) | Crystal structure of the Y42F mutant of manganese catalase from Lactobacillus plantarum at 1.33A resolution | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, MANGANESE (III) ION, ... | 著者 | Barynin, V.V, Whittaker, M.M, Whittaker, J.W. | 登録日 | 2002-12-13 | 公開日 | 2003-12-18 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.33 Å) | 主引用文献 | Outer Sphere Mutagenesis of Lactobacillus Plantarum Manganese Catalase Disrupts the Cluster Core. Mechanistic Implications. Eur.J.Biochem., 270, 2003
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4GRN
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7XOI
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![BU of 7xoi by Molmil](/molmil-images/mine/7xoi) | Aspergillus sojae alpha-glucosidase AsojAgdL in complex with trehalose | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, SODIUM ION, ... | 著者 | Tonozuka, T. | 登録日 | 2022-05-01 | 公開日 | 2022-06-15 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural basis for proteolytic processing of Aspergillus sojae alpha-glucosidase L with strong transglucosylation activity. J.Struct.Biol., 214, 2022
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