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8FPZ
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LBD conformation 3 (LBDconf3) of GluA2 flip Q isoform of AMPA receptor in complex with gain-of-function TARP gamma-2, with 500mM NaCl, 330uM CTZ, and 100mM glutamate (Open-Na610)
分子名称: CYCLOTHIAZIDE, GLUTAMIC ACID, Glutamate receptor 2
著者Nakagawa, T.
登録日2023-01-05
公開日2024-03-06
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (3.01 Å)
主引用文献The open gate of the AMPA receptor forms a Ca 2+ binding site critical in regulating ion transport.
Nat.Struct.Mol.Biol., 31, 2024
8FQA
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BU of 8fqa by Molmil
LBD conformation 2 (LBDconf2) of GluA2 flip Q isoform of AMPA receptor in complex with gain-of-function TARP gamma2, with 140mM NMDG, 330uM CTZ, and 100mM L-glutamate (Open-Na110)
分子名称: CYCLOTHIAZIDE, GLUTAMIC ACID, Glutamate receptor 2
著者Nakagawa, T.
登録日2023-01-05
公開日2024-03-06
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (3.35 Å)
主引用文献The open gate of the AMPA receptor forms a Ca 2+ binding site critical in regulating ion transport.
Nat.Struct.Mol.Biol., 31, 2024
8GPR
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BU of 8gpr by Molmil
GluK1-1a receptor captured in the desensitized state
分子名称: Glutamate receptor
著者Dhingra, S, Kumar, J.
登録日2022-08-26
公開日2023-08-30
最終更新日2024-03-13
実験手法ELECTRON MICROSCOPY (8.2 Å)
主引用文献Functional Implications of the Exon 9 Splice Insert in GluK1 Kainate Receptors
Elife, 2023
8GC2
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Domoate-bound GluK2 kainate receptor in partially-open conformation 1
分子名称: (2S,3S,4S)-2-CARBOXY-4-[(1Z,3E,5R)-5-CARBOXY-1-METHYL-1,3-HEXADIENYL]-3-PYRROLIDINEACETIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Bogdanovic, N, Tajima, N.
登録日2023-03-01
公開日2024-03-13
実験手法ELECTRON MICROSCOPY (4.1 Å)
主引用文献Structural basis for kainate receptor activation by a partial agonist
To Be Published
8GC4
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Domoate-bound GluK2 kainate receptor in partially-open conformation 3
分子名称: (2S,3S,4S)-2-CARBOXY-4-[(1Z,3E,5R)-5-CARBOXY-1-METHYL-1,3-HEXADIENYL]-3-PYRROLIDINEACETIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Bogdanovic, N, Tajima, N.
登録日2023-03-01
公開日2024-03-13
実験手法ELECTRON MICROSCOPY (3.93 Å)
主引用文献Structural basis for kainate receptor activation by a partial agonist
To Be Published
8GC3
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Domote-bound GluK2 kainate receptors in partially-open conformation 2
分子名称: (2S,3S,4S)-2-CARBOXY-4-[(1Z,3E,5R)-5-CARBOXY-1-METHYL-1,3-HEXADIENYL]-3-PYRROLIDINEACETIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Bogdanovic, N, Tajima, N.
登録日2023-03-01
公開日2024-03-13
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献Structural basis for kainate receptor activation by a partial agonist
To Be Published
8GC5
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Domoate-bound GluK2 kainate receptors in non-active conformation
分子名称: (2S,3S,4S)-2-CARBOXY-4-[(1Z,3E,5R)-5-CARBOXY-1-METHYL-1,3-HEXADIENYL]-3-PYRROLIDINEACETIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Bogdanovic, N, Tajima, N.
登録日2023-03-01
公開日2024-03-13
実験手法ELECTRON MICROSCOPY (3.93 Å)
主引用文献Structural basis for kainate receptor activation by a partial agonist
To Be Published
8HDK
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BU of 8hdk by Molmil
Structure of the Rat GluN1-GluN2C NMDA receptor in complex with glycine and glutamate (minor class in symmetry)
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, ...
著者Zhang, M, Zhang, J, Guo, F, Li, Y, Zhu, S.
登録日2022-11-04
公開日2023-03-29
最終更新日2023-05-31
実験手法ELECTRON MICROSCOPY (4.3 Å)
主引用文献Distinct structure and gating mechanism in diverse NMDA receptors with GluN2C and GluN2D subunits.
Nat.Struct.Mol.Biol., 30, 2023
7F57
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BU of 7f57 by Molmil
Kainate-bound GluK2-1xNeto2 complex, at the desensitized state
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, kainate 2, ...
著者He, L.L, Gao, Y.W, Li, B, Zhao, Y.
登録日2021-06-21
公開日2021-09-29
最終更新日2021-12-01
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献Kainate receptor modulation by NETO2.
Nature, 599, 2021
7F56
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DNQX-bound GluK2-1xNeto2 complex, with asymmetric LBD
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, kainate 2, ...
著者He, L.L, Gao, Y.W, Li, B, Zhao, Y.
登録日2021-06-21
公開日2021-09-29
最終更新日2021-12-01
実験手法ELECTRON MICROSCOPY (4.1 Å)
主引用文献Kainate receptor modulation by NETO2.
Nature, 599, 2021
7F5A
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BU of 7f5a by Molmil
DNQX-bound GluK2-2xNeto2 complex
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, kainate 2, ...
著者He, L.L, Gao, Y.W, Li, B, Zhao, Y.
登録日2021-06-21
公開日2021-09-29
最終更新日2021-12-01
実験手法ELECTRON MICROSCOPY (6.4 Å)
主引用文献Kainate receptor modulation by NETO2.
Nature, 599, 2021
7F59
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DNQX-bound GluK2-1xNeto2 complex
分子名称: (1S)-2-{[{[(2R)-2,3-DIHYDROXYPROPYL]OXY}(HYDROXY)PHOSPHORYL]OXY}-1-[(PALMITOYLOXY)METHYL]ETHYL STEARATE, 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor ionotropic, ...
著者He, L.L, Gao, Y.W, Li, B, Zhao, Y.
登録日2021-06-21
公開日2021-09-29
最終更新日2021-12-01
実験手法ELECTRON MICROSCOPY (4.2 Å)
主引用文献Kainate receptor modulation by NETO2.
Nature, 599, 2021
7F5B
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BU of 7f5b by Molmil
LBD-TMD focused reconstruction of DNQX-bound GluK2-1xNeto2 complex
分子名称: (1S)-2-{[{[(2R)-2,3-DIHYDROXYPROPYL]OXY}(HYDROXY)PHOSPHORYL]OXY}-1-[(PALMITOYLOXY)METHYL]ETHYL STEARATE, 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者He, L.L, Gao, Y.W, Li, B, Zhao, Y.
登録日2021-06-21
公開日2021-09-29
最終更新日2021-12-01
実験手法ELECTRON MICROSCOPY (3.9 Å)
主引用文献Kainate receptor modulation by NETO2.
Nature, 599, 2021

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件を2024-06-12に公開中

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