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2QR8
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2.0A X-ray structure of C-terminal kinase domain of p90 ribosomal S6 kinase 2 (RSK2)
分子名称: Ribosomal protein S6 kinase alpha-3, SODIUM ION
著者Tereshko, V, Malakhova, M, Dong, Z.
登録日2007-07-27
公開日2007-12-11
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural basis for activation of the autoinhibitory C-terminal kinase domain of p90 RSK2.
Nat.Struct.Mol.Biol., 15, 2008
2QR9
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Crystal Structure of the Estrogen Receptor Alpha Ligand Binding Domain Complexed with an Oxabicyclic Derivative Compound
分子名称: Estrogen receptor, Nuclear receptor coactivator 2, dimethyl (1R,4S)-5,6-bis(4-hydroxyphenyl)-7-oxabicyclo[2.2.1]hepta-2,5-diene-2,3-dicarboxylate
著者Nettles, K.W, Bruning, J.B.
登録日2007-07-27
公開日2008-03-18
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献NFkappaB selectivity of estrogen receptor ligands revealed by comparative crystallographic analyses
Nat.Chem.Biol., 4, 2008
2QRA
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Crystal structure of XIAP BIR1 domain (P21 form)
分子名称: Baculoviral IAP repeat-containing protein 4, ETHANOL, ZINC ION
著者Lin, S.-C.
登録日2007-07-27
公開日2007-09-18
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of the BIR1 domain of XIAP in two crystal forms
J.Mol.Biol., 372, 2007
2QRB
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Crystal structure of chloride saturated bovine lactoperoxidase at 2.5 A resolution shows multiple halide binding sites
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, CHLORIDE ION, ...
著者Singh, A.K, Singh, N, Sharma, S, Kaur, P, Singh, T.P.
登録日2007-07-28
公開日2007-08-14
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of chloride saturated bovine lactoperoxidase at 2.5 A resolution shows multiple halide binding sites
To be Published
2QRC
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Crystal structure of the adenylate sensor from AMP-activated protein kinase in complex with ADP and AMP
分子名称: ADENOSINE MONOPHOSPHATE, ADENOSINE-5'-DIPHOSPHATE, Protein C1556.08c, ...
著者Jin, X, Townley, R, Shapiro, L.
登録日2007-07-28
公開日2007-10-23
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structural Insight into AMPK Regulation: ADP Comes into Play.
Structure, 15, 2007
2QRD
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Crystal Structure of the Adenylate Sensor from AMP-activated Protein Kinase in complex with ADP and ATP
分子名称: ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, Protein C1556.08c, ...
著者Jin, X, Townley, R, Shapiro, L.
登録日2007-07-28
公開日2007-10-23
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.41 Å)
主引用文献Structural Insight into AMPK Regulation: ADP Comes into Play.
Structure, 15, 2007
2QRE
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Crystal structure of the adenylate sensor from AMP-activated protein kinase in complex with 5-aminoimidazole-4-carboxamide 1-beta-D-ribofuranotide (ZMP)
分子名称: AMINOIMIDAZOLE 4-CARBOXAMIDE RIBONUCLEOTIDE, Protein C1556.08c, SNF1-like protein kinase ssp2, ...
著者Jin, X, Townley, R, Shapiro, L.
登録日2007-07-28
公開日2007-10-23
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (3.01 Å)
主引用文献Structural Insight into AMPK Regulation: ADP Comes into Play.
Structure, 15, 2007
2QRF
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Green Fluorescent Protein: Cyclized-only Intermediate of Chromophore Maturation in the Q183E variant
分子名称: 1,2-ETHANEDIOL, Green fluorescent protein, MAGNESIUM ION
著者Wood, T.I, Barondeau, D.P, Hitomi, C, Tainer, J.A, Getzoff, E.D.
登録日2007-07-28
公開日2009-04-21
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Green Fluorescent Protein Chromophore - Cyclized Intermediate
To be Published
2QRG
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Glycogen Phosphorylase b in complex with (1R)-3'-(4-methoxyphenyl)-spiro[1,5-anhydro-D-glucitol-1,5'-isoxazoline]
分子名称: (5R,7R,8S,9S,10R)-7-(HYDROXYMETHYL)-3-(4-METHOXYPHENYL)-1,6-DIOXA-2-AZASPIRO[4.5]DEC-2-ENE-8,9,10-TRIOL, Glycogen phosphorylase, muscle form
著者Kizilis, G, Alexacou, K.-M, Chrysina, E.D, Zographos, S.E, Leonidas, D.D, Oikonomakos, N.G.
登録日2007-07-28
公開日2008-08-05
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Glucose-based spiro-isoxazolines: a new family of potent glycogen phosphorylase inhibitors.
Bioorg.Med.Chem., 17, 2009
2QRH
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Glycogen Phosphorylase b in complex with (1R)-3'-phenylspiro[1,5-anhydro-D-glucitol-1,5'-isoxazoline]
分子名称: (5R,7R,8S,9S,10R)-7-(hydroxymethyl)-3-phenyl-1,6-dioxa-2-azaspiro[4.5]dec-2-ene-8,9,10-triol, Glycogen phosphorylase, muscle form
著者Kizilis, G, Alexacou, K.-M, Chrysina, E.D, Zographos, S.E, Leonidas, D.D, Oikonomakos, N.G.
登録日2007-07-28
公開日2008-08-05
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.83 Å)
主引用文献Glucose-based spiro-isoxazolines: a new family of potent glycogen phosphorylase inhibitors.
Bioorg.Med.Chem., 17, 2009
2QRI
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Crystal structure of a single chain trimer composed of the MHC I heavy chain H-2Kb WT, beta-2microglobulin, and ovalbumin-derived peptide.
分子名称: H-2 class I histocompatibility antigen K-B alpha chain, Beta-2 microglobulin, ovalbumin-derived peptide
著者Mitaksov, V.E, Fremont, D.H.
登録日2007-07-28
公開日2007-11-06
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural engineering of pMHC reagents for T cell vaccines and diagnostics.
Chem.Biol., 14, 2007
2QRJ
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BU of 2qrj by Molmil
Crystal Structure of Sulfate-bound Saccharopine Dehydrogenase (L-Lys Forming) from Saccharomyces cerevisiae
分子名称: CHLORIDE ION, SULFATE ION, Saccharopine dehydrogenase, ...
著者Andi, B, Xu, H, Cook, P.F, West, A.H.
登録日2007-07-28
公開日2007-10-30
最終更新日2024-10-09
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Crystal Structures of Ligand-Bound Saccharopine Dehydrogenase from Saccharomyces cerevisiae
Biochemistry, 46, 2007
2QRK
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Crystal Structure of AMP-bound Saccharopine Dehydrogenase (L-Lys Forming) from Saccharomyces cerevisiae
分子名称: ADENOSINE MONOPHOSPHATE, Saccharopine dehydrogenase [NAD+, L-lysine-forming
著者Andi, B, Xu, H, Cook, P.F, West, A.H.
登録日2007-07-28
公開日2007-10-30
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Crystal Structures of Ligand-Bound Saccharopine Dehydrogenase from Saccharomyces cerevisiae
Biochemistry, 46, 2007
2QRL
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Crystal Structure of Oxalylglycine-bound Saccharopine Dehydrogenase (L-Lys Forming) from Saccharomyces cerevisiae
分子名称: N-OXALYLGLYCINE, Saccharopine dehydrogenase, NAD+, ...
著者Andi, B, Xu, H, Cook, P.F, West, A.H.
登録日2007-07-28
公開日2007-10-30
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Crystal Structures of Ligand-Bound Saccharopine Dehydrogenase from Saccharomyces cerevisiae
Biochemistry, 46, 2007
2QRM
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Glycogen Phosphorylase b in complex with (1R)-3'-(4-nitrophenyl)-spiro[1,5-anhydro-D-glucitol-1,5'-isoxazoline]
分子名称: (3S,5R,7R,8S,9S,10R)-7-(hydroxymethyl)-3-(4-nitrophenyl)-1,6-dioxa-2-azaspiro[4.5]decane-8,9,10-triol, Glycogen phosphorylase, muscle form
著者Gizilis, G, Alexacou, K.M, Chrysina, E.D, Zographos, S.E, Leonidas, D.D, Oikonomakos, N.G.
登録日2007-07-28
公開日2008-07-29
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Glucose-based spiro-isoxazolines: a new family of potent glycogen phosphorylase inhibitors.
Bioorg.Med.Chem., 17, 2009
2QRN
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Human Deoxycytidine kinase dCMP, UDP, Mg ion product complex
分子名称: 2'-DEOXYCYTIDINE-5'-MONOPHOSPHATE, Deoxycytidine kinase, MAGNESIUM ION, ...
著者Ealick, S.E, Soriano, E.V.
登録日2007-07-28
公開日2007-12-11
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (3.4 Å)
主引用文献Structures of human deoxycytidine kinase product complexes.
Acta Crystallogr.,Sect.D, 63, 2007
2QRO
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Human Deoxycytidine kinase dAMP, UDP, Mg ion product complex
分子名称: 2'-DEOXYADENOSINE-5'-MONOPHOSPHATE, Deoxycytidine kinase, MAGNESIUM ION, ...
著者Ealick, S.E, Soriano, E.V.
登録日2007-07-28
公開日2007-12-11
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (3.45 Å)
主引用文献Structures of human deoxycytidine kinase product complexes.
Acta Crystallogr.,Sect.D, 63, 2007
2QRP
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Glycogen Phosphorylase b in complex with (1R)-3'-(2-naphthyl)-spiro[1,5-anhydro-D-glucitol-1,5'-isoxazoline]
分子名称: (3S,5R,7R,8S,9S,10R)-7-(hydroxymethyl)-3-(2-naphthyl)-1,6-dioxa-2-azaspiro[4.5]decane-8,9,10-triol, DIMETHYL SULFOXIDE, Glycogen phosphorylase, ...
著者Gizilis, G, Alexacou, K.M, Chrysina, E.D, Zographos, S.E, Leonidas, D.D, Oikonomakos, N.G.
登録日2007-07-28
公開日2008-07-29
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献Glucose-based spiro-isoxazolines: a new family of potent glycogen phosphorylase inhibitors.
Bioorg.Med.Chem., 17, 2009
2QRQ
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Glycogen Phosphorylase b in complex with (1R)-3'-(4-methylphenyl)-spiro[1,5-anhydro-D-glucitol-1,5'-isoxazoline]
分子名称: (3S,5R,7R,8S,9S,10R)-7-(hydroxymethyl)-3-(4-methylphenyl)-1,6-dioxa-2-azaspiro[4.5]decane-8,9,10-triol, DIMETHYL SULFOXIDE, Glycogen phosphorylase, ...
著者Gizilis, G, Alexacou, K.M, Chrysina, E.D, Zographos, S.E, Leonidas, D.D, Oikonomakos, N.G.
登録日2007-07-28
公開日2008-07-29
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Glucose-based spiro-isoxazolines: a new family of potent glycogen phosphorylase inhibitors.
Bioorg.Med.Chem., 17, 2009
2QRR
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Crystal structure of the soluble domain of the ABC transporter, ATP-binding protein from Vibrio parahaemolyticus
分子名称: CHLORIDE ION, Methionine import ATP-binding protein metN
著者Kim, Y, Zhou, M, Freeman, L, Joachimiak, A, Midwest Center for Structural Genomics (MCSG)
登録日2007-07-28
公開日2007-08-14
最終更新日2017-10-25
実験手法X-RAY DIFFRACTION (1.71 Å)
主引用文献The Soluble Domain of the ABC Transporter, ATP-binding Protein from Vibrio parahaemolyticus.
To be Published
2QRS
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Crystal Structure of a single chain trimer composed of the MHC I heavy chain H-2Kb Y84A, beta-2microglobulin, and ovalbumin-derived peptide.
分子名称: H-2 class I histocompatibility antigen K-B alpha chain, Beta-2 microglobulin, ovalbumin-derived peptide
著者Mitaksov, V.E, Fremont, D.H.
登録日2007-07-29
公開日2007-11-06
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural engineering of pMHC reagents for T cell vaccines and diagnostics.
Chem.Biol., 14, 2007
2QRT
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Crystal Structure of a disulfide trapped single chain trimer composed of the MHC I heavy chain H-2Kb Y84C, beta-2microglobulin, and ovalbumin-derived peptide.
分子名称: H-2 class I histocompatibility antigen K-B alpha chain, Beta-2 microglobulin, ovalbumin-derived peptide
著者Mitaksov, V.E, Fremont, D.H.
登録日2007-07-29
公開日2007-11-06
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural engineering of pMHC reagents for T cell vaccines and diagnostics.
Chem.Biol., 14, 2007
2QRU
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Crystal structure of an alpha/beta hydrolase superfamily protein from Enterococcus faecalis
分子名称: 1,2-ETHANEDIOL, PHOSPHATE ION, Uncharacterized protein
著者Cuff, M.E, Volkart, L, Moy, S, Joachimiak, A, Midwest Center for Structural Genomics (MCSG)
登録日2007-07-29
公開日2007-09-11
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Structure of an alpha/beta hydrolase superfamily protein from Enterococcus faecalis.
TO BE PUBLISHED
2QRV
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Structure of Dnmt3a-Dnmt3L C-terminal domain complex
分子名称: DNA (cytosine-5)-methyltransferase 3-like, DNA (cytosine-5)-methyltransferase 3A, S-ADENOSYL-L-HOMOCYSTEINE
著者Jia, D, Cheng, X.
登録日2007-07-29
公開日2007-12-04
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.89 Å)
主引用文献Structure of Dnmt3a bound to Dnmt3L suggests a model for de novo DNA methylation.
Nature, 449, 2007
2QRW
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Crystal structure of Mycobacterium tuberculosis trHbO WG8F mutant
分子名称: CYANIDE ION, Hemoglobin-like protein HbO, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Milani, M, Bolognesi, M.
登録日2007-07-30
公開日2007-11-06
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献The Roles of Tyr(CD1) and Trp(G8) in Mycobacterium tuberculosis Truncated Hemoglobin O in Ligand Binding and on the Heme Distal Site Architecture
Biochemistry, 46, 2007

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