2QO3
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![BU of 2qo3 by Molmil](/molmil-images/mine/2qo3) | Crystal Structure of [KS3][AT3] didomain from module 3 of 6-deoxyerthronolide B synthase | 分子名称: | (2S, 3R)-3-HYDROXY-4-OXO-7,10-TRANS,TRANS-DODECADIENAMIDE, ACETATE ION, ... | 著者 | Khosla, C, Cane, E.D, Tang, Y, Chen, Y.A, Kim, C.Y. | 登録日 | 2007-07-19 | 公開日 | 2007-09-04 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.59 Å) | 主引用文献 | Structural and mechanistic analysis of protein interactions in module 3 of the 6-deoxyerythronolide B synthase Chem.Biol., 14, 2007
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4IMO
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![BU of 4imo by Molmil](/molmil-images/mine/4imo) | Crystal structure of wild type human Lipocalin PGDS in complex with substrate analog U44069 | 分子名称: | (5E)-7-{(1R,4S,5S,6R)-5-[(1E,3S)-3-hydroxyoct-1-en-1-yl]-2-oxabicyclo[2.2.1]hept-6-yl}hept-5-enoic acid, Lipocalin-type prostaglandin-D synthase, THIOCYANATE ION | 著者 | Lim, S.M, Chen, D, Teo, H, Roos, A, Nyman, T, Tresaugues, L, Pervushin, K, Nordlund, P. | 登録日 | 2013-01-03 | 公開日 | 2013-03-20 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.88 Å) | 主引用文献 | Structural and dynamic insights into substrate binding and catalysis of human lipocalin prostaglandin D synthase. J.Lipid Res., 54, 2013
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7DRK
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![BU of 7drk by Molmil](/molmil-images/mine/7drk) | Crystal structure of phosphatidylglycerol phosphate synthase in complex with cytidine diphosphate-diacylglycerol | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 1,4-BUTANEDIOL, 5'-O-[(R)-{[(S)-{(2R)-2,3-bis[(9E)-octadec-9-enoyloxy]propoxy}(hydroxy)phosphoryl]oxy}(hydroxy)phosphoryl]cytidine, ... | 著者 | Yang, B.W, Liu, Z.F. | 登録日 | 2020-12-28 | 公開日 | 2021-12-08 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | The phosphatidylglycerol phosphate synthase PgsA utilizes a trifurcated amphipathic cavity for catalysis at the membrane-cytosol interface. Curr Res Struct Biol, 3, 2021
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7DRJ
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![BU of 7drj by Molmil](/molmil-images/mine/7drj) | Crystal structure of phosphatidylglycerol phosphate synthase in complex with phosphatidylglycerol phosphate | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 1,4-BUTANEDIOL, ACETIC ACID, ... | 著者 | Yang, B.W, Liu, Z.F. | 登録日 | 2020-12-28 | 公開日 | 2021-12-08 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | The phosphatidylglycerol phosphate synthase PgsA utilizes a trifurcated amphipathic cavity for catalysis at the membrane-cytosol interface. Curr Res Struct Biol, 3, 2021
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8GHD
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![BU of 8ghd by Molmil](/molmil-images/mine/8ghd) | The structure of h12-LOX in hexameric form bound to inhibitor ML355 and arachidonic acid | 分子名称: | ARACHIDONIC ACID, FE (II) ION, N-(1,3-benzothiazol-2-yl)-4-{[(2-hydroxy-3-methoxyphenyl)methyl]amino}benzene-1-sulfonamide, ... | 著者 | Black, K.A, Mobbs, J.I, Venugopal, H, Thal, D.M, Glukhova, A. | 登録日 | 2023-03-09 | 公開日 | 2023-08-09 | 最終更新日 | 2023-10-11 | 実験手法 | ELECTRON MICROSCOPY (2.2 Å) | 主引用文献 | Cryo-EM structures of human arachidonate 12S-lipoxygenase bound to endogenous and exogenous inhibitors. Blood, 142, 2023
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4QAV
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3ILS
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![BU of 3ils by Molmil](/molmil-images/mine/3ils) | The Thioesterase Domain from PksA | 分子名称: | Aflatoxin biosynthesis polyketide synthase | 著者 | Korman, T.P. | 登録日 | 2009-08-07 | 公開日 | 2010-04-07 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structure and function of an iterative polyketide synthase thioesterase domain catalyzing Claisen cyclization in aflatoxin biosynthesis. Proc.Natl.Acad.Sci.USA, 107, 2010
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2GYO
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![BU of 2gyo by Molmil](/molmil-images/mine/2gyo) | Methanethiol-Cys 112 Inhibition Complex of E. Coli Ketoacyl Synthase III (FabH) and Coenzyme A | 分子名称: | 3-oxoacyl-[acyl-carrier-protein] synthase 3, COENZYME A, METHANETHIOL, ... | 著者 | Alhamadsheh, M.M, Musayev, F, Komissarov, A.A, Sachdeva, S, Wright, H.T, Scarsdale, N, Florova, G, Reynolds, K.A. | 登録日 | 2006-05-09 | 公開日 | 2007-06-05 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Alkyl-CoA Disulfides as Inhibitors and Mechanistic Probes for FabH Enzymes. Chem.Biol., 14, 2007
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3LED
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![BU of 3led by Molmil](/molmil-images/mine/3led) | Crystal structure of 3-oxoacyl-(acyl carrier protein) synthase III from Rhodopseudomonas palustris CGA009 | 分子名称: | 3-oxoacyl-acyl carrier protein synthase III, FORMIC ACID | 著者 | Chang, C, Xu, X, Cui, H, Savchenko, A, Edwards, A, Joachimiak, A, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2010-01-14 | 公開日 | 2010-01-26 | 最終更新日 | 2017-11-01 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Crystal structure of 3-oxoacyl-(acyl carrier protein) synthase III from Rhodopseudomonas palustris CGA009 To be Published
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7RIG
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![BU of 7rig by Molmil](/molmil-images/mine/7rig) | Structure of ACLY-D1026A-substrates | 分子名称: | (3S)-citryl-Coenzyme A, ADENOSINE-5'-DIPHOSPHATE, ATP-citrate synthase, ... | 著者 | Wei, X, Marmorstein, R. | 登録日 | 2021-07-19 | 公開日 | 2023-05-10 | 最終更新日 | 2024-06-05 | 実験手法 | ELECTRON MICROSCOPY (2.2 Å) | 主引用文献 | Allosteric role of the citrate synthase homology domain of ATP citrate lyase. Nat Commun, 14, 2023
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7RKZ
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7RMP
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![BU of 7rmp by Molmil](/molmil-images/mine/7rmp) | Structure of ACLY D1026A - substrates-asym | 分子名称: | (3S)-citryl-Coenzyme A, ADENOSINE-5'-DIPHOSPHATE, ATP-citrate synthase, ... | 著者 | Wei, X, Marmorstein, R. | 登録日 | 2021-07-28 | 公開日 | 2023-05-10 | 最終更新日 | 2024-06-05 | 実験手法 | ELECTRON MICROSCOPY (2.7 Å) | 主引用文献 | Allosteric role of the citrate synthase homology domain of ATP citrate lyase. Nat Commun, 14, 2023
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6R7D
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![BU of 6r7d by Molmil](/molmil-images/mine/6r7d) | Crystal structure of LTC4S in complex with AZ13690257 | 分子名称: | (1~{S},2~{S})-2-[5-[cyclopropylmethyl(naphthalen-1-yl)amino]-4-methoxy-pyrimidin-2-yl]carbonylcyclopropane-1-carboxylic acid, DODECYL-BETA-D-MALTOSIDE, Leukotriene C4 synthase, ... | 著者 | Kack, H, Ek, M. | 登録日 | 2019-03-28 | 公開日 | 2019-08-28 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Discovery of the Oral Leukotriene C4 Synthase Inhibitor (1S,2S)-2-({5-[(5-Chloro-2,4-difluorophenyl)(2-fluoro-2-methylpropyl)amino]-3-methoxypyrazin-2-yl}carbonyl)cyclopropanecarboxylic Acid (AZD9898) as a New Treatment for Asthma. J.Med.Chem., 62, 2019
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6QCL
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8G1F
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![BU of 8g1f by Molmil](/molmil-images/mine/8g1f) | Structure of ACLY-D1026A-products | 分子名称: | (3S)-citryl-Coenzyme A, ACETYL COENZYME *A, ADENOSINE-5'-DIPHOSPHATE, ... | 著者 | Wei, X, Marmorstein, R. | 登録日 | 2023-02-02 | 公開日 | 2023-05-10 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (2.4 Å) | 主引用文献 | Allosteric role of the citrate synthase homology domain of ATP citrate lyase. Nat Commun, 14, 2023
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8G5C
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8G5D
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8G1E
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![BU of 8g1e by Molmil](/molmil-images/mine/8g1e) | Structure of ACLY-D1026A-products-asym | 分子名称: | (3S)-citryl-Coenzyme A, ACETYL COENZYME *A, ADENOSINE-5'-DIPHOSPHATE, ... | 著者 | Wei, X, Marmorstein, R. | 登録日 | 2023-02-02 | 公開日 | 2023-05-10 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (2.8 Å) | 主引用文献 | Allosteric role of the citrate synthase homology domain of ATP citrate lyase. Nat Commun, 14, 2023
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4AMN
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5FM0
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![BU of 5fm0 by Molmil](/molmil-images/mine/5fm0) | Crystal structure of the 6-carboxyhexanoate-CoA ligase (BioW)from Bacillus subtilis (PtCl4 derivative) | 分子名称: | 6-CARBOXYHEXANOATE--COA LIGASE, MAGNESIUM ION, PIMELOYL-AMP, ... | 著者 | Moynie, L, Wang, M, Campopiano, D.J, Naismith, J.H. | 登録日 | 2015-10-29 | 公開日 | 2016-11-16 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.44 Å) | 主引用文献 | Using the pimeloyl-CoA synthetase adenylation fold to synthesize fatty acid thioesters. Nat. Chem. Biol., 13, 2017
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2QC3
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![BU of 2qc3 by Molmil](/molmil-images/mine/2qc3) | Crystal structure of MCAT from Mycobacterium tuberculosis | 分子名称: | ACETIC ACID, Malonyl CoA-acyl carrier protein transacylase | 著者 | Li, Z, Huang, Y, Ge, J, Bartlam, M, Wang, H, Rao, Z. | 登録日 | 2007-06-19 | 公開日 | 2007-08-28 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | The Crystal Structure of MCAT from Mycobacterium tuberculosis Reveals Three New Catalytic Models. J.Mol.Biol., 371, 2007
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7F27
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![BU of 7f27 by Molmil](/molmil-images/mine/7f27) | Crystal structure of polyketide ketosynthase | 分子名称: | 3-oxoacyl-(Acyl-carrier-protein) synthase | 著者 | Kim, Y, Lee, W.C. | 登録日 | 2021-06-10 | 公開日 | 2022-06-15 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.806 Å) | 主引用文献 | Structural basis of the complementary activity of two ketosynthases in aryl polyene biosynthesis. Sci Rep, 11, 2021
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7F28
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![BU of 7f28 by Molmil](/molmil-images/mine/7f28) | Crystal structure of a bacterial ketosynthase | 分子名称: | Ketoacyl_synth_N domain-containing protein, Putative 3-oxoacyl-[ACP] synthase FabV | 著者 | Lee, W.C, Kim, Y. | 登録日 | 2021-06-10 | 公開日 | 2022-06-15 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.877 Å) | 主引用文献 | Structural basis of the complementary activity of two ketosynthases in aryl polyene biosynthesis. Sci Rep, 11, 2021
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4AMM
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4AMP
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![BU of 4amp by Molmil](/molmil-images/mine/4amp) | |