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5SY1
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Structure of the STRA6 receptor for retinol uptake in complex with calmodulin
分子名称: CALCIUM ION, CHOLESTEROL, Calmodulin, ...
著者Clarke, O.B, Chen, Y, Mancia, F.
登録日2016-08-10
公開日2016-08-24
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.9 Å)
主引用文献Structure of the STRA6 receptor for retinol uptake.
Science, 353, 2016
1SK6
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Crystal structure of the adenylyl cyclase domain of anthrax edema factor (EF) in complex with calmodulin, 3',5' cyclic AMP (cAMP), and pyrophosphate
分子名称: ADENOSINE-3',5'-CYCLIC-MONOPHOSPHATE, CALCIUM ION, Calmodulin, ...
著者Guo, Q, Shen, Y, Zhukovskaya, N.L, Tang, W.J.
登録日2004-03-04
公開日2004-06-08
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structural and kinetic analyses of the interaction of anthrax adenylyl cyclase toxin with reaction products cAMP and pyrophosphate.
J.Biol.Chem., 279, 2004
1PK0
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Crystal Structure of the EF3-CaM complexed with PMEApp
分子名称: (ADENIN-9-YL-ETHOXYMETHYL)-HYDROXYPHOSPHINYL-DIPHOSPHATE, CALCIUM ION, Calmodulin, ...
著者Shen, Y, Tang, W.J.
登録日2003-06-04
公開日2004-02-10
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Selective inhibition of anthrax edema factor by adefovir, a drug for chronic hepatitis B virus infection.
Proc.Natl.Acad.Sci.USA, 101, 2004
4N5X
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Crystal structure of N-terminal calmodulin-like Calcium sensor of human mitochondrial ATP-Mg/Pi carrier SCaMC1
分子名称: CALCIUM ION, Calcium-binding mitochondrial carrier protein SCaMC-1, DI(HYDROXYETHYL)ETHER
著者Yang, Q, Bruschweiler, S, Chou, J.
登録日2013-10-10
公開日2013-12-18
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献A Self-Sequestered Calmodulin-like Ca(2+) Sensor of Mitochondrial SCaMC Carrier and Its Implication to Ca(2+)-Dependent ATP-Mg/Pi Transport.
Structure, 22, 2014
4JQ0
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Voltage-gated sodium channel 1.5 C-terminal domain in complex with FGF12B and Ca2+/calmodulin
分子名称: CALCIUM ION, Calmodulin, Fibroblast growth factor 12, ...
著者Wang, C, Chung, B.C, Yan, H, Wang, H.G, Lee, S.Y, Pitt, G.S.
登録日2013-03-19
公開日2014-05-21
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.84 Å)
主引用文献Structural analyses of Ca(2+)/CaM interaction with NaV channel C-termini reveal mechanisms of calcium-dependent regulation.
Nat Commun, 5, 2014
4JPZ
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Voltage-gated sodium channel 1.2 C-terminal domain in complex with FGF13U and Ca2+/calmodulin
分子名称: CALCIUM ION, Calmodulin, Fibroblast growth factor 13, ...
著者Wang, C, Chung, B.C, Yan, H, Wang, H.G, Lee, S.Y, Pitt, G.S.
登録日2013-03-19
公開日2014-04-16
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.02 Å)
主引用文献Structural analyses of Ca(2+)/CaM interaction with NaV channel C-termini reveal mechanisms of calcium-dependent regulation.
Nat Commun, 5, 2014
3OX5
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BU of 3ox5 by Molmil
Crystal Structure of the calcium sensor calcium-binding protein 1 (CaBP1)
分子名称: CALCIUM ION, Calcium-binding protein 1
著者Findeisen, F, Minor, D.L.
登録日2010-09-21
公開日2010-12-22
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structural Basis for the Differential Effects of CaBP1 and Calmodulin on Ca(V)1.2 Calcium-Dependent Inactivation.
Structure, 18, 2010
6OF9
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Structure of the Chlamydamonas reinhardtii CamKII hub homology domain
分子名称: CaMKII hub
著者McSpadden, E.D, Chi, C.C, Gee, C.L, Kuriyan, J.
登録日2019-03-28
公開日2019-04-17
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Variation in assembly stoichiometry in non-metazoan homologs of the hub domain of Ca2+/calmodulin-dependent protein kinase II.
Protein Sci., 28, 2019
3OX6
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Crystal Structure of the calcium sensor calcium-binding protein 1 (CaBP1)
分子名称: CALCIUM ION, Calcium-binding protein 1, HEXANE-1,6-DIOL
著者Findeisen, F, Minor, D.L.
登録日2010-09-21
公開日2010-12-22
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural Basis for the Differential Effects of CaBP1 and Calmodulin on Ca(V)1.2 Calcium-Dependent Inactivation.
Structure, 18, 2010
6O20
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Cryo-EM structure of TRPV5 with calmodulin bound
分子名称: CALCIUM ION, Calmodulin, Transient receptor potential cation channel subfamily V member 5
著者Dang, S, van Goor, M.K, Asarnow, D, Wang, Y, Julius, D, Cheng, Y, van der Wijst, J.
登録日2019-02-22
公開日2019-04-24
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Structural insight into TRPV5 channel function and modulation.
Proc.Natl.Acad.Sci.USA, 116, 2019
3I6X
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Crystal structure of the calponin homology domain of IQGAP1
分子名称: Ras GTPase-activating-like protein IQGAP1
著者Kurella, V.B.
登録日2009-07-07
公開日2010-07-21
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The IQGAP1 N-Terminus Forms Dimers, and the Dimer Interface Is Required for Binding F-Actin and Calcium-Bound Calmodulin.
Biochemistry, 55, 2016
1TN4
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FOUR CALCIUM TNC
分子名称: CALCIUM ION, TROPONIN C
著者Love, M.L, Dominguez, R, Houdusse, A, Cohen, C.
登録日1997-09-18
公開日1998-04-08
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Structures of four Ca2+-bound troponin C at 2.0 A resolution: further insights into the Ca2+-switch in the calmodulin superfamily.
Structure, 5, 1997
6SZ5
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BU of 6sz5 by Molmil
Human calmodulin bound to a peptide of human NADPH oxidase 5
分子名称: CALCIUM ION, Calmodulin-2, NADPH oxidase 5
著者Millana, E, Mattevi, A.
登録日2019-10-02
公開日2019-12-11
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.23 Å)
主引用文献On the mechanism of calcium-dependent activation of NADPH oxidase 5 (NOX5).
Febs J., 287, 2020
1X02
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Solution structure of stereo array isotope labeled (SAIL) calmodulin
分子名称: CALCIUM ION, calmodulin
著者Kainosho, M, Torizawa, T, Terauchi, T, Ono, A.M, Guntert, P.
登録日2005-03-11
公開日2006-03-07
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Optimal isotope labelling for NMR protein structure determinations.
Nature, 440, 2006
6OQQ
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BU of 6oqq by Molmil
Legionella pneumophila SidJ/Saccharomyces cerevisiae calmodulin complex
分子名称: 1,2-ETHANEDIOL, ADENOSINE MONOPHOSPHATE, CALCIUM ION, ...
著者Tomchick, D.R, Tagliabracci, V.S, Black, M, Osinski, A.
登録日2019-04-28
公開日2019-05-15
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.102 Å)
主引用文献Bacterial pseudokinase catalyzes protein polyglutamylation to inhibit the SidE-family ubiquitin ligases.
Science, 364, 2019
5DBR
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BU of 5dbr by Molmil
Ca2+ CaM with human cardiac Na+ channel (NaV1.5) inactivation gate
分子名称: CALCIUM ION, Calmodulin, Sodium channel protein type 5 subunit alpha
著者Johnson, C.N, Thompson, M.K, Chazin, W.J.
登録日2015-08-21
公開日2017-02-22
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Enhanced Understanding of Ca2+ Modulation of the Human Cardiac Sodium Channel: Tight Binding of Calmodulin to the Inactivation Gate
To Be Published
7B16
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TRPC4 in complex with inhibitor GFB-9289
分子名称: 2-(HEXADECANOYLOXY)-1-[(PHOSPHONOOXY)METHYL]ETHYL HEXADECANOATE, 5-chloranyl-4-(4-cyclohexyl-3-oxidanylidene-piperazin-1-yl)-1~{H}-pyridazin-6-one, CALCIUM ION, ...
著者Vinayagam, D, Quentin, D, Sistel, O, Merino, F, Stabrin, M, Hofnagel, O, Ledeboer, M.W, Malojcic, G, Raunser, S.
登録日2020-11-23
公開日2020-12-09
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (3.15 Å)
主引用文献Structural basis of TRPC4 regulation by calmodulin and pharmacological agents.
Elife, 9, 2020
7B0S
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TRPC4 in complex with inhibitor GFB-8438
分子名称: (2R)-3-(phosphonooxy)propane-1,2-diyl dihexanoate, 5-chloranyl-4-[3-oxidanylidene-4-[[2-(trifluoromethyl)phenyl]methyl]piperazin-1-yl]-1~{H}-pyridazin-6-one, CALCIUM ION, ...
著者Vinayagam, D, Quentin, D, Sistel, O, Merino, F, Stabrin, M, Hofnagel, O, Ledeboer, M.W, Malojcic, G, Raunser, S.
登録日2020-11-21
公開日2020-12-09
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Structural basis of TRPC4 regulation by calmodulin and pharmacological agents.
Elife, 9, 2020
7B0J
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TRPC4 in LMNG detergent
分子名称: 2-(HEXADECANOYLOXY)-1-[(PHOSPHONOOXY)METHYL]ETHYL HEXADECANOATE, CALCIUM ION, Transient receptor potential cation channel subfamily c member 4a
著者Vinayagam, D, Quentin, D, Sistel, O, Merino, F, Stabrin, M, Hofnagel, O, Ledeboer, M.W, Malojcic, G, Raunser, S.
登録日2020-11-20
公開日2020-12-09
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (2.85 Å)
主引用文献Structural basis of TRPC4 regulation by calmodulin and pharmacological agents.
Elife, 9, 2020
7B05
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TRPC4 in complex with inhibitor GFB-8749
分子名称: (2R)-3-(phosphonooxy)propane-1,2-diyl dihexanoate, 4-[4-[[4,4-bis(fluoranyl)cyclohexyl]methyl]-3-oxidanylidene-piperazin-1-yl]-5-chloranyl-1~{H}-pyridazin-6-one, CALCIUM ION, ...
著者Vinayagam, D, Quentin, D, Sistel, O, Merino, F, Stabrin, M, Hofnagel, O, Ledeboer, M.W, Malojcic, G, Raunser, S.
登録日2020-11-18
公開日2020-12-09
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献Structural basis of TRPC4 regulation by calmodulin and pharmacological agents.
Elife, 9, 2020
2TN4
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FOUR CALCIUM TNC
分子名称: CALCIUM ION, TROPONIN C
著者Love, M.L, Dominguez, R, Houdusse, A, Cohen, C.
登録日1997-09-18
公開日1998-04-08
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structures of four Ca2+-bound troponin C at 2.0 A resolution: further insights into the Ca2+-switch in the calmodulin superfamily.
Structure, 5, 1997
2AAO
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BU of 2aao by Molmil
Regulatory apparatus of Calcium Dependent protein kinase from Arabidopsis thaliana
分子名称: CALCIUM ION, Calcium-dependent protein kinase, isoform AK1
著者Chandran, V, Stollar, E.J, Lindorff-Larsen, K, Harper, J.F, Chazin, W.J, Dobson, C.M, Luisi, B.F, Christodoulou, J.
登録日2005-07-13
公開日2005-12-27
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure of the regulatory apparatus of a calcium-dependent protein kinase (CDPK): a novel mode of calmodulin-target recognition.
J.Mol.Biol., 357, 2006
3HBX
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Crystal structure of GAD1 from Arabidopsis thaliana
分子名称: Glutamate decarboxylase 1
著者Gut, H, Dominici, P, Pilati, S, Gruetter, M.G, Capitani, G.
登録日2009-05-05
公開日2009-07-28
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.672 Å)
主引用文献A common structural basis for pH- and calmodulin-mediated regulation in plant glutamate decarboxylase.
J.Mol.Biol., 392, 2009
7OAJ
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Crystal structure of pseudokinase CASK in complex with compound 7
分子名称: 1,2-ETHANEDIOL, 4-(cyclopentylamino)-2-[(3,4-dichlorophenyl)methylamino]-N-[3-(2-oxidanylidenepyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide, Peripheral plasma membrane protein CASK
著者Chaikuad, A, Russ, N, Knapp, S, Structural Genomics Consortium (SGC)
登録日2021-04-19
公開日2021-05-19
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献Design and Development of a Chemical Probe for Pseudokinase Ca 2+ /calmodulin-Dependent Ser/Thr Kinase.
J.Med.Chem., 64, 2021
7OAI
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Crystal structure of pseudokinase CASK in complex with PFE-PKIS12
分子名称: 1,2-ETHANEDIOL, 4-(Cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-N-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide, Peripheral plasma membrane protein CASK
著者Chaikuad, A, Knapp, S, Structural Genomics Consortium (SGC)
登録日2021-04-19
公開日2021-05-19
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Design and Development of a Chemical Probe for Pseudokinase Ca 2+ /calmodulin-Dependent Ser/Thr Kinase.
J.Med.Chem., 64, 2021

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