7OAI
Crystal structure of pseudokinase CASK in complex with PFE-PKIS12
Summary for 7OAI
Entry DOI | 10.2210/pdb7oai/pdb |
Descriptor | Peripheral plasma membrane protein CASK, 4-(Cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-N-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide, 1,2-ETHANEDIOL, ... (4 entities in total) |
Functional Keywords | pseudokinase, kinase, inhibitor, structural genomics, structural genomics consortium, sgc, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 4 |
Total formula weight | 161230.72 |
Authors | Chaikuad, A.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2021-04-19, release date: 2021-05-19, Last modification date: 2024-01-31) |
Primary citation | Russ, N.,Schroder, M.,Berger, B.T.,Mandel, S.,Aydogan, Y.,Mauer, S.,Pohl, C.,Drewry, D.H.,Chaikuad, A.,Muller, S.,Knapp, S. Design and Development of a Chemical Probe for Pseudokinase Ca 2+ /calmodulin-Dependent Ser/Thr Kinase. J.Med.Chem., 64:14358-14376, 2021 Cited by PubMed: 34543009DOI: 10.1021/acs.jmedchem.1c00845 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.3 Å) |
Structure validation
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