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5IVF
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Linked KDM5A Jmj Domain Bound to the Inhibitor N10 8-(1-methyl-1H-imidazol-4-yl)-2-(4,4,4-trifluorobutoxy)pyrido[3,4-d]pyrimidin-4-ol
分子名称: 8-(1-methyl-1H-imidazol-4-yl)-2-(4,4,4-trifluorobutoxy)pyrido[3,4-d]pyrimidin-4-ol, Lysine-specific demethylase 5A, MANGANESE (II) ION
著者Horton, J.R, Cheng, X.
登録日2016-03-20
公開日2016-07-27
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.683 Å)
主引用文献Structural Basis for KDM5A Histone Lysine Demethylase Inhibition by Diverse Compounds.
Cell Chem Biol, 23, 2016
5XS8
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Crystal structure of solute-binding protein complexed with unsaturated chondroitin disaccharide with two sulfate groups at C-4 and C-6 positions of GalNAc
分子名称: 4-deoxy-alpha-L-threo-hex-4-enopyranuronic acid-(1-3)-2-acetamido-2-deoxy-4,6-di-O-sulfo-beta-D-galactopyranose, CALCIUM ION, Extracellular solute-binding protein family 1
著者Oiki, S, Kamochi, R, Mikami, B, Murata, K, Hashimoto, W.
登録日2017-06-12
公開日2018-01-17
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.952 Å)
主引用文献Alternative substrate-bound conformation of bacterial solute-binding protein involved in the import of mammalian host glycosaminoglycans.
Sci Rep, 7, 2017
1BS5
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PEPTIDE DEFORMYLASE AS ZN2+ CONTAINING FORM
分子名称: PROTEIN (PEPTIDE DEFORMYLASE), SULFATE ION, ZINC ION
著者Becker, A, Schlichting, I, Kabsch, W, Groche, D, Schultz, S, Wagner, A.F.V.
登録日1998-09-01
公開日1999-08-27
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Iron center, substrate recognition and mechanism of peptide deformylase.
Nat.Struct.Biol., 5, 1998
1BSS
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ECORV-T93A/DNA/CA2+
分子名称: 5'-D(*AP*AP*AP*GP*AP*TP*AP*TP*CP*TP*T)-3', CALCIUM ION, ECORV ENDONUCLEASE
著者Perona, J.J, Horton, N.C.
登録日1998-08-30
公開日1998-09-02
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Metal ion-mediated substrate-assisted catalysis in type II restriction endonucleases
Proc.Natl.Acad.Sci.USA, 95, 1998
7A0K
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Crystal structure of the entire ectodomain from the Physcomitrella patens receptor kinase CR4
分子名称: 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Hothorn, M, Okuda, S.
登録日2020-08-09
公開日2021-08-18
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal structures of Arabidopsis and Physcomitrella CR4 reveal the molecular architecture of CRINKLY4 receptor kinases.
To Be Published
1BTX
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Episelection: Novel Ki ~Nanomolar Inhibitors of Serine Proteases Selected by Binding or Chemistry on an Enzyme Surface
分子名称: BETA-TRYPSIN, CALCIUM ION, N-(tert-butoxycarbonyl)-L-alanyl-N-[(1S)-5-amino-1-(diethoxyboranyl)pentyl]-L-valinamide
著者Stroud, R.M, Katz, B.A, Finer-Moore, J.
登録日1995-05-17
公開日1995-10-15
最終更新日2012-12-12
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Episelection: novel Ki approximately nanomolar inhibitors of serine proteases selected by binding or chemistry on an enzyme surface.
Biochemistry, 34, 1995
1BUA
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STRUCTURAL AND ENERGETIC ORIGINS OF INDIRECT READOUT IN SITE-SPECIFIC DNA CLEAVAGE BY A RESTRICTION ENDONUCLEASE
分子名称: DNA (5'-D(*AP*AP*AP*GP*AP*CP*IP*TP*CP*TP*T)-3'), ENDONUCLEASE ECORV
著者Perona, J.J, Martin, A.M.
登録日1998-09-03
公開日1998-09-09
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Structural and energetic origins of indirect readout in site-specific DNA cleavage by a restriction endonuclease.
Nat.Struct.Biol., 6, 1999
7AC7
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Structure of accomodated trans-translation complex on E. Coli stalled ribosome.
分子名称: 16S ribosomal RNA, 23S ribosomal RNA, 30S ribosomal protein S10, ...
著者Guyomar, C, D'Urso, G, Chat, S, Giudice, E, Gillet, R.
登録日2020-09-10
公開日2021-08-18
最終更新日2024-04-24
実験手法ELECTRON MICROSCOPY (3.08 Å)
主引用文献Structures of tmRNA and SmpB as they transit through the ribosome.
Nat Commun, 12, 2021
1BV4
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BU of 1bv4 by Molmil
APO-MANNOSE-BINDING PROTEIN-C
分子名称: PROTEIN (MANNOSE-BINDING PROTEIN-C)
著者Ng, K.K.-S, Weis, W.I.
登録日1998-09-22
公開日1999-01-13
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Ca2+-dependent structural changes in C-type mannose-binding proteins.
Biochemistry, 37, 1998
1BVO
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BU of 1bvo by Molmil
DORSAL HOMOLOGUE GAMBIF1 BOUND TO DNA
分子名称: DNA DUPLEX, TRANSCRIPTION FACTOR GAMBIF1
著者Cramer, P, Varrot, A, Barillas-Mury, C, Kafatos, F.C, Mueller, C.W.
登録日1998-09-16
公開日1999-07-12
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structure of the specificity domain of the Dorsal homologue Gambif1 bound to DNA.
Structure Fold.Des., 7, 1999
1BVV
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BU of 1bvv by Molmil
SUGAR RING DISTORTION IN THE GLYCOSYL-ENZYME INTERMEDIATE OF A FAMILY G/11 XYLANASE
分子名称: ENDO-1,4-BETA-XYLANASE, beta-D-xylopyranose-(1-4)-1,5-anhydro-2-deoxy-2-fluoro-D-xylitol
著者Sidhu, G, Brayer, G.D.
登録日1998-09-18
公開日1999-06-08
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Sugar ring distortion in the glycosyl-enzyme intermediate of a family G/11 xylanase.
Biochemistry, 38, 1999
7AE5
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BU of 7ae5 by Molmil
Structure of Sedimentibacter hydroxybenzoicus vanillic acid decarboxylase (ShVdcCD) in open form
分子名称: Phenolic acid decarboxylase, Protein ShdD, RUBIDIUM ION, ...
著者Marshall, S.A, Leys, D.
登録日2020-09-17
公開日2021-08-25
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.19 Å)
主引用文献Domain mobility and allosteric activation of UbiD decarboxylases
To Be Published
5EUJ
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BU of 5euj by Molmil
PYRUVATE DECARBOXYLASE FROM ZYMOBACTER PALMAE
分子名称: 1,2-ETHANEDIOL, MAGNESIUM ION, Pyruvate decarboxylase, ...
著者Buddrus, L, Crennell, S.J, Leak, D.J, Danson, M.J, Andrews, E.S.V, Arcus, V.L.
登録日2015-11-18
公開日2016-09-14
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Crystal structure of pyruvate decarboxylase from Zymobacter palmae.
Acta Crystallogr.,Sect.F, 72, 2016
5F38
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X-ray crystal structure of a thiolase from Escherichia coli at 1.8 A resolution
分子名称: 1,2-ETHANEDIOL, Acetyl-CoA acetyltransferase, COENZYME A, ...
著者Ithayaraja, M, Neelanjana, J, Wierenga, R, Savithri, H.S, Murthy, M.R.N.
登録日2015-12-02
公開日2016-07-13
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structure of a thiolase from Escherichia coli at 1.8 angstrom resolution.
Acta Crystallogr.,Sect.F, 72, 2016
1BWB
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HIV-1 PROTEASE (V82F/I84V) DOUBLE MUTANT COMPLEXED WITH SD146 OF DUPONT PHARMACEUTICALS
分子名称: PROTEIN (HIV-1 PROTEASE), [4R-(4ALPHA,5ALPHA,6ALPHA,7ALPHA)]-3,3'-{{TETRAHYDRO-5,6-DIHYDROXY-2-OXO-4,7-BIS(PHENYLMETHYL)-1H-1,3-DIAZEPINE-1,3(2H)-DIYL]BIS(METHYLENE)]BIS[N-1H-BENZIMIDAZOL-2-YLBENZAMIDE]
著者Ala, P, Chang, C.H.
登録日1998-09-22
公開日1998-09-30
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Counteracting HIV-1 protease drug resistance: structural analysis of mutant proteases complexed with XV638 and SD146, cyclic urea amides with broad specificities.
Biochemistry, 37, 1998
1BS8
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PEPTIDE DEFORMYLASE AS ZN2+ CONTAINING FORM IN COMPLEX WITH TRIPEPTIDE MET-ALA-SER
分子名称: PROTEIN (MET-ALA-SER), PROTEIN (PEPTIDE DEFORMYLASE), SULFATE ION, ...
著者Becker, A, Schlichting, I, Kabsch, W, Groche, D, Schultz, S, Wagner, A.F.V.
登録日1998-09-01
公開日1999-08-27
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Iron center, substrate recognition and mechanism of peptide deformylase.
Nat.Struct.Biol., 5, 1998
1BSO
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BU of 1bso by Molmil
12-BROMODODECANOIC ACID BINDS INSIDE THE CALYX OF BOVINE BETA-LACTOGLOBULIN
分子名称: 12-BROMODODECANOIC ACID, PROTEIN (BOVINE BETA-LACTOGLOBULIN A)
著者Qin, B.Y, Creamer, L.K, Baker, E.N, Jameson, G.B.
登録日1998-08-29
公開日1999-09-02
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.23 Å)
主引用文献12-Bromododecanoic acid binds inside the calyx of bovine beta-lactoglobulin.
FEBS Lett., 438, 1998
1BWI
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THE 1.8 A STRUCTURE OF MICROBATCH OIL DROP GROWN TETRAGONAL HEN EGG WHITE LYSOZYME
分子名称: PROTEIN (LYSOZYME)
著者Dong, J, Boggon, T.J, Chayen, N.E, Raftery, J, Bi, R.C.
登録日1998-09-24
公開日1998-09-30
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Bound-solvent structures for microgravity-, ground control-, gel- and microbatch-grown hen egg-white lysozyme crystals at 1.8 A resolution.
Acta Crystallogr.,Sect.D, 55, 1999
1BWK
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OLD YELLOW ENZYME (OYE1) MUTANT H191N
分子名称: FLAVIN MONONUCLEOTIDE, PROTEIN (NADPH DEHYDROGENASE 1)
著者Brown, B.J, Deng, Z, Karplus, P.A, Massey, V.
登録日1998-09-24
公開日1998-09-30
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献On the active site of Old Yellow Enzyme. Role of histidine 191 and asparagine 194.
J.Biol.Chem., 273, 1998
1BTJ
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HUMAN SERUM TRANSFERRIN, RECOMBINANT N-TERMINAL LOBE, APO FORM, CRYSTAL FORM 2
分子名称: PROTEIN (SERUM TRANSFERRIN)
著者Jeffrey, P.D, Bewley, M.C, Macgillivray, R.T.A, Mason, A.B, Woodworth, R.C, Baker, E.N.
登録日1998-09-01
公開日1999-01-13
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Ligand-induced conformational change in transferrins: crystal structure of the open form of the N-terminal half-molecule of human transferrin.
Biochemistry, 37, 1998
1BWZ
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DIAMINOPIMELATE EPIMERASE FROM HEMOPHILUS INFLUENZAE
分子名称: PROTEIN (DIAMINOPIMELATE EPIMERASE)
著者Cirilli, M, Zheng, R, Scapin, G, Blanchard, J.S.
登録日1998-09-29
公開日1998-12-16
最終更新日2017-10-04
実験手法X-RAY DIFFRACTION (2.72 Å)
主引用文献Structural symmetry: the three-dimensional structure of Haemophilus influenzae diaminopimelate epimerase.
Biochemistry, 37, 1998
5EZM
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Crystal Structure of ArnT from Cupriavidus metallidurans in the apo state
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, 4-amino-4-deoxy-L-arabinose transferase or related glycosyltransferases of PMT family, CHLORIDE ION, ...
著者Petrou, V.I, Clarke, O.B, Tomasek, D, Banerjee, S, Rajashankar, K.R, Mancia, F, New York Consortium on Membrane Protein Structure (NYCOMPS)
登録日2015-11-26
公開日2016-02-17
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structures of aminoarabinose transferase ArnT suggest a molecular basis for lipid A glycosylation.
Science, 351, 2016
1BU8
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RAT PANCREATIC LIPASE RELATED PROTEIN 2
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, PROTEIN (PANCREATIC LIPASE RELATED PROTEIN 2)
著者Roussel, A, Cambillau, C.
登録日1998-09-14
公開日1998-12-23
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structure and activity of rat pancreatic lipase-related protein 2.
J.Biol.Chem., 273, 1998
1BXT
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STREPTOCOCCAL SUPERANTIGEN (SSA) FROM STREPTOCOCCUS PYOGENES
分子名称: PROTEIN (STREPTOCOCCAL SUPERANTIGEN)
著者Sundberg, E, Jardetzky, T.
登録日1998-10-08
公開日1998-10-14
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Structural basis for HLA-DQ binding by the streptococcal superantigen SSA.
Nat.Struct.Biol., 6, 1999
1BUL
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6ALPHA-(HYDROXYPROPYL)PENICILLANATE ACYLATED ON NMC-A BETA-LACTAMASE FROM ENTEROBACTER CLOACAE
分子名称: 2-(1-CARBOXY-2-HYDROXY-2-METHYL-PROPYL)-5,5-DIMETHYL-THIAZOLIDINE-4-CARBOXYLIC ACID, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, NMC-A BETA-LACTAMASE
著者Mourey, L, Swaren, P, Miyashita, K, Bulychev, A, Mobashery, S, Samama, J.P.
登録日1998-09-04
公開日1998-12-30
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.89 Å)
主引用文献Inhibition of the Nmc-A B-Lactamase by a Penicillanic Acid Derivative, and the Structural Bases for the Increase in Substrate Profile of This Antibiotic Resistance Enzyme
J.Am.Chem.Soc., 120, 1998

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