8Y8Z
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![BU of 8y8z by Molmil](/molmil-images/mine/8y8z) | Structure of NET-Maprotiline in outward-open state | 分子名称: | CHLORIDE ION, SODIUM ION, Sodium-dependent noradrenaline transporter, ... | 著者 | Zhang, H, Xu, E.H, Jiang, Y. | 登録日 | 2024-02-06 | 公開日 | 2024-05-29 | 最終更新日 | 2024-07-03 | 実験手法 | ELECTRON MICROSCOPY (3.29 Å) | 主引用文献 | Dimerization and antidepressant recognition at noradrenaline transporter. Nature, 630, 2024
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8Y8Y
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![BU of 8y8y by Molmil](/molmil-images/mine/8y8y) | Crystal structure of the PTPN21 FERM domain | 分子名称: | CHLORIDE ION, Tyrosine-protein phosphatase non-receptor type 21 | 著者 | Lee, H.S, Ku, B. | 登録日 | 2024-02-06 | 公開日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (2.099 Å) | 主引用文献 | Structural analysis of the FERM domain of human protein tyrosine phosphatase non-receptor type 21. Acta Crystallogr.,Sect.F, 80, 2024
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8Y6P
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8Y6I
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![BU of 8y6i by Molmil](/molmil-images/mine/8y6i) | P-glycoprotein in complex with UIC2 Fab and triple elacridar molecules in nanodisc | 分子名称: | 1,2-Distearoyl-sn-glycerophosphoethanolamine, ATP-dependent translocase ABCB1,mNeonGreen, CHOLESTEROL, ... | 著者 | Hamaguchi-Suzuki, N, Adachi, N, Moriya, T, Kawasaki, M, Suzuki, K, Anzai, N, Senda, T, Murata, T. | 登録日 | 2024-02-02 | 公開日 | 2024-04-17 | 実験手法 | ELECTRON MICROSCOPY (2.54 Å) | 主引用文献 | Cryo-EM structure of P-glycoprotein bound to triple elacridar inhibitor molecules. Biochem.Biophys.Res.Commun., 709, 2024
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8Y6H
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![BU of 8y6h by Molmil](/molmil-images/mine/8y6h) | P-glycoprotein in complex with UIC2 Fab and triple elacridar molecules in LMNG detergent | 分子名称: | ATP-dependent translocase ABCB1,mNeonGreen, UIC2 Fab heavy chain, UIC2 Fab light chain, ... | 著者 | Hamaguchi-Suzuki, N, Adachi, N, Moriya, T, Kawasaki, M, Suzuki, K, Anzai, N, Senda, T, Murata, T. | 登録日 | 2024-02-02 | 公開日 | 2024-04-17 | 実験手法 | ELECTRON MICROSCOPY (2.49 Å) | 主引用文献 | Cryo-EM structure of P-glycoprotein bound to triple elacridar inhibitor molecules. Biochem.Biophys.Res.Commun., 709, 2024
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8Y6D
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![BU of 8y6d by Molmil](/molmil-images/mine/8y6d) | Norovirus GII.10 P domain and 2'-FL (tablet) | 分子名称: | 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, GII.10 norovirus P domain in complex with 2'-FL (tablet), ... | 著者 | Hansman, G, Tame, J.R.H, Kher, G, Pancera, M. | 登録日 | 2024-02-02 | 公開日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (1.41 Å) | 主引用文献 | Norovirus GII.10 P domain and 2'-FL (tablet) To Be Published
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8Y6C
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![BU of 8y6c by Molmil](/molmil-images/mine/8y6c) | Norovirus GII.10 P domain and 2'-FL (powder) | 分子名称: | 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, GII.10 norovirus P domain in complex with 2'FL (powder), ... | 著者 | Hansman, G, Tame, J.R.H, Kher, G, Pancera, M. | 登録日 | 2024-02-02 | 公開日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (1.47 Å) | 主引用文献 | Norovirus GII.10 P domain and 2'-FL (powder) To Be Published
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8Y66
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![BU of 8y66 by Molmil](/molmil-images/mine/8y66) | Cryo-EM structure of human urate transporter GLUT9 bound to inhibitor apigenin | 分子名称: | 5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one, Solute carrier family 2, facilitated glucose transporter member 9 | 著者 | Pan, X.J, Shen, Z.L, Xu, L, Huang, G.X.Y. | 登録日 | 2024-02-01 | 公開日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (3.28 Å) | 主引用文献 | Structural basis for urate recognition and apigenin inhibition of human GLUT9. Nat Commun, 15, 2024
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8Y65
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![BU of 8y65 by Molmil](/molmil-images/mine/8y65) | Cryo-EM structure of human urate transporter GLUT9 bound to substrate urate | 分子名称: | Solute carrier family 2, facilitated glucose transporter member 9, URIC ACID | 著者 | Pan, X.J, Shen, Z.L, Xu, L, Huang, G.X.Y. | 登録日 | 2024-02-01 | 公開日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (3.51 Å) | 主引用文献 | Structural basis for urate recognition and apigenin inhibition of human GLUT9. Nat Commun, 15, 2024
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8Y5V
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![BU of 8y5v by Molmil](/molmil-images/mine/8y5v) | GII.4 Sydney PD and 2'-FL | 分子名称: | 1,2-ETHANEDIOL, GII.4 Sydney PD in complex with 2'-FL (powder), alpha-L-fucopyranose-(1-2)-beta-D-galactopyranose-(1-4)-alpha-D-glucopyranose | 著者 | Hansman, G, Tame, J.R.H, Kher, G, Pancera, M. | 登録日 | 2024-02-01 | 公開日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (1.54 Å) | 主引用文献 | GII.4 Sydney PD and 2'-FL To Be Published
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8Y4J
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8Y46
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![BU of 8y46 by Molmil](/molmil-images/mine/8y46) | Crystal structure of L-2-keto-3-deoxyfuconate 4-dehydrogenase bound to L-KDF or L-2,4-DKDF | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, DI(HYDROXYETHYL)ETHER, L-2,4-diketo-3-deoxyfuconate, ... | 著者 | Akagashi, M, Watanabe, S. | 登録日 | 2024-01-30 | 公開日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (1.29 Å) | 主引用文献 | Crystal structure of L-2-keto-3-deoxyfuconate 4-dehydrogenase reveals a unique binding mode as a alpha-furanosyl hemiketal of substrates. Sci Rep, 14, 2024
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8Y3X
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![BU of 8y3x by Molmil](/molmil-images/mine/8y3x) | Cell divisome sPG hydrolysis machinery FtsEX-EnvC | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, Cell division ATP-binding protein FtsE, Cell division protein FtsX, ... | 著者 | Zhang, Z, Dong, H, Chen, Y. | 登録日 | 2024-01-29 | 公開日 | 2024-05-08 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (3.11 Å) | 主引用文献 | Structure and activity of the septal peptidoglycan hydrolysis machinery crucial for bacterial cell division. Plos Biol., 22, 2024
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8Y33
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![BU of 8y33 by Molmil](/molmil-images/mine/8y33) | A near-infrared fluorescent protein of de novo backbone design | 分子名称: | 3-[5-[(4-ethenyl-3-methyl-5-oxidanylidene-pyrrol-2-yl)methyl]-2-[[5-[(3-ethyl-4-methyl-5-oxidanylidene-pyrrol-2-yl)methyl]-3-(3-hydroxy-3-oxopropyl)-4-methyl-1~{H}-pyrrol-2-yl]methyl]-4-methyl-1~{H}-pyrrol-3-yl]propanoic acid, near-infrared fluorescent protein | 著者 | Hu, X, Xu, Y. | 登録日 | 2024-01-28 | 公開日 | 2024-02-28 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Using Protein Design and Directed Evolution to Monomerize a Bright Near-Infrared Fluorescent Protein. Acs Synth Biol, 13, 2024
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8Y2S
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![BU of 8y2s by Molmil](/molmil-images/mine/8y2s) | P-hydroxybenzoate hydroxylase complexed with 4-hydroxy-3-methylbenzoic acid | 分子名称: | 3-methyl-4-oxidanyl-benzoic acid, 4-hydroxybenzoate 3-monooxygenase, FLAVIN-ADENINE DINUCLEOTIDE | 著者 | Hara, K, Hashimoto, H, Matsushita, T, Kishimoto, S, Watanabe, K. | 登録日 | 2024-01-27 | 公開日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Functional Enhancement of Flavin-Containing Monooxygenase through Machine Learning Methodology Acs Catalysis, 14, 2024
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8Y22
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![BU of 8y22 by Molmil](/molmil-images/mine/8y22) | FGFR1 kinase domain with a covalent inhibitor 9g | 分子名称: | Fibroblast growth factor receptor 1, SULFATE ION, ~{N}-[4-[[4-azanyl-3-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrazolo[3,4-d]pyrimidin-1-yl]methyl]phenyl]propanamide | 著者 | Chen, X.J, Chen, Y.H. | 登録日 | 2024-01-25 | 公開日 | 2024-06-26 | 実験手法 | X-RAY DIFFRACTION (2.792 Å) | 主引用文献 | Design, synthesis and biological evaluation of 5-amino-1H-pyrazole-4-carboxamide derivatives as pan-FGFR covalent inhibitors. Eur.J.Med.Chem., 275, 2024
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8Y1R
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![BU of 8y1r by Molmil](/molmil-images/mine/8y1r) | in situ room temperature Laue crystallography | 分子名称: | Lysozyme C | 著者 | Wang, Z.J, Wang, S.S, Pan, Q.Y, Yu, L, Su, Z.H, Yang, T.Y, Wang, Y.Z, Zhang, W.Z, Hao, Q, Gao, X.Y. | 登録日 | 2024-01-25 | 公開日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | BL03HB: Laue crystallography beamline at SSRF To Be Published
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8Y1M
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![BU of 8y1m by Molmil](/molmil-images/mine/8y1m) | Xylanase R from Bacillus sp. TAR-1 complexed with xylobiose. | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ACETATE ION, ... | 著者 | Nakamura, T, Kuwata, K, Takita, T, Mizutani, K, Mikami, B, Nakamura, S, Yasukawa, K. | 登録日 | 2024-01-25 | 公開日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Activity-stability trade-off observed in variants at position 315 of the GH10 xylanase XynR. Sci Rep, 14, 2024
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8Y14
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8Y11
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8Y0X
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![BU of 8y0x by Molmil](/molmil-images/mine/8y0x) | Dormant ribosome with SERBP1 | 分子名称: | 18S rRNA, 28S rRNA, 40S ribosomal protein S10, ... | 著者 | Du, M, Zeng, F. | 登録日 | 2024-01-23 | 公開日 | 2024-02-07 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | The global structure of dormant ribosome To Be Published
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8Y0W
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8Y0G
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8XZ7
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![BU of 8xz7 by Molmil](/molmil-images/mine/8xz7) | FGFR1 kinase domain with a covalent inhibitor 10h | 分子名称: | 5-azanyl-3-[2-[4,6-bis(fluoranyl)-2-methyl-3~{H}-benzimidazol-5-yl]ethynyl]-1-[[3-(prop-2-enoylamino)phenyl]methyl]pyrazole-4-carboxamide, Fibroblast growth factor receptor 1, SULFATE ION | 著者 | Chen, X.J, Chen, Y.H. | 登録日 | 2024-01-20 | 公開日 | 2024-06-26 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Design, synthesis and biological evaluation of 5-amino-1H-pyrazole-4-carboxamide derivatives as pan-FGFR covalent inhibitors. Eur.J.Med.Chem., 275, 2024
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8XZ2
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![BU of 8xz2 by Molmil](/molmil-images/mine/8xz2) | The structural model of a homodimeric D-Ala-D-Ala metallopeptidase, VanX, from vancomycin-resistant bacteria | 分子名称: | D-alanyl-D-alanine dipeptidase | 著者 | Konuma, T, Takai, T, Tsuchiya, C, Nishida, M, Hashiba, M, Yamada, Y, Shirai, H, Motoda, Y, Nagadoi, A, Chikaishi, E, Akagi, K, Akashi, S, Yamazaki, T, Akutsu, H, Oe, A, Ikegami, T. | 登録日 | 2024-01-20 | 公開日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Analysis of the homodimeric structure of a D-Ala-D-Ala metallopeptidase, VanX, from vancomycin-resistant bacteria. Protein Sci., 33, 2024
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