4WD5
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6P8Q
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![BU of 6p8q by Molmil](/molmil-images/mine/6p8q) | EGFR in complex with a dihydrodibenzodiazepinone allosteric inhibitor. | 分子名称: | 1,2-ETHANEDIOL, 10-benzyl-2-fluoro-5,10-dihydro-11H-dibenzo[b,e][1,4]diazepin-11-one, ADENOSINE MONOPHOSPHATE, ... | 著者 | Yun, C.H, Heppner, D.E, Eck, M.J. | 登録日 | 2019-06-07 | 公開日 | 2019-12-18 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Discovery and Optimization of Dibenzodiazepinones as Allosteric Mutant-Selective EGFR Inhibitors. Acs Med.Chem.Lett., 10, 2019
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6JXT
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6JWL
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6JX0
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![BU of 6jx0 by Molmil](/molmil-images/mine/6jx0) | |
5CZH
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![BU of 5czh by Molmil](/molmil-images/mine/5czh) | |
5CZI
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5J87
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4LRM
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![BU of 4lrm by Molmil](/molmil-images/mine/4lrm) | EGFR D770_N771insNPG in complex with PD168393 | 分子名称: | Epidermal growth factor receptor, N-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | 著者 | Yun, C.H, Eck, M.J. | 登録日 | 2013-07-20 | 公開日 | 2014-01-15 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (3.526 Å) | 主引用文献 | Structural, Biochemical, and Clinical Characterization of Epidermal Growth Factor Receptor (EGFR) Exon 20 Insertion Mutations in Lung Cancer. Sci Transl Med, 5, 2013
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4LL0
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![BU of 4ll0 by Molmil](/molmil-images/mine/4ll0) | EGFR L858R/T790M in complex with PD168393 | 分子名称: | Epidermal growth factor receptor, N-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | 著者 | Yun, C.H, Eck, M.J. | 登録日 | 2013-07-09 | 公開日 | 2013-09-11 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (4 Å) | 主引用文献 | Mechanism for activation of mutated epidermal growth factor receptors in lung cancer. Proc.Natl.Acad.Sci.USA, 110, 2013
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7BTT
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8IZR
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8IZP
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5X28
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![BU of 5x28 by Molmil](/molmil-images/mine/5x28) | Crystal structure of EGFR 696-1022 L858R in complex with SKLB(6) | 分子名称: | 9-cyclohexyl-N2-[4-(4-methylpiperazin-1-yl)phenyl]-N8-phenyl-purine-2,8-diamine, CHLORIDE ION, Epidermal growth factor receptor | 著者 | Yun, C.H. | 登録日 | 2017-01-31 | 公開日 | 2018-02-07 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.952 Å) | 主引用文献 | Structural insights into drug development strategy targeting EGFR T790M/C797S. Oncotarget, 9, 2018
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5X2C
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5X2F
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5X27
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![BU of 5x27 by Molmil](/molmil-images/mine/5x27) | Crystal structure of EGFR 696-1022 L858R in complex with SKLB(5) | 分子名称: | 9-cyclopentyl-N2-[4-(4-methylpiperazin-1-yl)phenyl]-N8-phenyl-purine-2,8-diamine, CHLORIDE ION, Epidermal growth factor receptor | 著者 | Yun, C.H. | 登録日 | 2017-01-31 | 公開日 | 2018-02-07 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.952 Å) | 主引用文献 | Structural insights into drug development strategy targeting EGFR T790M/C797S. Oncotarget, 9, 2018
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5X2A
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5X26
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![BU of 5x26 by Molmil](/molmil-images/mine/5x26) | Crystal structure of EGFR 696-1022 L858R in complex with SKLB(3) | 分子名称: | CHLORIDE ION, Epidermal growth factor receptor, N2-[4-(4-methylpiperazin-1-yl)phenyl]-N8-phenyl-9-propan-2-yl-purine-2,8-diamine | 著者 | Yun, C.H. | 登録日 | 2017-01-31 | 公開日 | 2018-02-07 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.951 Å) | 主引用文献 | Structural insights into drug development strategy targeting EGFR T790M/C797S. Oncotarget, 9, 2018
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4LQM
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![BU of 4lqm by Molmil](/molmil-images/mine/4lqm) | EGFR L858R in complex with PD168393 | 分子名称: | CHLORIDE ION, Epidermal growth factor receptor, N-[4-(3-BROMO-PHENYLAMINO)-QUINAZOLIN-6-YL]-ACRYLAMIDE | 著者 | Yun, C.H, Eck, M.J. | 登録日 | 2013-07-19 | 公開日 | 2014-01-15 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structural, Biochemical, and Clinical Characterization of Epidermal Growth Factor Receptor (EGFR) Exon 20 Insertion Mutations in Lung Cancer. Sci Transl Med, 5, 2013
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4ZSE
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1RFJ
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![BU of 1rfj by Molmil](/molmil-images/mine/1rfj) | Crystal Structure of Potato Calmodulin PCM6 | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, CALCIUM ION, calmodulin | 著者 | Liang, D.C, Yun, C.H, Chang, W.R. | 登録日 | 2003-11-10 | 公開日 | 2004-06-29 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure of potato calmodulin PCM6: the first report of the three-dimensional structure of a plant calmodulin. Acta Crystallogr.,Sect.D, 60, 2004
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1TGR
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![BU of 1tgr by Molmil](/molmil-images/mine/1tgr) | Crystal Structure of mini-IGF-1(2) | 分子名称: | Insulin-like growth factor IA | 著者 | Liang, D.C, Yun, C.H, Chang, W.R. | 登録日 | 2004-05-29 | 公開日 | 2004-12-28 | 最終更新日 | 2021-11-10 | 実験手法 | X-RAY DIFFRACTION (1.42 Å) | 主引用文献 | 1.42A crystal structure of mini-IGF-1(2): an analysis of the disulfide isomerization property and receptor binding property of IGF-1 based on the three-dimensional structure Biochem.Biophys.Res.Commun., 326, 2004
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6LF6
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![BU of 6lf6 by Molmil](/molmil-images/mine/6lf6) | Crystal structure of ZmCGTa in complex with UDP | 分子名称: | UDP-glycosyltransferase 708A6, URIDINE-5'-DIPHOSPHATE | 著者 | Gao, H.M, Yun, C.H. | 登録日 | 2019-11-29 | 公開日 | 2020-11-18 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.044 Å) | 主引用文献 | Dissection of the general two-step di- C -glycosylation pathway for the biosynthesis of (iso)schaftosides in higher plants. Proc.Natl.Acad.Sci.USA, 117, 2020
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6LG1
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![BU of 6lg1 by Molmil](/molmil-images/mine/6lg1) | Crystal structure of LpCGTa in complex with UDP | 分子名称: | LpCGTa, URIDINE-5'-DIPHOSPHATE | 著者 | Gao, H.M, Yun, C.H. | 登録日 | 2019-12-04 | 公開日 | 2020-11-18 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (3.047 Å) | 主引用文献 | Dissection of the general two-step di- C -glycosylation pathway for the biosynthesis of (iso)schaftosides in higher plants. Proc.Natl.Acad.Sci.USA, 117, 2020
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