3IF5
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![BU of 3if5 by Molmil](/molmil-images/mine/3if5) | Crystal Structure Analysis of Mglu | 分子名称: | Salt-tolerant glutaminase | 著者 | Yoshimune, K, Shirakihara, Y. | 登録日 | 2009-07-24 | 公開日 | 2009-08-04 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.44 Å) | 主引用文献 | Crystal structure of salt-tolerant glutaminase from Micrococcus luteus K-3 in the presence and absence of its product L-glutamate and its activator Tris. Febs J., 277, 2010
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3IHB
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5B57
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![BU of 5b57 by Molmil](/molmil-images/mine/5b57) | Inward-facing conformation of ABC heme importer BhuUV from Burkholderia cenocepacia | 分子名称: | DECYL-BETA-D-MALTOPYRANOSIDE, Hemin import ATP-binding protein HmuV, Putative hemin ABC transport system, ... | 著者 | Naoe, Y, Nakamura, N, Doi, A, Shiro, Y, Sugimoto, H. | 登録日 | 2016-04-25 | 公開日 | 2016-11-16 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Crystal structure of bacterial haem importer complex in the inward-facing conformation Nat Commun, 7, 2016
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5AYV
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![BU of 5ayv by Molmil](/molmil-images/mine/5ayv) | Crystal structure of archaeal ketopantoate reductase complexed with coenzyme A and 2-oxopantoate | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 2-dehydropantoate 2-reductase, ACETATE ION, ... | 著者 | Aikawa, Y, Nishitani, Y, Miki, K. | 登録日 | 2015-09-08 | 公開日 | 2016-01-27 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.647 Å) | 主引用文献 | Crystal structure of archaeal ketopantoate reductase complexed with coenzyme a and 2-oxopantoate provides structural insights into feedback regulation Proteins, 84, 2016
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5B2V
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![BU of 5b2v by Molmil](/molmil-images/mine/5b2v) | Crystal Structure of P450BM3 with N-perfluorohexanoyl-L-tryptophan | 分子名称: | (2~{S})-3-(1~{H}-indol-3-yl)-2-[2,2,3,3,4,4,5,5,6,6,6-undecakis(fluoranyl)hexanoylamino]propanoic acid, Bifunctional cytochrome P450/NADPH--P450 reductase, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Cong, Z, Shoji, O, Kasai, C, Sugimoto, H, Shiro, Y, Watanabe, Y. | 登録日 | 2016-02-03 | 公開日 | 2017-02-08 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal Structure of P450BM3 with decoy molecules to be published
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8JLB
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![BU of 8jlb by Molmil](/molmil-images/mine/8jlb) | Cryo-EM structure of the 145 bp human nucleosome containing H3.2 C110A mutant | 分子名称: | DNA (145-MER), Histone H2A type 1-B/E, Histone H2B type 1-J, ... | 著者 | Oishi, T, Hatazawa, S, Kujirai, T, Kato, J, Kobayashi, Y, Ogasawara, M, Akatsu, M, Takizawa, Y, Kurumizaka, H. | 登録日 | 2023-06-02 | 公開日 | 2023-10-04 | 最終更新日 | 2023-11-08 | 実験手法 | ELECTRON MICROSCOPY (2.36 Å) | 主引用文献 | Contributions of histone tail clipping and acetylation in nucleosome transcription by RNA polymerase II. Nucleic Acids Res., 51, 2023
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8JL9
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![BU of 8jl9 by Molmil](/molmil-images/mine/8jl9) | Cryo-EM structure of the human nucleosome with scFv | 分子名称: | DNA (193-MER), Histone H2A type 1-B/E, Histone H2B type 1-J, ... | 著者 | Oishi, T, Hatazawa, S, Kujirai, T, Kato, J, Kobayashi, Y, Ogasawara, M, Akatsu, M, Takizawa, Y, Kurumizaka, H. | 登録日 | 2023-06-02 | 公開日 | 2023-10-04 | 最終更新日 | 2023-11-08 | 実験手法 | ELECTRON MICROSCOPY (2.65 Å) | 主引用文献 | Contributions of histone tail clipping and acetylation in nucleosome transcription by RNA polymerase II. Nucleic Acids Res., 51, 2023
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8JLD
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![BU of 8jld by Molmil](/molmil-images/mine/8jld) | Cryo-EM structure of the 145 bp human nucleosome containing acetylated H3 tail | 分子名称: | DNA (145-MER), Histone H2A type 1-B/E, Histone H2B type 1-J, ... | 著者 | Oishi, T, Hatazawa, S, Kujirai, T, Kato, J, Kobayashi, Y, Ogasawara, M, Akatsu, M, Takizawa, Y, Kurumizaka, H. | 登録日 | 2023-06-02 | 公開日 | 2023-10-04 | 最終更新日 | 2023-11-15 | 実験手法 | ELECTRON MICROSCOPY (2.48 Å) | 主引用文献 | Contributions of histone tail clipping and acetylation in nucleosome transcription by RNA polymerase II. Nucleic Acids Res., 51, 2023
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8JLA
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![BU of 8jla by Molmil](/molmil-images/mine/8jla) | Cryo-EM structure of the human nucleosome lacking N-terminal region of H2A, H2B, H3, and H4 | 分子名称: | DNA (193-MER), Histone H2A type 1-B/E, Histone H2B type 1-J, ... | 著者 | Oishi, T, Hatazawa, S, Kujirai, T, Kato, J, Kobayashi, Y, Ogasawara, M, Akatsu, M, Takizawa, Y, Kurumizaka, H. | 登録日 | 2023-06-02 | 公開日 | 2023-10-04 | 最終更新日 | 2023-11-08 | 実験手法 | ELECTRON MICROSCOPY (3.44 Å) | 主引用文献 | Contributions of histone tail clipping and acetylation in nucleosome transcription by RNA polymerase II. Nucleic Acids Res., 51, 2023
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4EBW
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![BU of 4ebw by Molmil](/molmil-images/mine/4ebw) | Structure of Focal Adhesion Kinase catalytic domain in complex with novel allosteric inhibitor | 分子名称: | 1-ethyl-8-(4-ethylphenyl)-5-methyl-1,5-dihydropyrazolo[4,3-c][2,1]benzothiazine 4,4-dioxide, Focal adhesion kinase 1 | 著者 | Iwatani, M, Iwata, H, Okabe, A, Skene, R.J, Tomita, N, Hayashi, Y, Aramaki, Y, Hosfield, D.J, Hori, A, Baba, A, Miki, H. | 登録日 | 2012-03-25 | 公開日 | 2012-07-25 | 最終更新日 | 2013-03-27 | 実験手法 | X-RAY DIFFRACTION (2.65 Å) | 主引用文献 | Discovery and characterization of novel allosteric FAK inhibitors. Eur.J.Med.Chem., 61, 2013
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5B2X
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![BU of 5b2x by Molmil](/molmil-images/mine/5b2x) | Crystal Structure of P450BM3 mutant with N-perfluoroheptanoyl-L-tryptophan | 分子名称: | (2~{S})-3-(1~{H}-indol-3-yl)-2-[2,2,3,3,4,4,5,5,6,6,7,7,7-tridecakis(fluoranyl)heptanoylamino]propanoic acid, Bifunctional cytochrome P450/NADPH--P450 reductase, DIMETHYL SULFOXIDE, ... | 著者 | Cong, Z, Shoji, O, Kasai, C, Sugimoto, H, Shiro, Y, Watanabe, Y. | 登録日 | 2016-02-03 | 公開日 | 2017-02-08 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal Structure of P450BM3 with decoy molecules to be published
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5B5E
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![BU of 5b5e by Molmil](/molmil-images/mine/5b5e) | Crystal structure analysis of Photosystem II complex | 分子名称: | (3R)-beta,beta-caroten-3-ol, 1,2-DI-O-ACYL-3-O-[6-DEOXY-6-SULFO-ALPHA-D-GLUCOPYRANOSYL]-SN-GLYCEROL, 1,2-DIPALMITOYL-PHOSPHATIDYL-GLYCEROLE, ... | 著者 | Tanaka, A, Fukushima, Y, Kamiya, N. | 登録日 | 2016-05-02 | 公開日 | 2017-02-01 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | Two Different Structures of the Oxygen-Evolving Complex in the Same Polypeptide Frameworks of Photosystem II J. Am. Chem. Soc., 139, 2017
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4GVJ
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![BU of 4gvj by Molmil](/molmil-images/mine/4gvj) | Tyk2 (JH1) in complex with adenosine di-phosphate | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Non-receptor tyrosine-protein kinase TYK2 | 著者 | Liang, J, Abbema, A.V, Bao, L, Barrett, K, Beresini, M, Berezhkovskiy, L, Blair, W, Chang, C, Driscoll, J, Eigenbrot, C, Ghilardi, N, Gibbons, P, Halladay, J, Johnson, A, Kohli, P.B, Lai, Y, Liimatta, M, Mantik, P, Menghrajani, K, Murray, J, Sambrone, A, Shao, Y, Shia, S, Shin, Y, Smith, J, Sohn, S, Stanley, M, Tsui, V, Ultsch, M, Wu, L, Zhang, B, Magnuson, S. | 登録日 | 2012-08-30 | 公開日 | 2013-08-14 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.03 Å) | 主引用文献 | Lead identification of novel and selective TYK2 inhibitors. Eur.J.Med.Chem., 67, 2013
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7COY
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![BU of 7coy by Molmil](/molmil-images/mine/7coy) | Structure of the far-red light utilizing photosystem I of Acaryochloris marina | 分子名称: | 1,2-DIPALMITOYL-PHOSPHATIDYL-GLYCEROLE, 1,2-DISTEAROYL-MONOGALACTOSYL-DIGLYCERIDE, CHLOROPHYLL D, ... | 著者 | Kawakami, K, Yonekura, K, Hamaguchi, T, Kashino, Y, Shinzawa-Itoh, K, Inoue-Kashino, N, Itoh, S, Ifuku, K, Yamashita, E. | 登録日 | 2020-08-05 | 公開日 | 2021-03-31 | 最終更新日 | 2021-05-05 | 実験手法 | ELECTRON MICROSCOPY (2.5 Å) | 主引用文献 | Structure of the far-red light utilizing photosystem I of Acaryochloris marina. Nat Commun, 12, 2021
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8JOG
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![BU of 8jog by Molmil](/molmil-images/mine/8jog) | solution structure of Ras Binding Domein (RBD) in C-RAF with negative allosteric modulator. | 分子名称: | RAF proto-oncogene serine/threonine-protein kinase | 著者 | Makino, Y, Matsumoto, S, Yoshikawa, Y, Kawamura, T, Kumasaka, T, Shima, F. | 登録日 | 2023-06-07 | 公開日 | 2024-06-12 | 実験手法 | SOLUTION NMR | 主引用文献 | Small-molecule RAS/RAF-binding Inhibitors Allosterically Disrupt RAF Conformation and Exert Efficacy Against Broad-spectrum RAS-driven Cancers To Be Published
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8JOF
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![BU of 8jof by Molmil](/molmil-images/mine/8jof) | solution-structure of Ras Binding Domain (RBD) in C-RAF | 分子名称: | RAF proto-oncogene serine/threonine-protein kinase | 著者 | Makino, Y, Matsumoto, S, Yoshikawa, Y, Kawamura, T, Kumasaka, T, Shima, F. | 登録日 | 2023-06-07 | 公開日 | 2024-06-12 | 実験手法 | SOLUTION NMR | 主引用文献 | Small-molecule RAS/RAF-binding Inhibitors Allosterically Disrupt RAF Conformation and Exert Efficacy Against Broad-spectrum RAS-driven Cancers To Be Published
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3ORY
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![BU of 3ory by Molmil](/molmil-images/mine/3ory) | Crystal structure of Flap endonuclease 1 from hyperthermophilic archaeon Desulfurococcus amylolyticus | 分子名称: | PHOSPHATE ION, flap endonuclease 1 | 著者 | Mase, T, Kubota, K, Miyazono, K, Kawarabayashii, Y, Tanokura, M. | 登録日 | 2010-09-08 | 公開日 | 2011-02-09 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure of flap endonuclease 1 from the hyperthermophilic archaeon Desulfurococcus amylolyticus Acta Crystallogr.,Sect.F, 67, 2011
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7CG3
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![BU of 7cg3 by Molmil](/molmil-images/mine/7cg3) | Staggered ring conformation of CtHsp104 (Hsp104 from Chaetomium Thermophilum) | 分子名称: | Heat shock protein 104 | 著者 | Inoue, Y, Hanazono, Y, Noi, K, Kawamoto, A, Kimatsuka, M, Harada, R, Takeda, K, Iwamasa, N, Shibata, K, Noguchi, K, Shigeta, Y, Namba, K, Ogura, T, Miki, K, Shinohara, K, Yohda, M. | 登録日 | 2020-06-30 | 公開日 | 2021-04-28 | 最終更新日 | 2024-05-29 | 実験手法 | ELECTRON MICROSCOPY (5.1 Å) | 主引用文献 | Split conformation of Chaetomium thermophilum Hsp104 disaggregase. Structure, 29, 2021
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3MCH
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![BU of 3mch by Molmil](/molmil-images/mine/3mch) | Crystal structure of the molybdopterin biosynthesis enzyme MoaB (TTHA0341) from thermus theromophilus HB8 | 分子名称: | 1,2-ETHANEDIOL, Molybdopterin biosynthesis enzyme, MoaB | 著者 | Jeyakanthan, J, Kanaujia, S.P, Sekar, K, Baba, S, Ebihara, A, Kuramitsu, S, Shinkai, A, Shiro, Y, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2010-03-29 | 公開日 | 2011-01-19 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.64 Å) | 主引用文献 | Crystal structures, dynamics and functional implications of molybdenum-cofactor biosynthesis protein MogA from two thermophilic organisms Acta Crystallogr.,Sect.F, 67, 2011
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5B2Y
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![BU of 5b2y by Molmil](/molmil-images/mine/5b2y) | Crystal Structure of P450BM3 with N-perfluorodecanoyl-L-tryptophan | 分子名称: | (2~{S})-3-(1~{H}-indol-3-yl)-2-[2,2,3,3,4,4,5,5,6,6,7,7,8,8,9,9,10,10,10-nonadecakis(fluoranyl)decanoylamino]propanoic acid, Bifunctional cytochrome P450/NADPH--P450 reductase, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Cong, Z, Shoji, O, Kasai, C, Sugimoto, H, Shiro, Y, Watanabe, Y. | 登録日 | 2016-02-07 | 公開日 | 2017-02-08 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.01 Å) | 主引用文献 | Crystal Structure of P450BM3 with decoy molecules to be published
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5B58
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![BU of 5b58 by Molmil](/molmil-images/mine/5b58) | Inward-facing conformation of ABC heme importer BhuUV in complex with periplasmic heme binding protein BhuT from Burkholderia cenocepacia | 分子名称: | Hemin import ATP-binding protein HmuV, Putative hemin ABC transport system, membrane protein, ... | 著者 | Naoe, Y, Nakamura, N, Doi, A, Shiro, Y, Sugimoto, H. | 登録日 | 2016-04-25 | 公開日 | 2016-11-23 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (3.21 Å) | 主引用文献 | Crystal structure of bacterial haem importer complex in the inward-facing conformation Nat Commun, 7, 2016
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3OV3
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![BU of 3ov3 by Molmil](/molmil-images/mine/3ov3) | G211F mutant of curcumin synthase 1 from Curcuma longa | 分子名称: | Curcumin synthase, MALONATE ION | 著者 | Katsuyama, Y, Miyazono, K, Tanokura, M, Ohnishi, Y, Horinouchi, S. | 登録日 | 2010-09-15 | 公開日 | 2010-12-08 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | A hydrophobic cavity discovered in a curcumin synthase facilitates utilization of a beta-keto acid as an extender substrate for the atypical type III polyleteide synthase To be Published
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4KEQ
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![BU of 4keq by Molmil](/molmil-images/mine/4keq) | Crystal structure of 4-pyridoxolactonase, 5-pyridoxolactone bound | 分子名称: | 1,2-ETHANEDIOL, 4-pyridoxolactonase, 7-hydroxy-6-methylfuro[3,4-c]pyridin-3(1H)-one, ... | 著者 | Kobayashi, J, Yoshikane, Y, Baba, S, Mizutani, K, Takahashi, N, Mikami, B, Yagi, T. | 登録日 | 2013-04-26 | 公開日 | 2014-04-09 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.279 Å) | 主引用文献 | Structure of 4-pyridoxolactonase from Mesorhizobium loti. Acta Crystallogr.,Sect.F, 70, 2014
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3OIT
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![BU of 3oit by Molmil](/molmil-images/mine/3oit) | Crystal structure of curcuminoid synthase CUS from Oryza sativa | 分子名称: | Os07g0271500 protein | 著者 | Miyazono, K, Um, J, Imai, F.L, Katsuyama, Y, Ohnishi, Y, Horinouchi, S, Tanokura, M. | 登録日 | 2010-08-19 | 公開日 | 2010-10-20 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal structure of curcuminoid synthase CUS from Oryza sativa Proteins, 79, 2011
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5ZLE
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![BU of 5zle by Molmil](/molmil-images/mine/5zle) | Human duodenal cytochrome b (Dcytb) in substrate free form | 分子名称: | Cytochrome b reductase 1, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Ganasen, M, Togashi, H, Mauk, G.A, Shiro, Y, Sawai, H, Sugimoto, H. | 登録日 | 2018-03-27 | 公開日 | 2018-10-31 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structural basis for promotion of duodenal iron absorption by enteric ferric reductase with ascorbate. Commun Biol, 1, 2018
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