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PDB: 27399 件

8CN2
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Pa.FabF-C164Q in complex with N-isobutyl-1H-pyrazole-3-carboxamide
分子名称: 3-oxoacyl-[acyl-carrier-protein] synthase 2, DIMETHYL SULFOXIDE, ~{N}-(2-methylpropyl)-1~{H}-pyrazole-3-carboxamide
著者Georgiou, C, Brenk, R.
登録日2023-02-21
公開日2024-01-10
実験手法X-RAY DIFFRACTION (1.88 Å)
主引用文献New starting points for antibiotics targeting P. aeruginosa FabF discovered by crystallographic fragment screening followed by hit expansion
Chemrxiv, 2023
5GQV
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Crystal structure of branching enzyme from Cyanothece sp. ATCC 51142 in complex with maltohexaose
分子名称: 1,4-alpha-glucan branching enzyme GlgB, GLYCEROL, MAGNESIUM ION, ...
著者Suzuki, R, Suzuki, E.
登録日2016-08-08
公開日2017-02-22
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Bound Substrate in the Structure of Cyanobacterial Branching Enzyme Supports a New Mechanistic Model
J. Biol. Chem., 292, 2017
5GR4
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Crystal structure of branching enzyme L541A mutant from Cyanothece sp. ATCC 51142 in complex with maltoheptaose
分子名称: 1,4-alpha-glucan branching enzyme GlgB, GLYCEROL, MAGNESIUM ION, ...
著者Suzuki, R, Suzuki, E.
登録日2016-08-08
公開日2017-08-16
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural basis for substrate binding and catalysis of branching enzyme from Cyanothece sp. ATCC 51142
To be published
8C64
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Crystal structure of arsenoplatin-1/B-DNA adduct obtained upon 48 h of soaking
分子名称: DNA (5'-D(*CP*GP*CP*GP*AP*AP*TP*TP*CP*GP*CP*G)-3'), PLATINUM (II) ION, arsenoplatin-1
著者Troisi, R, Tito, G, Ferraro, G, Sica, F, Merlino, A.
登録日2023-01-11
公開日2024-01-31
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.51 Å)
主引用文献On the mechanism of action of arsenoplatins: arsenoplatin-1 binding to a B-DNA dodecamer.
Dalton Trans, 53, 2024
8C9H
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AQP7_inhibitor
分子名称: Aquaporin-7, ethyl 4-[(4-pyrazol-1-ylphenyl)methylcarbamoylamino]benzoate
著者Huang, P, Venskutonyte, R, Gourdon, P, Lindkvist-Petersson, K.
登録日2023-01-22
公開日2024-01-31
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Molecular basis for human aquaporin inhibition.
Proc.Natl.Acad.Sci.USA, 121, 2024
8C62
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Crystal structure of cisplatin/B-DNA adduct
分子名称: DNA (5'-D(*CP*GP*CP*GP*AP*AP*TP*TP*CP*GP*CP*G)-3'), PLATINUM (II) ION
著者Troisi, R, Tito, G, Ferraro, G, Sica, F, Merlino, A.
登録日2023-01-11
公開日2024-01-31
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.31 Å)
主引用文献On the mechanism of action of arsenoplatins: arsenoplatin-1 binding to a B-DNA dodecamer.
Dalton Trans, 53, 2024
1IMF
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STRUCTURAL STUDIES OF METAL BINDING BY INOSITOL MONOPHOSPHATASE: EVIDENCE FOR TWO-METAL ION CATALYSIS
分子名称: INOSITOL MONOPHOSPHATASE
著者Bone, R.
登録日1994-02-08
公開日1995-02-27
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural studies of metal binding by inositol monophosphatase: evidence for two-metal ion catalysis.
Biochemistry, 33, 1994
2YMD
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BU of 2ymd by Molmil
Crystal structure of a mutant binding protein (5HTBP-AChBP) in complex with serotonin (5-hydroxytryptamine)
分子名称: GLYCEROL, PHOSPHATE ION, SEROTONIN, ...
著者Kesters, D, Thompson, A.J, Brams, M, Elk, R.v, Spurny, R, Geitmann, M, Villalgordo, J.M, Guskov, A, Danielson, U.H, Lummis, S.C.R, Smit, A.B, Ulens, C.
登録日2012-10-09
公開日2012-12-12
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献Structural Basis of Ligand Recognition in 5-Ht(3) Receptors.
Embo Rep., 14, 2013
8C9L
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Crystal structure of SARS-CoV-2 Mpro-S144A mutant, free enzyme
分子名称: 3C-like proteinase nsp5
著者El Kilani, H, Ibrahim, M, Hilgenfeld, R.
登録日2023-01-23
公開日2024-02-07
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structure of SARS-CoV-2 Mpro-S144A mutant, free enzyme
To Be Published
8C9O
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Crystal structure of SARS-CoV-2 Mpro-S144A mutant in complex with 13b-K
分子名称: 3C-like proteinase nsp5, ~{tert}-butyl ~{N}-[1-[(2~{S})-3-cyclopropyl-1-oxidanylidene-1-[[(2~{S},3~{R})-3-oxidanyl-4-oxidanylidene-1-[(3~{S})-2-oxidanylidenepyrrolidin-3-yl]-4-[(phenylmethyl)amino]butan-2-yl]amino]propan-2-yl]-2-oxidanylidene-pyridin-3-yl]carbamate
著者Ibrahim, M, El Kilani, H, Hilgenfeld, R.
登録日2023-01-23
公開日2024-02-07
実験手法X-RAY DIFFRACTION (1.69 Å)
主引用文献Crystal structure of SARS-CoV-2 Mpro_S144A mutant in complex with 13b-K
To Be Published
1N62
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Crystal Structure of the Mo,Cu-CO Dehydrogenase (CODH), n-butylisocyanide-bound state
分子名称: CU(I)-S-MO(IV)(=O)O-NBIC CLUSTER, Carbon monoxide dehydrogenase large chain, Carbon monoxide dehydrogenase medium chain, ...
著者Dobbek, H, Gremer, L, Kiefersauer, R, Huber, R, Meyer, O.
登録日2002-11-08
公開日2002-12-18
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.09 Å)
主引用文献Catalysis at a dinuclear [CuSMo(=O)OH] cluster in a CO dehydrogenase resolved at 1.1-A resolution
Proc.Natl.Acad.Sci.USA, 99, 2002
4MIV
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BU of 4miv by Molmil
Crystal Structure of Sulfamidase, Crystal Form L
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Sidhu, N.S, Uson, I, Schreiber, K, Proepper, K, Becker, S, Sheldrick, G.M, Gaertner, J, Kraetzner, R, Steinfeld, R.
登録日2013-09-02
公開日2014-05-14
最終更新日2021-06-02
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structure of sulfamidase provides insight into the molecular pathology of mucopolysaccharidosis IIIA.
Acta Crystallogr.,Sect.D, 70, 2014
1N60
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Crystal Structure of the Cu,Mo-CO Dehydrogenase (CODH); Cyanide-inactivated Form
分子名称: Carbon monoxide dehydrogenase large chain, Carbon monoxide dehydrogenase medium chain, Carbon monoxide dehydrogenase small chain, ...
著者Dobbek, H, Gremer, L, Kiefersauer, R, Huber, R, Meyer, O.
登録日2002-11-08
公開日2002-12-18
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.19 Å)
主引用文献Catalysis at a dinuclear [CuSMo(=O)OH] cluster in a CO dehydrogenase resolved at 1.1-A resolution
Proc.Natl.Acad.Sci.USA, 99, 2002
5GQY
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BU of 5gqy by Molmil
Crystal structure of branching enzyme from Cyanothece sp. ATCC 51142 in complex with maltoheptaose
分子名称: 1,4-alpha-glucan branching enzyme GlgB, GLYCEROL, MAGNESIUM ION, ...
著者Suzuki, R, Suzuki, E.
登録日2016-08-08
公開日2017-08-16
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural basis for substrate binding and catalysis of branching enzyme from Cyanothece sp. ATCC 51142
To be published
8COD
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BU of 8cod by Molmil
Crystal structure of S-adenosyl-L-homocysteine hydrolase from Mus musculus in complex with inosine
分子名称: Adenosylhomocysteinase, INOSINE, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ...
著者Saleem-Batcha, R, Popadic, D, Koeppl, L.H, Andexer, J.N.
登録日2023-02-27
公開日2024-03-06
最終更新日2024-09-18
実験手法X-RAY DIFFRACTION (2.48 Å)
主引用文献Structure, function and substrate preferences of archaeal S-adenosyl-L-homocysteine hydrolases.
Commun Biol, 7, 2024
8CKH
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BU of 8ckh by Molmil
Crystal structure of IspE from Klebsiella pneumoniae
分子名称: 4-diphosphocytidyl-2-C-methyl-D-erythritol kinase, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER
著者Hamid, R.
登録日2023-02-15
公開日2024-02-28
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal structure of IspE from Klebsiella pneumoniae
To Be Published
1IMC
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BU of 1imc by Molmil
STRUCTURAL STUDIES OF METAL BINDING BY INOSITOL MONOPHOSPHATASE: EVIDENCE FOR TWO-METAL ION CATALYSIS
分子名称: CHLORIDE ION, INOSITOL MONOPHOSPHATASE, MANGANESE (II) ION
著者Bone, R.
登録日1994-02-08
公開日1995-02-27
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structural studies of metal binding by inositol monophosphatase: evidence for two-metal ion catalysis.
Biochemistry, 33, 1994
8F41
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3-methylcrotonyl-CoA carboxylase in filament, alpha-subunit centered
分子名称: 3-methylcrotonyl-CoA carboxylase, alpha-subunit, beta-subunit, ...
著者Hu, J.J, Lee, J.K.J, Liu, Y.T, Yu, C, Huang, L, Afasizheva, I, Afasizhev, R, Zhou, Z.H.
登録日2022-11-10
公開日2023-01-11
最終更新日2024-06-19
実験手法ELECTRON MICROSCOPY (3.9 Å)
主引用文献Discovery, structure, and function of filamentous 3-methylcrotonyl-CoA carboxylase.
Structure, 31, 2023
8CMV
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BU of 8cmv by Molmil
Engineered PETase enzyme from LCC - C09 mutant
分子名称: GLYCEROL, ISOPROPYL ALCOHOL, Leaf-branch compost cutinase
著者Bhattacharya, S, Estiri, H, Castagna, R, Parisini, E.
登録日2023-02-21
公開日2024-03-06
実験手法X-RAY DIFFRACTION (1.28 Å)
主引用文献Engineered PETase Enzyme
To Be Published
2ZCE
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BU of 2zce by Molmil
Crystal structure of the catalytic domain of pyrrolysyl-tRNA synthetase in complex with pyrrolysine and an ATP analogue
分子名称: MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, PYRROLYSINE, ...
著者Yanagisawa, T, Ishii, R, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2007-11-08
公開日2008-04-22
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystallographic Studies on Multiple Conformational States of Active-site Loops in Pyrrolysyl-tRNA Synthetase
J.Mol.Biol., 378, 2008
2ZIN
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Crystal structure of the catalytic domain of pyrrolysyl-tRNA synthetase in complex with BocLys and an ATP analogue
分子名称: 1,2-ETHANEDIOL, MAGNESIUM ION, N~6~-(tert-butoxycarbonyl)-L-lysine, ...
著者Yanagisawa, T, Ishii, R, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2008-02-19
公開日2008-12-02
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.79 Å)
主引用文献Multistep Engineering of Pyrrolysyl-tRNA Synthetase to Genetically Encode N(varepsilon)-(o-Azidobenzyloxycarbonyl) lysine for Site-Specific Protein Modification
Chem.Biol., 15, 2008
4MP4
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BU of 4mp4 by Molmil
Crystal structure of a glutathione transferase family member from Acinetobacter baumannii, Target EFI-501785, apo structure
分子名称: Glutathione S-transferase, SULFATE ION
著者Vetting, M.W, Toro, R, Bhosle, R, Al Obaidi, N.F, Morisco, L.L, Wasserman, S.R, Sojitra, S, Stead, M, Scott Glenn, A, Chowdhury, S, Evans, B, Hillerich, B, Love, J, Seidel, R.D, Imker, H.J, Gerlt, J.A, Armstrong, R.N, Almo, S.C, Enzyme Function Initiative (EFI)
登録日2013-09-12
公開日2013-10-09
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.498 Å)
主引用文献Crystal structure of a glutathione transferase family member from Acinetobacter baumannii, Target EFI-501785, apo structure
To be Published
6Y0P
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isopenicillin N synthase in complex with IPN and Fe using FT-SSX methods
分子名称: FE (III) ION, ISOPENICILLIN N, Isopenicillin N synthase, ...
著者Rabe, P, Beale, J.H, Lang, P.A, Dirr, A.S, Leissing, T.M, Butryn, A, Aller, P, Kamps, J.J.A.G, Axford, D, McDonough, M.A, Orville, A.M, Owen, R, Schofield, C.J.
登録日2020-02-10
公開日2021-02-17
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献X-ray free-electron laser studies reveal correlated motion during isopenicillin N synthase catalysis.
Sci Adv, 7, 2021
6PTO
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BU of 6pto by Molmil
Structure of Ctf4 trimer in complex with three CMG helicases
分子名称: ADENOSINE-5'-TRIPHOSPHATE, Cell division control protein 45, DNA polymerase alpha-binding protein, ...
著者Yuan, Z, Georgescu, R, Bai, L, Santos, R, Donnell, M, Li, H.
登録日2019-07-16
公開日2019-11-20
最終更新日2019-12-18
実験手法ELECTRON MICROSCOPY (7 Å)
主引用文献Ctf4 organizes sister replisomes and Pol alpha into a replication factory.
Elife, 8, 2019
1HM5
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BU of 1hm5 by Molmil
CRYSTAL STRUCTURE ANALYSIS OF THE RABBIT D-GLUCOSE 6-PHOSPHATE ISOMERASE (NO LIGAND BOUND)
分子名称: PHOSPHOGLUCOSE ISOMERASE
著者Arsenieva, D.A, Jeffery, C.J, Hardre, R, Salmon, L.
登録日2000-12-04
公開日2002-09-27
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Conformational Changes in Phosphoglucose Isomerase Induced by Ligand Binding
J.Mol.Biol., 323, 2002

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件を2024-09-18に公開中

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