2YWP
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![BU of 2ywp by Molmil](/molmil-images/mine/2ywp) | Crystal Structure of CHK1 with a Urea Inhibitor | 分子名称: | 1-(5-CHLORO-2,4-DIMETHOXYPHENYL)-3-(5-CYANOPYRAZIN-2-YL)UREA, Serine/threonine-protein kinase Chk1 | 著者 | Park, C. | 登録日 | 2007-04-21 | 公開日 | 2007-05-08 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Synthesis and biological evaluation of 1-(2,4,5-trisubstituted phenyl)-3-(5-cyanopyrazin-2-yl)ureas as potent Chk1 kinase inhibitors Bioorg.Med.Chem.Lett., 16, 2006
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3GJW
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![BU of 3gjw by Molmil](/molmil-images/mine/3gjw) | PARP complexed with A968427 | 分子名称: | 7-(pyrrolidin-1-ylmethyl)pyrrolo[1,2-a]quinoxalin-4(5H)-one, Poly [ADP-ribose] polymerase 1 | 著者 | Park, C.H. | 登録日 | 2009-03-09 | 公開日 | 2010-03-09 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Synthesis and SAR of novel tricyclic quinoxalinone inhibitors of poly(ADP-ribose)polymerase-1 (PARP-1) Bioorg.Med.Chem.Lett., 19, 2009
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3GN7
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![BU of 3gn7 by Molmil](/molmil-images/mine/3gn7) | PARP complexed with A861696 | 分子名称: | 2-[(2S)-2-methylpyrrolidin-2-yl]-1H-benzimidazole-7-carboxamide, Poly [ADP-ribose] polymerase 1 | 著者 | Park, C.H. | 登録日 | 2009-03-16 | 公開日 | 2010-03-16 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | PARP complexed with A861696 To be Published
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2GHG
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![BU of 2ghg by Molmil](/molmil-images/mine/2ghg) | h-CHK1 complexed with A431994 | 分子名称: | 5-{5-[(S)-2-AMINO-3-(1H-INDOL-3-YL)-PROPOXYL]-PYRIDIN-3-YL}-3-[1-(1H-PYRROL-2-YL)-METH-(Z)-YLIDENE]-1,3-DIHYDRO-INDOL-2-ONE, Serine/threonine-protein kinase Chk1 | 著者 | Park, C. | 登録日 | 2006-03-27 | 公開日 | 2007-03-27 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | Discovery and SAR of oxindole-pyridine-based protein kinase B/Akt inhibitors for treating cancers. Bioorg.Med.Chem.Lett., 16, 2006
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2QF6
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![BU of 2qf6 by Molmil](/molmil-images/mine/2qf6) | HSP90 complexed with A56322 | 分子名称: | 6-(3-BROMO-2-NAPHTHYL)-1,3,5-TRIAZINE-2,4-DIAMINE, Heat shock protein HSP 90-alpha | 著者 | Park, C.H. | 登録日 | 2007-06-26 | 公開日 | 2008-07-01 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Discovery and design of novel HSP90 inhibitors using multiple fragment-based design strategies. Chem.Biol.Drug Des., 70, 2007
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2QG2
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![BU of 2qg2 by Molmil](/molmil-images/mine/2qg2) | HSP90 complexed with A917985 | 分子名称: | 3-({2-[(2-AMINO-6-METHYLPYRIMIDIN-4-YL)ETHYNYL]BENZYL}AMINO)-1,3-OXAZOL-2(3H)-ONE, Heat shock protein HSP 90-alpha | 著者 | Park, C.H. | 登録日 | 2007-06-28 | 公開日 | 2008-07-01 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Discovery and design of novel HSP90 inhibitors using multiple fragment-based design strategies. Chem.Biol.Drug Des., 70, 2007
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2QG0
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![BU of 2qg0 by Molmil](/molmil-images/mine/2qg0) | HSP90 complexed with A943037 | 分子名称: | Heat shock protein HSP 90-alpha, N-[(2-AMINO-6-METHYLPYRIMIDIN-4-YL)METHYL]-3-{[(E)-(2-OXODIHYDROFURAN-3(2H)-YLIDENE)METHYL]AMINO}BENZENESULFONAMIDE | 著者 | Park, C.H. | 登録日 | 2007-06-28 | 公開日 | 2008-07-01 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Discovery and design of novel HSP90 inhibitors using multiple fragment-based design strategies. Chem.Biol.Drug Des., 70, 2007
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2QFO
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![BU of 2qfo by Molmil](/molmil-images/mine/2qfo) | HSP90 complexed with A143571 and A516383 | 分子名称: | (3E)-3-[(phenylamino)methylidene]dihydrofuran-2(3H)-one, 4-METHYL-6-(TRIFLUOROMETHYL)PYRIMIDIN-2-AMINE, Heat shock protein HSP 90-alpha | 著者 | Park, C.H. | 登録日 | 2007-06-27 | 公開日 | 2008-07-01 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.68 Å) | 主引用文献 | Discovery and design of novel HSP90 inhibitors using multiple fragment-based design strategies. CHEM.BIOL.DRUG DES., 70, 2007
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3HQD
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![BU of 3hqd by Molmil](/molmil-images/mine/3hqd) | Human kinesin Eg5 motor domain in complex with AMPPNP and Mg2+ | 分子名称: | Kinesin-like protein KIF11, MAGNESIUM ION, PHOSPHATE ION, ... | 著者 | Parke, C.L, Wojcik, E.J, Kim, S, Worthylake, D.K. | 登録日 | 2009-06-05 | 公開日 | 2009-12-08 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.19 Å) | 主引用文献 | ATP Hydrolysis in Eg5 Kinesin Involves a Catalytic Two-water Mechanism. J.Biol.Chem., 285, 2010
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3KEN
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![BU of 3ken by Molmil](/molmil-images/mine/3ken) | Human Eg5 in complex with S-trityl-L-cysteine | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, Kinesin-like protein KIF11, MAGNESIUM ION, ... | 著者 | Parke, C.L, Wojcik, E.J, Kim, S, Worthylake, D.K. | 登録日 | 2009-10-26 | 公開日 | 2010-03-16 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Allosteric drug discrimination is coupled to mechanochemical changes in the kinesin-5 motor core. J.Biol.Chem., 285, 2010
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1X8D
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![BU of 1x8d by Molmil](/molmil-images/mine/1x8d) | Crystal structure of E. coli YiiL protein containing L-rhamnose | 分子名称: | Hypothetical protein yiiL, L-RHAMNOSE | 著者 | Ryu, K.S, Kim, J.I, Cho, S.J, Park, D, Park, C, Lee, J.O, Choi, B.S. | 登録日 | 2004-08-18 | 公開日 | 2005-05-17 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structural Insights into the Monosaccharide Specificity of Escherichia coli Rhamnose Mutarotase J.Mol.Biol., 349, 2005
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7C0I
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![BU of 7c0i by Molmil](/molmil-images/mine/7c0i) | Crystal structure of chimeric mutant of E3L in complex with Z-DNA | 分子名称: | DNA (5'-D(*TP*CP*GP*CP*GP*CP*G)-3'), Double-stranded RNA-binding protein,Double-stranded RNA-specific adenosine deaminase, SULFATE ION | 著者 | Choi, H.J, Park, C.H, Kim, J.S. | 登録日 | 2020-05-01 | 公開日 | 2020-12-16 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Dual conformational recognition by Z-DNA binding protein is important for the B-Z transition process. Nucleic Acids Res., 48, 2020
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7C0J
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4AEE
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![BU of 4aee by Molmil](/molmil-images/mine/4aee) | CRYSTAL STRUCTURE OF MALTOGENIC AMYLASE FROM S.MARINUS | 分子名称: | ALPHA AMYLASE, CATALYTIC REGION | 著者 | Jung, T.Y, Park, C.H, Yoon, S.M, Park, S.H, Park, K.H, Woo, E.J. | 登録日 | 2012-01-10 | 公開日 | 2012-01-18 | 最終更新日 | 2012-03-21 | 実験手法 | X-RAY DIFFRACTION (2.28 Å) | 主引用文献 | Association of Novel Domain in Active Site of Archaic Hyperthermophilic Maltogenic Amylase from Staphylothermus Marinus. J.Biol.Chem., 287, 2012
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2RVC
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![BU of 2rvc by Molmil](/molmil-images/mine/2rvc) | Solution structure of Zalpha domain of goldfish ZBP-containing protein kinase | 分子名称: | Interferon-inducible and double-stranded-dependent eIF-2kinase | 著者 | Lee, A, Park, C, Park, J, Kwon, M, Choi, Y, Kim, K, Choi, B, Lee, J. | 登録日 | 2015-07-08 | 公開日 | 2016-02-03 | 最終更新日 | 2024-05-01 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the Z-DNA binding domain of PKR-like protein kinase from Carassius auratus and quantitative analyses of the intermediate complex during B-Z transition. Nucleic Acids Res., 44, 2016
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4CMR
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![BU of 4cmr by Molmil](/molmil-images/mine/4cmr) | The crystal structure of novel exo-type maltose-forming amylase(Py04_0872) from Pyrococcus sp. ST04 | 分子名称: | GLYCOSYL HYDROLASE/DEACETYLASE FAMILY PROTEIN | 著者 | Park, K.-H, Jung, J.-H, Park, C.-S, Woo, E.-J. | 登録日 | 2014-01-17 | 公開日 | 2014-10-22 | 最終更新日 | 2019-10-16 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structural Features Underlying the Selective Cleavage of a Novel Exo-Type Maltose-Forming Amylase from Pyrococcus Sp. St04 Acta Crystallogr.,Sect.D, 70, 2014
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1DC3
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1DC4
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![BU of 1dc4 by Molmil](/molmil-images/mine/1dc4) | STRUCTURAL ANALYSIS OF GLYCERALDEHYDE 3-PHOSPHATE DEHYDROGENASE FROM ESCHERICHIA COLI: DIRECT EVIDENCE FOR SUBSTRATE BINDING AND COFACTOR-INDUCED CONFORMATIONAL CHANGES | 分子名称: | GLYCERALDEHYDE 3-PHOSPHATE DEHYDROGENASE, SN-GLYCEROL-3-PHOSPHATE | 著者 | Yun, M, Park, C.-G, Kim, J.-Y, Park, H.-W. | 登録日 | 1999-11-04 | 公開日 | 2000-08-23 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structural analysis of glyceraldehyde 3-phosphate dehydrogenase from Escherichia coli: direct evidence of substrate binding and cofactor-induced conformational changes. Biochemistry, 39, 2000
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1DC5
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1DC6
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![BU of 1dc6 by Molmil](/molmil-images/mine/1dc6) | STRUCTURAL ANALYSIS OF GLYCERALDEHYDE 3-PHOSPHATE DEHYDROGENASE FROM ESCHERICHIA COLI: DIRECT EVIDENCE FOR SUBSTRATE BINDING AND COFACTOR-INDUCED CONFORMATIONAL CHANGES. | 分子名称: | GLYCERALDEHYDE-3-PHOSPHATE DEHYDROGENASE, NICOTINAMIDE-ADENINE-DINUCLEOTIDE | 著者 | Yun, M, Park, C.-G, Kim, J.-Y, Park, H.-W. | 登録日 | 1999-11-04 | 公開日 | 2000-08-23 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structural analysis of glyceraldehyde 3-phosphate dehydrogenase from Escherichia coli: direct evidence of substrate binding and cofactor-induced conformational changes. Biochemistry, 39, 2000
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2X1I
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![BU of 2x1i by Molmil](/molmil-images/mine/2x1i) | glycoside hydrolase family 77 4-alpha-glucanotransferase from thermus brockianus | 分子名称: | 1,2,3,4,5,6-HEXAHYDROXY-CYCLOHEXANE, 4-ALPHA-GLUCANOTRANSFERASE, PHOSPHATE ION, ... | 著者 | Yoon, S.-M, Jung, J.-H, Jung, T.-Y, Song, H.-N, Park, C.-S, Woo, E.-J. | 登録日 | 2009-12-28 | 公開日 | 2010-10-27 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.36 Å) | 主引用文献 | Structural and Functional Analysis of Substrate Recognition by the 250S Loop in Amylomaltase from Thermus Brockianus. Proteins, 79, 2011
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6E6J
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![BU of 6e6j by Molmil](/molmil-images/mine/6e6j) | BRD2_Bromodomain2 complex with inhibitor 744 | 分子名称: | Bromodomain-containing protein 2, N-ethyl-4-[2-(4-fluoro-2,6-dimethylphenoxy)-5-(2-hydroxypropan-2-yl)phenyl]-6-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridine-2-carboxamide | 著者 | Longenecker, K.L, Park, C.H, Bigelow, L. | 登録日 | 2018-07-25 | 公開日 | 2019-07-31 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.44 Å) | 主引用文献 | Selective inhibition of the BD2 bromodomain of BET proteins in prostate cancer. Nature, 578, 2020
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8JB9
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7YON
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![BU of 7yon by Molmil](/molmil-images/mine/7yon) | Complex structure of Neuropeptide Y Y2 receptor in complex with PYY(3-36) and Gi | 分子名称: | Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1, Guanine nucleotide-binding protein G(i) subunit alpha-1, ... | 著者 | Kang, H, Park, C, Kim, J, Choi, H.-J. | 登録日 | 2022-08-01 | 公開日 | 2023-03-22 | 実験手法 | ELECTRON MICROSCOPY (2.95 Å) | 主引用文献 | Structural basis for Y2 receptor-mediated neuropeptide Y and peptide YY signaling. Structure, 31, 2023
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7YOO
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![BU of 7yoo by Molmil](/molmil-images/mine/7yoo) | Complex structure of Neuropeptide Y Y2 receptor in complex with NPY and Gi | 分子名称: | Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1, Guanine nucleotide-binding protein G(i) subunit alpha-1, ... | 著者 | Kang, H, Park, C, Kim, J, Choi, H.-J. | 登録日 | 2022-08-01 | 公開日 | 2023-03-22 | 実験手法 | ELECTRON MICROSCOPY (3.11 Å) | 主引用文献 | Structural basis for Y2 receptor-mediated neuropeptide Y and peptide YY signaling. Structure, 31, 2023
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