4JDM
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![BU of 4jdm by Molmil](/molmil-images/mine/4jdm) | Secreted Chlamydial Protein PGP3, full-length | 分子名称: | Virulence plasmid protein pGP3-D | 著者 | Galaleldeen, A, Taylor, A.B, Chen, D, Holloway, S.P, Zhong, G, Hart, P.J. | 登録日 | 2013-02-25 | 公開日 | 2013-06-05 | 最終更新日 | 2013-10-09 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Structure of the Chlamydia trachomatis immunodominant antigen Pgp3. J.Biol.Chem., 288, 2013
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4JFH
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![BU of 4jfh by Molmil](/molmil-images/mine/4jfh) | High Affinity alpha24-beta17 T Cell Receptor for A2 HLA-Melanoma peptide complex | 分子名称: | 1,2-ETHANEDIOL, GLYCEROL, SULFATE ION, ... | 著者 | Rizkallah, P.J, Cole, D.K, Madura, F, Sewell, A.K. | 登録日 | 2013-02-28 | 公開日 | 2013-05-29 | 最終更新日 | 2013-07-17 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | T-cell receptor specificity maintained by altered thermodynamics. J.Biol.Chem., 288, 2013
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5US1
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![BU of 5us1 by Molmil](/molmil-images/mine/5us1) | Crystal structure of aminoglycoside acetyltransferase AAC(2')-Ia in complex with N2'-acetylgentamicin C1A and coenzyme A | 分子名称: | (1R,2S,3S,4R,6S)-4,6-diamino-3-{[3-deoxy-4-C-methyl-3-(methylamino)-beta-L-arabinopyranosyl]oxy}-2-hydroxycyclohexyl 2-(acetylamino)-6-amino-2,3,4,6-tetradeoxy-alpha-D-erythro-hexopyranoside, ACETYL COENZYME *A, Aminoglycoside 2'-N-acetyltransferase, ... | 著者 | Stogios, P.J, Evdokimova, E, Xu, Z, Wawrzak, Z, Savchenko, A, Anderson, W.F, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2017-02-13 | 公開日 | 2017-03-15 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.48 Å) | 主引用文献 | Plazomicin Retains Antibiotic Activity against Most Aminoglycoside Modifying Enzymes. ACS Infect Dis, 4, 2018
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5UXC
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![BU of 5uxc by Molmil](/molmil-images/mine/5uxc) | Crystal structure of macrolide 2'-phosphotransferase MphH from Brachybacterium faecium in complex with GDP | 分子名称: | AZITHROMYCIN, CHLORIDE ION, GLYCEROL, ... | 著者 | Stogios, P.J, Skarina, T, Wawrzak, Z, Yim, V, Savchenko, A, Anderson, W.F, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2017-02-22 | 公開日 | 2017-08-16 | 最終更新日 | 2019-12-11 | 実験手法 | X-RAY DIFFRACTION (1.72 Å) | 主引用文献 | The evolution of substrate discrimination in macrolide antibiotic resistance enzymes. Nat Commun, 9, 2018
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4JDS
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![BU of 4jds by Molmil](/molmil-images/mine/4jds) | SETD7 in complex with inhibitor PF-5426 and S-adenosyl-methionine | 分子名称: | Histone-lysine N-methyltransferase SETD7, N-[(2R)-3-(3-cyanophenyl)-1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-8-fluoro-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide, S-ADENOSYLMETHIONINE, ... | 著者 | Dong, A, Wu, H, Zeng, H, Park, H, El Bakkouri, M, Barsyte, D, Vedadi, M, Tatlock, J, Owen, D, Bunnage, M, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Brown, P.J, Structural Genomics Consortium (SGC) | 登録日 | 2013-02-25 | 公開日 | 2013-03-27 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | SETD7 in complex with inhibitor PF-5426 and S-adenosyl-methionine to be published
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5V0Z
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![BU of 5v0z by Molmil](/molmil-images/mine/5v0z) | Crystal structure of Galactoside O-acetyltransferase complex with CoA (P32 space group). | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, COENZYME A, ... | 著者 | Czub, M.P, Porebski, P.J, Knapik, A.A, Niedzialkowska, E, Anderson, W.F, Minor, W, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2017-02-28 | 公開日 | 2017-03-15 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.26 Å) | 主引用文献 | Crystal structure of Galactoside O-acetyltransferase complex with CoA (P32 space group). to be published
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4JFP
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![BU of 4jfp by Molmil](/molmil-images/mine/4jfp) | A2 HLA complex with G4A heteroclitic variant of Melanoma peptide | 分子名称: | 1,2-ETHANEDIOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Beta-2-microglobulin, ... | 著者 | Rizkallah, P.J, Cole, D.K, Madura, F, Sewell, A.K. | 登録日 | 2013-02-28 | 公開日 | 2013-05-29 | 最終更新日 | 2013-07-17 | 実験手法 | X-RAY DIFFRACTION (1.91 Å) | 主引用文献 | T-cell receptor specificity maintained by altered thermodynamics. J.Biol.Chem., 288, 2013
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5UXB
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![BU of 5uxb by Molmil](/molmil-images/mine/5uxb) | Crystal structure of macrolide 2'-phosphotransferase MphH from Brachybacterium faecium, apoenzyme | 分子名称: | CHLORIDE ION, Macrolide 2'-phosphotransferase MphH | 著者 | Stogios, P.J, Skarina, T, Yim, V, Savchenko, A, Anderson, W.F, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2017-02-22 | 公開日 | 2017-07-26 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.794 Å) | 主引用文献 | The evolution of substrate discrimination in macrolide antibiotic resistance enzymes. Nat Commun, 9, 2018
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4IQG
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![BU of 4iqg by Molmil](/molmil-images/mine/4iqg) | Crystal structure of BPRO0239 oxidoreductase from Polaromonas sp. JS666 in NADP bound form | 分子名称: | DI(HYDROXYETHYL)ETHER, FORMIC ACID, GLYCEROL, ... | 著者 | Niedzialkowska, E, Majorek, K.A, Porebski, P.J, Al Obaidi, N, Hammonds, J, Hillerich, B, Seidel, R, Bonanno, J.B, Almo, S.C, Minor, W, New York Structural Genomics Research Consortium (NYSGRC) | 登録日 | 2013-01-11 | 公開日 | 2013-01-30 | 最終更新日 | 2022-04-13 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Crystal structure of oxidoreductase from Polaromonas sp. in NADP bound form To be Published
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1QBY
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![BU of 1qby by Molmil](/molmil-images/mine/1qby) | THE SOLUTION STRUCTURE OF A BAY-REGION 1R-BENZ[A]ANTHRACENE OXIDE ADDUCT AT THE N6 POSITION OF ADENINE OF AN OLIGODEOXYNUCLEOTIDE CONTAINING THE HUMAN N-RAS CODON 61 SEQUENCE | 分子名称: | 1R,2S,3R,4S-TETRAHYDRO-BENZO[A]ANTHRACENE-2,3,4-TRIOL, 5'-D(*CP*GP*GP*AP*CP*(BZA)AP*AP*GP*AP*AP*G)-3', 5'-D(*CP*TP*TP*CP*TP*TP*GP*TP*CP*CP* G)-3' | 著者 | Li, Z, Mao, H, Kim, H.-Y, Tamura, P.J, Harris, C.M, Harris, T.M, Stone, M.P. | 登録日 | 1999-04-27 | 公開日 | 1999-05-06 | 最終更新日 | 2022-03-02 | 実験手法 | SOLUTION NMR | 主引用文献 | Intercalation of the (-)-(1R,2S,3R, 4S)-N6-[1-benz[a]anthracenyl]-2'-deoxyadenosyl adduct in an oligodeoxynucleotide containing the human N-ras codon 61 sequence. Biochemistry, 38, 1999
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5THR
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![BU of 5thr by Molmil](/molmil-images/mine/5thr) | |
4QL5
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![BU of 4ql5 by Molmil](/molmil-images/mine/4ql5) | Crystal structure of translation initiation factor IF-1 from Streptococcus pneumoniae TIGR4 | 分子名称: | ACETATE ION, GLYCEROL, Translation initiation factor IF-1, ... | 著者 | Stogios, P.J, Wawrzak, Z, Onopriyenko, O, Savchenko, A, Anderson, W.F, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2014-06-10 | 公開日 | 2014-07-02 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.025 Å) | 主引用文献 | Crystal structure of translation initiation factor IF-1 from Streptococcus pneumoniae TIGR4 TO BE PUBLISHED
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5TDO
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![BU of 5tdo by Molmil](/molmil-images/mine/5tdo) | |
4QOK
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![BU of 4qok by Molmil](/molmil-images/mine/4qok) | Structural basis for ineffective T-cell responses to MHC anchor residue improved heteroclitic peptides | 分子名称: | 1,2-ETHANEDIOL, Beta-2-microglobulin, HLA class I histocompatibility antigen, ... | 著者 | Rizkallah, P.J, Cole, D.K, Madura, F, Sewell, A.K. | 登録日 | 2014-06-20 | 公開日 | 2014-12-17 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structural basis for ineffective T-cell responses to MHC anchor residue-improved "heteroclitic" peptides. Eur.J.Immunol., 45, 2015
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5TIV
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![BU of 5tiv by Molmil](/molmil-images/mine/5tiv) | Schistosoma haematobium (Blood Fluke) Sulfotransferase | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ADENOSINE-3'-5'-DIPHOSPHATE, Sulfotransferase | 著者 | Taylor, A.B, Hart, P.J. | 登録日 | 2016-10-03 | 公開日 | 2017-05-31 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.43 Å) | 主引用文献 | Structural and enzymatic insights into species-specific resistance to schistosome parasite drug therapy. J. Biol. Chem., 292, 2017
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4RYL
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![BU of 4ryl by Molmil](/molmil-images/mine/4ryl) | Human Protein Arginine Methyltransferase 3 in complex with 1-isoquinolin-6-yl-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]urea | 分子名称: | 1-isoquinolin-6-yl-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]urea, PRMT3 protein, UNKNOWN ATOM OR ION | 著者 | Dong, A, Dobrovetsky, E, Kaniskan, H.U, Szewczyk, M, Yu, Z, Eram, M.S, Yang, X, Schmidt, K, Luo, X, Dai, M, He, F, Zang, I, Lin, Y, Kennedy, S, Li, F, Tempel, W, Smil, D, Min, S.J, Landon, M, Lin-Jones, J, Huang, X.P, Roth, B.L, Schapira, M, Atadja, P, Barsyte-Lovejoy, D, Bountra, C, Edwards, A.M, Arrowsmith, C.H, Brown, P.J, Zhao, K, Jin, J, Vedadi, M, Structural Genomics Consortium (SGC) | 登録日 | 2014-12-15 | 公開日 | 2015-02-25 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | A Potent, Selective and Cell-Active Allosteric Inhibitor of Protein Arginine Methyltransferase 3 (PRMT3). Angew.Chem.Int.Ed.Engl., 54, 2015
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1PP7
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![BU of 1pp7 by Molmil](/molmil-images/mine/1pp7) | Crystal structure of the T. vaginalis Initiator binding protein bound to the ferredoxin Inr | 分子名称: | 39 kDa initiator binding protein, FERREDOXIN INR, ZINC ION | 著者 | Schumacher, M.A, Lau, A.O.T, Johnson, P.J. | 登録日 | 2003-06-16 | 公開日 | 2003-11-18 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Structural Basis of Core Promoter Recognition in a Primitive Eukaryote Cell(Cambridge,Mass.), 115, 2003
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5TEY
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![BU of 5tey by Molmil](/molmil-images/mine/5tey) | Human METTL3-METTL14 complex | 分子名称: | 1,2-ETHANEDIOL, BETA-MERCAPTOETHANOL, MAGNESIUM ION, ... | 著者 | DONG, A, ZENG, H, LI, Y, TEMPEL, W, Seitova, A, Hutchinson, A, Bountra, C, Arrowsmith, C.H, Edwards, A.M, BROWN, P.J, WU, H, Structural Genomics Consortium (SGC) | 登録日 | 2016-09-23 | 公開日 | 2016-11-23 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Human METTL3-METTL14 complex to be published
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1PPO
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![BU of 1ppo by Molmil](/molmil-images/mine/1ppo) | DETERMINATION OF THE STRUCTURE OF PAPAYA PROTEASE OMEGA | 分子名称: | MERCURY (II) ION, PROTEASE OMEGA | 著者 | Pickersgill, R.W, Rizkallah, P.J, Harris, G.W, Goodenough, P.W. | 登録日 | 1991-07-12 | 公開日 | 1993-10-31 | 最終更新日 | 2017-11-29 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Determination of the Structure of Papaya Protease Omega Acta Crystallogr.,Sect.B, 47, 1991
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1PVX
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![BU of 1pvx by Molmil](/molmil-images/mine/1pvx) | DO-1,4-BETA-XYLANASE, ROOM TEMPERATURE, PH 4.5 | 分子名称: | PROTEIN (ENDO-1,4-BETA-XYLANASE) | 著者 | Rajeshkumar, P, Eswaramoorthy, S, Vithayathil, P.J, Viswamitra, M.A. | 登録日 | 1998-10-20 | 公開日 | 1999-10-20 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.59 Å) | 主引用文献 | The tertiary structure at 1.59 A resolution and the proposed amino acid sequence of a family-11 xylanase from the thermophilic fungus Paecilomyces varioti bainier. J.Mol.Biol., 295, 2000
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5TIY
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![BU of 5tiy by Molmil](/molmil-images/mine/5tiy) | Schistosoma haematobium (Blood Fluke) Sulfotransferase/S-oxamniquine Complex | 分子名称: | ADENOSINE-3'-5'-DIPHOSPHATE, Sulfotransferase, {(2S)-7-nitro-2-[(propan-2-ylamino)methyl]-1,2,3,4-tetrahydroquinolin-6-yl}methanol | 著者 | Taylor, A.B, Hart, P.J. | 登録日 | 2016-10-03 | 公開日 | 2017-05-31 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.76 Å) | 主引用文献 | Structural and enzymatic insights into species-specific resistance to schistosome parasite drug therapy. J. Biol. Chem., 292, 2017
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4J8A
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![BU of 4j8a by Molmil](/molmil-images/mine/4j8a) | Irradiated-state structure of sfGFP containing the unnatural amino acid p-azido-phenylalanine at residue 145 | 分子名称: | 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Green fluorescent protein, ... | 著者 | Reddington, S.C, Jones, D.D, Rizkallah, P.J, Tippmann, E.M. | 登録日 | 2013-02-14 | 公開日 | 2013-05-15 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (1.26 Å) | 主引用文献 | Different Photochemical Events of a Genetically Encoded Phenyl Azide Define and Modulate GFP Fluorescence. Angew.Chem.Int.Ed.Engl., 52, 2013
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1Q3T
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![BU of 1q3t by Molmil](/molmil-images/mine/1q3t) | Solution structure and function of an essential CMP kinase of Streptococcus pneumoniae | 分子名称: | Cytidylate kinase | 著者 | Yu, L, Mack, J, Hajduk, P.J, Kakavas, S.J, Saiki, A.Y, Lerner, C.G, Olejniczak, E.T. | 登録日 | 2003-07-31 | 公開日 | 2004-08-03 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure and function of an essential CMP kinase of Streptococcus pneumoniae Protein Sci., 12, 2003
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5UWL
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![BU of 5uwl by Molmil](/molmil-images/mine/5uwl) | Matrix metalloproteinase-13 complexed with selective inhibitor compound (S)-17a | 分子名称: | (S)-N-(3-methyl-1-(methylamino)-1-oxobutan-2-yl)-5-(4-(((4-oxo-4,5,6,7-tetrahydro-3H-cyclopenta[d]pyrimidin-2-yl)thio)methyl)phenyl)furan-2-carboxamide, CALCIUM ION, Collagenase 3, ... | 著者 | Taylor, A.B, Cao, X, Hart, P.J. | 登録日 | 2017-02-21 | 公開日 | 2017-07-12 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.55 Å) | 主引用文献 | Structure-Based Design and Synthesis of Potent and Selective Matrix Metalloproteinase 13 Inhibitors. J. Med. Chem., 60, 2017
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4JFO
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![BU of 4jfo by Molmil](/molmil-images/mine/4jfo) | A2 HLA complex with E1A heteroclitic variant of Melanoma peptide | 分子名称: | Beta-2-microglobulin, E1A heteroclitic Melanoma peptide, GLYCEROL, ... | 著者 | Rizkallah, P.J, Cole, D.K, Madura, F, Sewell, A.K, Baker, B.M. | 登録日 | 2013-02-28 | 公開日 | 2013-05-29 | 最終更新日 | 2013-07-17 | 実験手法 | X-RAY DIFFRACTION (2.11 Å) | 主引用文献 | T-cell receptor specificity maintained by altered thermodynamics. J.Biol.Chem., 288, 2013
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