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5US1

Crystal structure of aminoglycoside acetyltransferase AAC(2')-Ia in complex with N2'-acetylgentamicin C1A and coenzyme A

Summary for 5US1
Entry DOI10.2210/pdb5us1/pdb
Related6C0C
DescriptorAminoglycoside 2'-N-acetyltransferase, (1R,2S,3S,4R,6S)-4,6-diamino-3-{[3-deoxy-4-C-methyl-3-(methylamino)-beta-L-arabinopyranosyl]oxy}-2-hydroxycyclohexyl 2-(acetylamino)-6-amino-2,3,4,6-tetradeoxy-alpha-D-erythro-hexopyranoside, D(-)-TARTARIC ACID, ... (7 entities in total)
Functional Keywordsgnat, gcn5-n-acetyltransferase, acetyltransferase, aminoglycoside, gentamicin, coenzyme a, acetylcoenzyme a antibiotic resistance, structural genomics, center for structural genomics of infectious diseases, csgid, national institute of allergy and infectious diseases, niaid, transferase
Biological sourceProvidencia stuartii
Total number of polymer chains12
Total formula weight263334.07
Authors
Stogios, P.J.,Evdokimova, E.,Xu, Z.,Wawrzak, Z.,Savchenko, A.,Anderson, W.F.,Center for Structural Genomics of Infectious Diseases (CSGID) (deposition date: 2017-02-13, release date: 2017-03-15, Last modification date: 2023-10-04)
Primary citationCox, G.,Ejim, L.,Stogios, P.J.,Koteva, K.,Bordeleau, E.,Evdokimova, E.,Sieron, A.O.,Savchenko, A.,Serio, A.W.,Krause, K.M.,Wright, G.D.
Plazomicin Retains Antibiotic Activity against Most Aminoglycoside Modifying Enzymes.
ACS Infect Dis, 4:980-987, 2018
Cited by
PubMed: 29634241
DOI: 10.1021/acsinfecdis.8b00001
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.48 Å)
Structure validation

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