7O9T
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7O9Z
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7O9X
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7OA9
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3K7Y
| Aspartate Aminotransferase of Plasmodium falciparum | 分子名称: | ACETATE ION, Aspartate aminotransferase, PYRIDOXAL-5'-PHOSPHATE | 著者 | Groves, M.R, Jordanova, R, Jain, R, Wrenger, C, Muller, I.B. | 登録日 | 2009-10-13 | 公開日 | 2010-10-13 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Specific Inhibition of the Aspartate Aminotransferase of Plasmodium falciparum. J.Mol.Biol., 405, 2011
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1PCI
| PROCARICAIN | 分子名称: | PROCARICAIN | 著者 | Groves, M.R, Taylor, M.A.J, Scott, M, Cummings, N.J, Pickersgill, R.W, Jenkins, J.A. | 登録日 | 1996-06-28 | 公開日 | 1997-04-01 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | The prosequence of procaricain forms an alpha-helical domain that prevents access to the substrate-binding cleft. Structure, 4, 1996
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2OB1
| ppm1 with 1,8-ANS | 分子名称: | Leucine carboxyl methyltransferase 1, PHOSPHATE ION | 著者 | Groves, M.R. | 登録日 | 2006-12-18 | 公開日 | 2007-01-30 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | A method for the general identification of protein crystals in crystallization experiments using a noncovalent fluorescent dye. Acta Crystallogr.,Sect.D, 63, 2007
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2OB2
| ppm1 in the absence of 1,8-ANS (cf 1JD) | 分子名称: | GLYCEROL, Leucine carboxyl methyltransferase 1, PHOSPHATE ION, ... | 著者 | Groves, M.R, Mueller, I.B, Kreplin, X, Mueller-Dieckmann, J. | 登録日 | 2006-12-18 | 公開日 | 2007-01-30 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.92 Å) | 主引用文献 | A method for the general identification of protein crystals in crystallization experiments using a noncovalent fluorescent dye. Acta Crystallogr.,Sect.D, 63, 2007
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1BZJ
| Human ptp1b complexed with tpicooh | 分子名称: | 6-(DIFLUORO-PHOSPHONO-METHYL)-NAPHTHALENE-2-CARBOXYLIC ACID, PROTEIN (PROTEIN-TYROSINE-PHOSPHATASE) | 著者 | Groves, M.R, Yao, Z.-J, Barford Jr, D.T.B. | 登録日 | 1998-10-29 | 公開日 | 1999-02-16 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Structural basis for inhibition of the protein tyrosine phosphatase 1B by phosphotyrosine peptide mimetics. Biochemistry, 37, 1998
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1BZC
| HUMAN PTP1B CATALYTIC DOMAIN COMPLEXED WITH TPI | 分子名称: | 4-CARBAMOYL-4-{[6-(DIFLUORO-PHOSPHONO-METHYL)-NAPHTHALENE-2-CARBONYL]-AMINO}-BUTYRIC ACID, PROTEIN (PROTEIN-TYROSINE-PHOSPHATASE) | 著者 | Groves, M.R, Yao, Z.J, Jr Burke, T.R, Barford, D. | 登録日 | 1998-10-27 | 公開日 | 1999-02-16 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Structural basis for inhibition of the protein tyrosine phosphatase 1B by phosphotyrosine peptide mimetics. Biochemistry, 37, 1998
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1B3U
| CRYSTAL STRUCTURE OF CONSTANT REGULATORY DOMAIN OF HUMAN PP2A, PR65ALPHA | 分子名称: | PROTEIN (PROTEIN PHOSPHATASE PP2A) | 著者 | Groves, M.R, Hanlon, N, Turowski, P, Hemmings, B, Barford, D. | 登録日 | 1998-12-14 | 公開日 | 1999-04-12 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | The structure of the protein phosphatase 2A PR65/A subunit reveals the conformation of its 15 tandemly repeated HEAT motifs. Cell(Cambridge,Mass.), 96, 1999
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1BZH
| Cyclic peptide inhibitor of human PTP1B | 分子名称: | PROTEIN (PROTEIN-TYROSINE-PHOSPHATASE 1B INHIBITOR), PROTEIN (PROTEIN-TYROSINE-PHOSPHATASE 1B) | 著者 | Groves, M.R, Yao, Z.J, Burke Jr, T.R, Barford, D. | 登録日 | 1998-10-28 | 公開日 | 1999-02-16 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structural basis for inhibition of the protein tyrosine phosphatase 1B by phosphotyrosine peptide mimetics. Biochemistry, 37, 1998
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1CZI
| CHYMOSIN COMPLEX WITH THE INHIBITOR CP-113972 | 分子名称: | CHYMOSIN, CP-113972 (NORSTATINE-S-METHYL CYSTEINE-IODO-PHENYLALANINE-PROLINE) | 著者 | Groves, M.R, Dhanaraj, V, Pitts, J.E, Badasso, M, Hoover, D, Nugent, P, Blundell, T.L. | 登録日 | 1997-01-15 | 公開日 | 1997-04-01 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | A 2.3 A resolution structure of chymosin complexed with a reduced bond inhibitor shows that the active site beta-hairpin flap is rearranged when compared with the native crystal structure. Protein Eng., 11, 1998
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6SKV
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6SKS
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6SKT
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6SU9
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6S2K
| Human Menin in complex with AJ21 | 分子名称: | Multiple endocrine neoplasia I, isoform CRA_b, ~{N}-[2-(4-methoxyphenyl)ethyl]-2-(4-nitrophenyl)imidazo[1,2-a]pyridin-3-amine | 著者 | Groves, M.R, Gao, K. | 登録日 | 2019-06-21 | 公開日 | 2021-01-13 | 最終更新日 | 2024-05-15 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Human Menin in complex with AJ21 To Be Published
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8AGF
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3L1P
| POU protein:DNA complex | 分子名称: | DNA (5'-D(*AP*TP*CP*CP*AP*TP*TP*TP*GP*CP*CP*TP*TP*TP*CP*AP*AP*AP*TP*GP*TP*GP*G)-3'), DNA (5'-D(*TP*CP*CP*AP*CP*AP*TP*TP*TP*GP*AP*AP*AP*GP*GP*CP*AP*AP*AP*TP*GP*GP*A)-3'), POU domain, ... | 著者 | Vahokoski, J, Groves, M.R, Pogenberg, V, Wilmanns, M. | 登録日 | 2009-12-14 | 公開日 | 2010-12-15 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | A unique Oct4 interface is crucial for reprogramming to pluripotency Nat.Cell Biol., 15, 2013
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6HL7
| Crystal structure of truncated aspartate transcarbamoylase from Plasmodium falciparum with mutated active site (R109A/K138A) and N-carbamoyl-L-phosphate bound | 分子名称: | Aspartate transcarbamoylase, PHOSPHORIC ACID MONO(FORMAMIDE)ESTER | 著者 | Bosch, S.S, Lunev, S, Wrenger, C, Groves, M.R. | 登録日 | 2018-09-10 | 公開日 | 2018-09-26 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Molecular Target Validation of Aspartate Transcarbamoylase fromPlasmodium falciparumby Torin 2. Acs Infect Dis., 6, 2020
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6ZRU
| Crystal structure of SARS CoV2 main protease in complex with inhibitor Boceprevir | 分子名称: | DIMETHYL SULFOXIDE, Main Protease, boceprevir (bound form) | 著者 | Oerlemans, R, Wang, W, Lunev, S, Domling, A, Groves, M.R. | 登録日 | 2020-07-14 | 公開日 | 2020-08-12 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Repurposing the HCV NS3-4A protease drug boceprevir as COVID-19 therapeutics. Rsc Med Chem, 12, 2020
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8R2H
| Cryo-EM structure of 1-deoxy-D-xylulose 5-phosphate synthase (DXPS) from Plasmodium falciparum | 分子名称: | 1-deoxy-D-xylulose-5-phosphate synthase, MAGNESIUM ION, THIAMINE DIPHOSPHATE | 著者 | Gawriljuk, V.O, Godoy, A.S, Oerlemans, R, Groves, M.R. | 登録日 | 2023-11-06 | 公開日 | 2024-06-12 | 最終更新日 | 2024-08-14 | 実験手法 | ELECTRON MICROSCOPY (2.42 Å) | 主引用文献 | Cryo-EM structure of 1-deoxy-D-xylulose 5-phosphate synthase DXPS from Plasmodium falciparum reveals a distinct N-terminal domain. Nat Commun, 15, 2024
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8Q5Z
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6FBA
| Crystal Structure of truncated aspartate transcarbamoylase from Plasmodium falciparum with bound inhibitor 2,3-naphthalenediol | 分子名称: | Aspartate transcarbamoylase, DI(HYDROXYETHYL)ETHER, DIMETHYL SULFOXIDE, ... | 著者 | Lunev, S, Bosch, S.S, Batista, F.A, Wang, C, Wrenger, C, Groves, M.R. | 登録日 | 2017-12-18 | 公開日 | 2018-02-21 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Identification of a non-competitive inhibitor of Plasmodium falciparum aspartate transcarbamoylase. Biochem. Biophys. Res. Commun., 497, 2018
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