4LXF
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![BU of 4lxf by Molmil](/molmil-images/mine/4lxf) | Crystal structure of M. tuberculosis TreS | Descriptor: | CALCIUM ION, GLYCEROL, SULFATE ION, ... | Authors: | Roy, R, Besra, G.S, Futterer, K. | Deposit date: | 2013-07-29 | Release date: | 2013-08-21 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (2.6 Å) | Cite: | Synthesis of alpha-glucan in mycobacteria involves a hetero-octameric complex of trehalose synthase TreS and Maltokinase Pep2. Acs Chem.Biol., 8, 2013
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3OKP
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![BU of 3okp by Molmil](/molmil-images/mine/3okp) | Crystal structure of Corynebacterium glutamicum PimB' bound to GDP-Man (orthorhombic crystal form) | Descriptor: | GDP-mannose-dependent alpha-(1-6)-phosphatidylinositol monomannoside mannosyltransferase, GUANOSINE-5'-DIPHOSPHATE-ALPHA-D-MANNOSE | Authors: | Batt, S.M, Jabeen, T, Besra, G.S, Futterer, K. | Deposit date: | 2010-08-25 | Release date: | 2010-09-15 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Acceptor substrate discrimination in phosphatidyl-myo-inositol mannoside synthesis: structural and mutational analysis of mannosyltransferase Corynebacterium glutamicum PimB'. J.Biol.Chem., 285, 2010
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3OKA
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![BU of 3oka by Molmil](/molmil-images/mine/3oka) | Crystal structure of Corynebacterium glutamicum PimB' in complex with GDP-Man (triclinic crystal form) | Descriptor: | GDP-mannose-dependent alpha-(1-6)-phosphatidylinositol monomannoside mannosyltransferase, GLYCEROL, GUANOSINE-5'-DIPHOSPHATE-ALPHA-D-MANNOSE, ... | Authors: | Batt, S.M, Jabeen, T, Besra, G.S, Futterer, K. | Deposit date: | 2010-08-24 | Release date: | 2010-09-15 | Last modified: | 2024-02-21 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Acceptor substrate discrimination in phosphatidyl-myo-inositol mannoside synthesis: structural and mutational analysis of mannosyltransferase Corynebacterium glutamicum PimB'. J.Biol.Chem., 285, 2010
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3OKC
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![BU of 3okc by Molmil](/molmil-images/mine/3okc) | Crystal structure of Corynebacterium glutamicum PimB' bound to GDP (orthorhombic crystal form) | Descriptor: | GDP-mannose-dependent alpha-(1-6)-phosphatidylinositol monomannoside mannosyltransferase, GUANOSINE-5'-DIPHOSPHATE | Authors: | Batt, S.M, Jabeen, T, Besra, G.S, Futterer, K. | Deposit date: | 2010-08-24 | Release date: | 2010-09-15 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (2.4 Å) | Cite: | Acceptor substrate discrimination in phosphatidyl-myo-inositol mannoside synthesis: structural and mutational analysis of mannosyltransferase Corynebacterium glutamicum PimB'. J.Biol.Chem., 285, 2010
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1B7X
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![BU of 1b7x by Molmil](/molmil-images/mine/1b7x) | STRUCTURE OF HUMAN ALPHA-THROMBIN Y225I MUTANT BOUND TO D-PHE-PRO-ARG-CHLOROMETHYLKETONE | Descriptor: | PROTEIN (INHIBITOR), PROTEIN (THROMBIN HEAVY CHAIN), PROTEIN (THROMBIN LIGHT CHAIN) | Authors: | Caccia, S, Futterer, K, Di Cera, E, Waksman, G. | Deposit date: | 1999-01-25 | Release date: | 1999-03-02 | Last modified: | 2023-08-09 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | Unexpected crucial role of residue 225 in serine proteases. Proc.Natl.Acad.Sci.USA, 96, 1999
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2Q74
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![BU of 2q74 by Molmil](/molmil-images/mine/2q74) | Mycobacterium tuberculosis SuhB | Descriptor: | Inositol-1-monophosphatase | Authors: | Brown, A.K, Meng, G, Ghadbane, H, Besra, G.S, Futterer, K. | Deposit date: | 2007-06-06 | Release date: | 2007-10-23 | Last modified: | 2023-08-30 | Method: | X-RAY DIFFRACTION (2.6 Å) | Cite: | Dimerization of inositol monophosphatase Mycobacterium tuberculosis SuhB is not constitutive, but induced by binding of the activator Mg2+ Bmc Struct.Biol., 7, 2007
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2QJ3
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![BU of 2qj3 by Molmil](/molmil-images/mine/2qj3) | Mycobacterium tuberculosis FabD | Descriptor: | Malonyl CoA-acyl carrier protein transacylase, NICKEL (II) ION | Authors: | Ghadbane, H, Brown, A.K, Kremer, L, Besra, G.S, Futterer, K. | Deposit date: | 2007-07-06 | Release date: | 2007-09-04 | Last modified: | 2011-07-13 | Method: | X-RAY DIFFRACTION (3 Å) | Cite: | Structure of Mycobacterium tuberculosis mtFabD, a malonyl-CoA:acyl carrier protein transacylase (MCAT). Acta Crystallogr.,Sect.F, 63, 2007
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2THF
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![BU of 2thf by Molmil](/molmil-images/mine/2thf) | STRUCTURE OF HUMAN ALPHA-THROMBIN Y225F MUTANT BOUND TO D-PHE-PRO-ARG-CHLOROMETHYLKETONE | Descriptor: | D-phenylalanyl-N-[(2S,3S)-6-{[amino(iminio)methyl]amino}-1-chloro-2-hydroxyhexan-3-yl]-L-prolinamide, SODIUM ION, THROMBIN HEAVY CHAIN, ... | Authors: | Caccia, S, Futterer, K, Di Cera, E, Waksman, G. | Deposit date: | 1999-01-26 | Release date: | 1999-03-07 | Last modified: | 2023-08-30 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | Unexpected crucial role of residue 225 in serine proteases. Proc.Natl.Acad.Sci.USA, 96, 1999
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1R88
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![BU of 1r88 by Molmil](/molmil-images/mine/1r88) | The crystal structure of Mycobacterium tuberculosis MPT51 (FbpC1) | Descriptor: | MPT51/MPB51 antigen | Authors: | Wilson, R.A, Maughan, W.N, Kremer, L, Besra, G.S, Futterer, K. | Deposit date: | 2003-10-23 | Release date: | 2003-12-30 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (1.71 Å) | Cite: | The structure of Mycobacterium tuberculosis MPT51 (FbpC1) defines a new family of non-catalytic alpha/beta hydrolases. J.Mol.Biol., 335, 2004
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3PTY
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![BU of 3pty by Molmil](/molmil-images/mine/3pty) | Crystal structure of the C-terminal extracellular domain of Mycobacterium tuberculosis EmbC | Descriptor: | Arabinosyltransferase C, CALCIUM ION, PHOSPHATE ION, ... | Authors: | Alderwick, L.J, Besra, G.S, Futterer, K. | Deposit date: | 2010-12-03 | Release date: | 2010-12-15 | Last modified: | 2020-07-29 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | The C-Terminal Domain of the Arabinosyltransferase Mycobacterium tuberculosis EmbC Is a Lectin-Like Carbohydrate Binding Module. Plos Pathog., 7, 2011
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1PT2
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![BU of 1pt2 by Molmil](/molmil-images/mine/1pt2) | |
1OYG
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![BU of 1oyg by Molmil](/molmil-images/mine/1oyg) | |
6HRD
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![BU of 6hrd by Molmil](/molmil-images/mine/6hrd) | |
4FF6
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![BU of 4ff6 by Molmil](/molmil-images/mine/4ff6) | Mycobacterium tuberculosis DprE1 in complex with CT325 - monoclinic crystal form | Descriptor: | 3-(hydroxyamino)-N-[(1R)-1-phenylethyl]-5-(trifluoromethyl)benzamide, FLAVIN-ADENINE DINUCLEOTIDE, IMIDAZOLE, ... | Authors: | Batt, S.M, Besra, G.S, Futterer, K. | Deposit date: | 2012-05-31 | Release date: | 2012-07-04 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (2.6 Å) | Cite: | Structural basis of inhibition of Mycobacterium tuberculosis DprE1 by benzothiazinone inhibitors. Proc.Natl.Acad.Sci.USA, 109, 2012
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4FDN
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![BU of 4fdn by Molmil](/molmil-images/mine/4fdn) | |
4FDP
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![BU of 4fdp by Molmil](/molmil-images/mine/4fdp) | |
4FDO
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![BU of 4fdo by Molmil](/molmil-images/mine/4fdo) | Mycobacterium tuberculosis DprE1 in complex with CT319 | Descriptor: | 3-nitro-N-[(1R)-1-phenylethyl]-5-(trifluoromethyl)benzamide, FLAVIN-ADENINE DINUCLEOTIDE, oxidoreductase DprE1 | Authors: | Batt, S.M, Besra, G.S, Futterer, K. | Deposit date: | 2012-05-29 | Release date: | 2012-07-04 | Last modified: | 2024-04-03 | Method: | X-RAY DIFFRACTION (2.403 Å) | Cite: | Structural basis of inhibition of Mycobacterium tuberculosis DprE1 by benzothiazinone inhibitors. Proc.Natl.Acad.Sci.USA, 109, 2012
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4FEH
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![BU of 4feh by Molmil](/molmil-images/mine/4feh) | |
5DU8
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![BU of 5du8 by Molmil](/molmil-images/mine/5du8) | Crystal structure of M. tuberculosis EchA6 bound to GSK572A | Descriptor: | (5R,7S)-5-(4-ethylphenyl)-N-[(5-fluoropyridin-2-yl)methyl]-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide, Probable enoyl-CoA hydratase echA6 | Authors: | Cox, J.A.G, Besra, G.S, Futterer, K. | Deposit date: | 2015-09-18 | Release date: | 2016-01-20 | Last modified: | 2024-01-10 | Method: | X-RAY DIFFRACTION (2.23 Å) | Cite: | THPP target assignment reveals EchA6 as an essential fatty acid shuttle in mycobacteria. Nat Microbiol, 1, 2016
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5DUC
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![BU of 5duc by Molmil](/molmil-images/mine/5duc) | Crystal structure of M. tuberculosis EchA6 bound to ligand GSK951A | Descriptor: | (5R,7S)-N-(1,3-benzodioxol-5-ylmethyl)-5-(4-ethylphenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide, Probable enoyl-CoA hydratase echA6 | Authors: | Cox, J.A.G, Besra, G.S, Futterer, K. | Deposit date: | 2015-09-18 | Release date: | 2016-01-20 | Last modified: | 2024-01-10 | Method: | X-RAY DIFFRACTION (2.704 Å) | Cite: | THPP target assignment reveals EchA6 as an essential fatty acid shuttle in mycobacteria. Nat Microbiol, 1, 2016
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5DUF
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![BU of 5duf by Molmil](/molmil-images/mine/5duf) | Crystal structure of M. tuberculosis EchA6 bound to ligand GSK729A | Descriptor: | (5R,7S)-5-(4-ethylphenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylic acid, Probable enoyl-CoA hydratase echA6 | Authors: | Cox, J.A.G, Besra, G.S, Futterer, K. | Deposit date: | 2015-09-18 | Release date: | 2016-01-20 | Last modified: | 2024-01-10 | Method: | X-RAY DIFFRACTION (1.5 Å) | Cite: | THPP target assignment reveals EchA6 as an essential fatty acid shuttle in mycobacteria. Nat Microbiol, 1, 2016
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5DU6
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![BU of 5du6 by Molmil](/molmil-images/mine/5du6) | Crystal structure of M. tuberculosis EchA6 bound to ligand GSK059A. | Descriptor: | (5R,7R)-5-(4-ethylphenyl)-N-(4-fluorobenzyl)-7-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide, Probable enoyl-CoA hydratase echA6 | Authors: | Cox, J.A.G, Besra, G.S, Futterer, K. | Deposit date: | 2015-09-18 | Release date: | 2016-01-20 | Last modified: | 2024-01-10 | Method: | X-RAY DIFFRACTION (2.61 Å) | Cite: | THPP target assignment reveals EchA6 as an essential fatty acid shuttle in mycobacteria. Nat Microbiol, 1, 2016
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5DTP
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![BU of 5dtp by Molmil](/molmil-images/mine/5dtp) | |
5DU4
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![BU of 5du4 by Molmil](/molmil-images/mine/5du4) | Crystal structure of M. tuberculosis EchA6 bound to ligand GSK366A | Descriptor: | (5R,7S)-5-(4-ethylphenyl)-N-(4-methoxybenzyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide, Probable enoyl-CoA hydratase echA6 | Authors: | Cox, J.A.G, Besra, G.S, Futterer, K. | Deposit date: | 2015-09-18 | Release date: | 2016-01-20 | Last modified: | 2024-01-10 | Method: | X-RAY DIFFRACTION (1.702 Å) | Cite: | THPP target assignment reveals EchA6 as an essential fatty acid shuttle in mycobacteria. Nat Microbiol, 1, 2016
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5DTW
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![BU of 5dtw by Molmil](/molmil-images/mine/5dtw) | |