5KWZ
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7RAZ
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![BU of 7raz by Molmil](/molmil-images/mine/7raz) | Small conductance mechanosensitive channel MscS | 分子名称: | PHOSPHATIDYLETHANOLAMINE, Small-conductance mechanosensitive channel | 著者 | Catalano, C, Ben-Hail, D, Qiu, W, des Georges, A, Guo, Y. | 登録日 | 2021-07-05 | 公開日 | 2022-07-13 | 最終更新日 | 2024-06-05 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Small conductance mechanosensitive channel MscS To Be Published
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6UNN
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5KZT
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![BU of 5kzt by Molmil](/molmil-images/mine/5kzt) | Listeria monocytogenes OppA bound to peptide | 分子名称: | Hexamer peptide: SER-ASP-GLU-SER-LYS-GLY, Hexamer peptide: SER-ASP-GLU-SER-SER-GLY, Peptide/nickel transport system substrate-binding protein | 著者 | Light, S.H, Whiteley, A.T, Minasov, G, Portnoy, D.A, Anderson, W.F, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2016-07-25 | 公開日 | 2016-08-10 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Listeria monocytogenes OppA bound to peptide To Be Published
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5AZ7
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6TXW
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![BU of 6txw by Molmil](/molmil-images/mine/6txw) | V30G Transthyretin structure in complex with Tolcalpone | 分子名称: | Tolcapone, Transthyretin | 著者 | Varejao, N, Reverter, D, Pinheiro, F, Pallares, I, Ventura, S. | 登録日 | 2020-01-14 | 公開日 | 2020-05-13 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.153 Å) | 主引用文献 | Tolcapone, a potent aggregation inhibitor for the treatment of familial leptomeningeal amyloidosis. Febs J., 288, 2021
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6QNA
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![BU of 6qna by Molmil](/molmil-images/mine/6qna) | Structure of bovine anti-RSV hybrid Fab B13HC-B4LC | 分子名称: | B13 Heavy chain, B4 light chain, GLYCEROL | 著者 | Ren, J, Nettleship, J.E, Harris, G, Mwangi, W, Rhaman, N, Grant, C, Kotecha, A, Fry, E, Charleston, B, Stuart, D.I, Hammond, J, Owens, R.J. | 登録日 | 2019-02-10 | 公開日 | 2019-05-29 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.62 Å) | 主引用文献 | The role of the light chain in the structure and binding activity of two cattle antibodies that neutralize bovine respiratory syncytial virus. Mol.Immunol., 112, 2019
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7R6R
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![BU of 7r6r by Molmil](/molmil-images/mine/7r6r) | Crystal Structure of a Mycobacteriophage Cluster A2 Immunity Repressor:DNA Complex | 分子名称: | DNA (5'-D(P*CP*CP*CP*GP*CP*TP*TP*GP*AP*CP*AP*GP*CP*CP*AP*CP*CP*GP*AP*AP*A)-3'), DNA (5'-D(P*TP*TP*TP*CP*GP*GP*TP*GP*GP*CP*TP*GP*TP*CP*AP*AP*GP*CP*GP*GP*G)-3'), Immunity repressor | 著者 | McGinnis, R.J, Brambley, C.A, Stamey, B, Green, W.C, Gragg, K.N, Cafferty, E.R, Terwilliger, T.C, Hammel, M, Hollis, T.J, Miller, J.M, Gainey, M.D, Wallen, J.R. | 登録日 | 2021-06-23 | 公開日 | 2022-07-20 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (3.13 Å) | 主引用文献 | A monomeric mycobacteriophage immunity repressor utilizes two domains to recognize an asymmetric DNA sequence. Nat Commun, 13, 2022
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6ES0
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![BU of 6es0 by Molmil](/molmil-images/mine/6es0) | Crystal structure of the kinase domain of human RIPK2 in complex with the activation loop targeting inhibitor CS-R35 | 分子名称: | 2-[2-fluoranyl-4-[[2-fluoranyl-4-[2-(methylcarbamoyl)pyridin-4-yl]oxy-phenyl]carbamoylamino]phenyl]sulfanylethanoic acid, Receptor-interacting serine/threonine-protein kinase 2 | 著者 | Pinkas, D.M, Bufton, J.C, Suebsuwong, C, Ray, S.S, Dai, B, Newman, J.A, Burgess-Brown, N.A, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Degterev, A, Cuny, G.D, Bullock, A.N. | 登録日 | 2017-10-19 | 公開日 | 2018-02-21 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.38 Å) | 主引用文献 | Activation loop targeting strategy for design of receptor-interacting protein kinase 2 (RIPK2) inhibitors. Bioorg. Med. Chem. Lett., 28, 2018
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6EBG
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![BU of 6ebg by Molmil](/molmil-images/mine/6ebg) | Ohr (Organic Hydroperoxide Resistance protein) mutant - C60S interacting with dihydrolipoamide | 分子名称: | (6S)-6,8-disulfanyloctanamide, Organic hydroperoxide resistance protein | 著者 | Domingos, R.M, Teixeira, R.D, Alegria, T.G.P, Vieira, P.S, Murakami, M.T, Netto, L.E.S. | 登録日 | 2018-08-06 | 公開日 | 2020-02-05 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Substrate and product-assisted catalysis: molecular aspects behind structural switches along Organic Hydroperoxide Resistance Protein catalytic cycle Acs Catalysis, 2020
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5IGH
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5IGV
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6ECD
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![BU of 6ecd by Molmil](/molmil-images/mine/6ecd) | Vlm2 thioesterase domain with genetically encoded 2,3-diaminopropionic acid bound with a tetradepsipeptide | 分子名称: | Vlm2, tetradepsipeptide | 著者 | Alonzo, D.A, Huguenin-Dezot, N, Heberlig, G.W, Mahesh, M, Nguyen, D.P, Dornan, M.H, Boddy, C.N, Chin, J.W, Schmeing, T.M. | 登録日 | 2018-08-07 | 公開日 | 2018-12-12 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Trapping biosynthetic acyl-enzyme intermediates with encoded 2,3-diaminopropionic acid. Nature, 565, 2019
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8EBM
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6U1Z
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7UHB
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5IH1
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6EE7
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![BU of 6ee7 by Molmil](/molmil-images/mine/6ee7) | Small tetraheme cytochrome c from Shewanella oneidensis | 分子名称: | HEME C, Periplasmic tetraheme cytochrome c CctA, ZINC ION | 著者 | Huang, J, Zarzycki, J, Ducat, D.C, Kramer, D.M. | 登録日 | 2018-08-13 | 公開日 | 2019-08-14 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.394 Å) | 主引用文献 | Mesoscopic to Macroscopic Electron Transfer by Hopping in a Crystal Network of Cytochromes. J.Am.Chem.Soc., 142, 2020
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5XF1
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![BU of 5xf1 by Molmil](/molmil-images/mine/5xf1) | Structure of the Full-length glucagon class B G protein-coupled receptor | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Zhang, H, Qiao, A, Yang, D, Yang, L, Dai, A, de Graaf, C, Reedtz-Runge, S, Dharmarajan, V, Zhang, H, Han, G.W, Grant, T, Sierra, R, Weierstall, U, Nelson, G, Liu, W, Wu, Y, Ma, L, Cai, X, Lin, G, Wu, X, Geng, Z, Dong, Y, Song, G, Griffin, P, Lau, J, Cherezov, V, Yang, H, Hanson, M, Stevens, R, Jiang, H, Wang, M, Zhao, Q, Wu, B. | 登録日 | 2017-04-06 | 公開日 | 2017-05-24 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (3.19 Å) | 主引用文献 | Structure of the full-length glucagon class B G-protein-coupled receptor. Nature, 546, 2017
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8SFA
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![BU of 8sfa by Molmil](/molmil-images/mine/8sfa) | Crystal structure of the engineered SsoPox variant IIIC1 | 分子名称: | Aryldialkylphosphatase, COBALT (II) ION, FE (III) ION | 著者 | Jacquet, P, Billot, R, Shimon, A, Hoekstra, N, Bergonzi, C, Jenks, A, Daude, D, Elias, M.H. | 登録日 | 2023-04-10 | 公開日 | 2024-04-17 | 実験手法 | X-RAY DIFFRACTION (2.32 Å) | 主引用文献 | Changes in Active Site Loops Conformation Relates to a Transition from Lactonase to Phosphotriesterase To Be Published
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7V6Z
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![BU of 7v6z by Molmil](/molmil-images/mine/7v6z) | Cryo-EM structure of Patched1 (V1084A mutant) in lipid nanodisc, 3.64 angstrom (reprocessed with the dataset of 7dzp) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CHOLESTEROL, ... | 著者 | Luo, Y, Zhao, Y, Qu, Q, Li, D. | 登録日 | 2021-08-20 | 公開日 | 2021-09-22 | 最終更新日 | 2022-02-16 | 実験手法 | ELECTRON MICROSCOPY (3.64 Å) | 主引用文献 | Cryo-EM study of patched in lipid nanodisc suggests a structural basis for its clustering in caveolae. Structure, 29, 2021
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8GMK
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![BU of 8gmk by Molmil](/molmil-images/mine/8gmk) | Pyruvate bound structure of Citrate Synthase (CitA) in Mycobacterium Tuberculosis | 分子名称: | 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, PYRUVIC ACID, ... | 著者 | Pathirage, R, Ronning, D, Yamsek, M. | 登録日 | 2023-03-26 | 公開日 | 2023-06-07 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.81 Å) | 主引用文献 | Mycobacterium tuberculosis CitA activity is modulated by cysteine oxidation and pyruvate binding. Rsc Med Chem, 14, 2023
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8EBL
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6WMQ
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8IZZ
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![BU of 8izz by Molmil](/molmil-images/mine/8izz) | |