1WO1
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![BU of 1wo1 by Molmil](/molmil-images/mine/1wo1) | |
1WO0
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![BU of 1wo0 by Molmil](/molmil-images/mine/1wo0) | |
4BWS
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![BU of 4bws by Molmil](/molmil-images/mine/4bws) | Crystal structure of the heterotrimer of PQBP1, U5-15kD and U5-52kD. | Descriptor: | CD2 ANTIGEN CYTOPLASMIC TAIL-BINDING PROTEIN 2, POLYGLUTAMINE-BINDING PROTEIN 1, THIOREDOXIN-LIKE PROTEIN 4A | Authors: | Mizuguchi, M, Obita, T, Serita, T, Kojima, R, Morimoto, T, Nabeshima, Y, Okazawa, H. | Deposit date: | 2013-07-04 | Release date: | 2014-04-30 | Last modified: | 2023-12-20 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Mutations in the Pqbp1 Gene Prevent its Interaction with the Spliceosomal Protein U5-15Kd. Nat.Commun., 5, 2014
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4CDO
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![BU of 4cdo by Molmil](/molmil-images/mine/4cdo) | Crystal structure of PQBP1 bound to spliceosomal U5-15kD | Descriptor: | THIOREDOXIN-LIKE PROTEIN 4A, POLYGLUTAMINE-BINDING PROTEIN | Authors: | Mizuguchi, M, Obita, T, Serita, T, Kojima, R, Nabeshima, Y, Okazawa, H. | Deposit date: | 2013-11-05 | Release date: | 2014-04-30 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Mutations in the Pqbp1 Gene Prevent its Interaction with the Spliceosomal Protein U5-15Kd. Nat.Commun., 5, 2014
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4BWQ
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![BU of 4bwq by Molmil](/molmil-images/mine/4bwq) | Crystal structure of U5-15kD in a complex with PQBP1 | Descriptor: | POLYGLUTAMINE-BINDING PROTEIN 1, THIOREDOXIN-LIKE PROTEIN 4A | Authors: | Mizuguchi, M, Obita, T, Serita, T, Kojima, R, Morimoto, T, Nabeshima, Y, Okazawa, H. | Deposit date: | 2013-07-04 | Release date: | 2014-04-30 | Last modified: | 2023-12-20 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | Mutations in the Pqbp1 Gene Prevent its Interaction with the Spliceosomal Protein U5-15Kd. Nat.Commun., 5, 2014
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8JOK
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![BU of 8jok by Molmil](/molmil-images/mine/8jok) | |
8JNU
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![BU of 8jnu by Molmil](/molmil-images/mine/8jnu) | |
8JQW
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![BU of 8jqw by Molmil](/molmil-images/mine/8jqw) | |
7W9Q
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![BU of 7w9q by Molmil](/molmil-images/mine/7w9q) | Crystal structure of V30M-TTR in complex with naringenin derivative-14 | Descriptor: | (2~{R})-2-(3-chloranyl-4-oxidanyl-phenyl)-5,7-bis(oxidanyl)-2,3-dihydrochromen-4-one, CALCIUM ION, Transthyretin | Authors: | Katayama, W, Shimane, A, Nabeshima, Y, Yokoyama, T, Mizuguchi, M. | Deposit date: | 2021-12-10 | Release date: | 2022-12-14 | Last modified: | 2023-11-29 | Method: | X-RAY DIFFRACTION (1.599 Å) | Cite: | Chlorinated Naringenin Analogues as Potential Inhibitors of Transthyretin Amyloidogenesis. J.Med.Chem., 65, 2022
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7W9R
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![BU of 7w9r by Molmil](/molmil-images/mine/7w9r) | Crystal structure of V30M-TTR in complex with naringenin derivative-18 | Descriptor: | (2~{R})-2-[3,5-bis(chloranyl)-4-oxidanyl-phenyl]-5,7-bis(oxidanyl)-2,3-dihydrochromen-4-one, Transthyretin | Authors: | Katayama, W, Shimane, A, Nabeshima, Y, Yokoyama, T, Mizuguchi, M. | Deposit date: | 2021-12-10 | Release date: | 2022-12-14 | Last modified: | 2023-11-29 | Method: | X-RAY DIFFRACTION (1.997 Å) | Cite: | Chlorinated Naringenin Analogues as Potential Inhibitors of Transthyretin Amyloidogenesis. J.Med.Chem., 65, 2022
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8I76
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![BU of 8i76 by Molmil](/molmil-images/mine/8i76) | |
8I75
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![BU of 8i75 by Molmil](/molmil-images/mine/8i75) | |
8I74
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![BU of 8i74 by Molmil](/molmil-images/mine/8i74) | |
1WRU
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![BU of 1wru by Molmil](/molmil-images/mine/1wru) | Structure of central hub elucidated by X-ray analysis of gene product 44; baseplate component of bacteriophage Mu | Descriptor: | 43 kDa tail protein | Authors: | Kondou, Y, Kitazawa, D, Takeda, S, Yamashita, E, Mizuguchi, M, Kawano, K, Tsukihara, T. | Deposit date: | 2004-10-27 | Release date: | 2005-09-20 | Last modified: | 2024-03-13 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | Structure of central hub elucidated by X-ray analysis of gene product 44; baseplate component of bacteriophage Mu To be Published
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4N87
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![BU of 4n87 by Molmil](/molmil-images/mine/4n87) | Crystal structure of V30M mutant human transthyretin complexed with glabridin | Descriptor: | 4-[(3R)-8,8-dimethyl-3,4-dihydro-2H,8H-pyrano[2,3-f]chromen-3-yl]benzene-1,3-diol, Transthyretin | Authors: | Yokoyama, T, Kosaka, Y, Mizuguchi, M. | Deposit date: | 2013-10-17 | Release date: | 2014-02-19 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (1.794 Å) | Cite: | Crystal structures of human transthyretin complexed with glabridin J.Med.Chem., 57, 2014
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4N85
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![BU of 4n85 by Molmil](/molmil-images/mine/4n85) | |
4N86
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![BU of 4n86 by Molmil](/molmil-images/mine/4n86) | Crystal structure of human transthyretin complexed with glabridin | Descriptor: | 4-[(3R)-8,8-dimethyl-3,4-dihydro-2H,8H-pyrano[2,3-f]chromen-3-yl]benzene-1,3-diol, CALCIUM ION, Transthyretin | Authors: | Yokoyama, T, Kosaka, Y, Mizuguchi, M. | Deposit date: | 2013-10-17 | Release date: | 2014-02-19 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (2.001 Å) | Cite: | Crystal structures of human transthyretin complexed with glabridin J.Med.Chem., 57, 2014
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2MDB
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![BU of 2mdb by Molmil](/molmil-images/mine/2mdb) | Tachyplesin I in the presence of lipopolysaccharide | Descriptor: | Tachyplesin-1 | Authors: | Kushibiki, T, Kamiya, M, Aizawa, T, Kumaki, Y, Kikukawa, T, Mizuguchi, M, Demura, M, Kawabata, S.I, Kawano, K. | Deposit date: | 2013-09-09 | Release date: | 2014-02-19 | Last modified: | 2023-06-14 | Method: | SOLUTION NMR | Cite: | Interaction between tachyplesin I, an antimicrobial peptide derived from horseshoe crab, and lipopolysaccharide. Biochim.Biophys.Acta, 1844, 2014
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5X2L
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![BU of 5x2l by Molmil](/molmil-images/mine/5x2l) | Crystal Structure of Human Serine Racemase | Descriptor: | MAGNESIUM ION, PYRIDOXAL-5'-PHOSPHATE, Serine racemase | Authors: | Obita, T, Matsumoto, K, Mori, H, Toyooka, N, Mizuguchi, M. | Deposit date: | 2017-02-01 | Release date: | 2018-01-31 | Last modified: | 2021-02-24 | Method: | X-RAY DIFFRACTION (1.806 Å) | Cite: | Design, synthesis, and evaluation of novel inhibitors for wild-type human serine racemase. Bioorg. Med. Chem. Lett., 2017
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7WL6
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![BU of 7wl6 by Molmil](/molmil-images/mine/7wl6) | |
2RTV
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![BU of 2rtv by Molmil](/molmil-images/mine/2rtv) | Tachyplesin I in water | Descriptor: | Tachyplesin-1 | Authors: | Kushibiki, T, Kamiya, M, Aizawa, T, Kumaki, Y, Kikukawa, T, Mizuguchi, M, Demura, M, Kawabata, S.I, Kawano, K. | Deposit date: | 2013-09-19 | Release date: | 2014-02-19 | Last modified: | 2023-06-14 | Method: | SOLUTION NMR | Cite: | Interaction between tachyplesin I, an antimicrobial peptide derived from horseshoe crab, and lipopolysaccharide. Biochim.Biophys.Acta, 1844, 2014
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2RNG
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![BU of 2rng by Molmil](/molmil-images/mine/2rng) | Solution structure of big defensin | Descriptor: | Big defensin | Authors: | Kouno, T, Fujitani, N, Osaki, T, Kawabata, S, Nishimura, S, Mizuguchi, M, Aizawa, T, Demura, M, Nitta, K, Kawano, K. | Deposit date: | 2007-12-27 | Release date: | 2008-10-14 | Last modified: | 2023-06-14 | Method: | SOLUTION NMR | Cite: | A novel beta-defensin structure: a potential strategy of big defensin for overcoming resistance by Gram-positive bacteria Biochemistry, 47, 2008
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2RQ2
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![BU of 2rq2 by Molmil](/molmil-images/mine/2rq2) | The solution structure of the N-terminal fragment of big defensin | Descriptor: | Big defensin | Authors: | Kouno, T, Mizuguchi, M, Aizawa, T, Shinoda, H, Demura, M, Kawabata, S, Kawano, K. | Deposit date: | 2009-01-07 | Release date: | 2009-08-25 | Last modified: | 2024-05-15 | Method: | SOLUTION NMR | Cite: | A novel beta-defensin structure: big defensin changes its N-terminal structure to associate with the target membrane Biochemistry, 48, 2009
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5AON
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![BU of 5aon by Molmil](/molmil-images/mine/5aon) | Crystal structure of the conserved N-terminal domain of Pex14 from Trypanosoma brucei | Descriptor: | PEROXIN 14, SULFATE ION | Authors: | Obita, T, Sugawara, Y, Mizuguchi, M, Watanabe, Y, Kawaguchi, K, Imanaka, T. | Deposit date: | 2015-09-11 | Release date: | 2015-12-23 | Last modified: | 2024-01-10 | Method: | X-RAY DIFFRACTION (1.646 Å) | Cite: | Characterization of the Interaction between Trypanosoma Brucei Pex5P and its Receptor Pex14P. FEBS Lett., 590, 2016
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6AA4
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![BU of 6aa4 by Molmil](/molmil-images/mine/6aa4) | Crystal structure of MTH1 in complex with alpha-mangostin (cocktail No. 9) | Descriptor: | 1,3,6-trihydroxy-7-methoxy-2,8-bis(3-methylbut-2-en-1-yl)-9H-xanthen-9-one, 7,8-dihydro-8-oxoguanine triphosphatase, SULFATE ION, ... | Authors: | Yokoyama, T, Kitakami, R, Mizuguchi, M. | Deposit date: | 2018-07-17 | Release date: | 2019-03-06 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Discovery of a new class of MTH1 inhibitor by X-ray crystallographic screening. Eur J Med Chem, 167, 2019
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