5NIJ
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![BU of 5nij by Molmil](/molmil-images/mine/5nij) | |
5O7E
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![BU of 5o7e by Molmil](/molmil-images/mine/5o7e) | |
5NZC
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![BU of 5nzc by Molmil](/molmil-images/mine/5nzc) | |
5NZB
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![BU of 5nzb by Molmil](/molmil-images/mine/5nzb) | |
5OBT
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![BU of 5obt by Molmil](/molmil-images/mine/5obt) | |
2Y6I
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![BU of 2y6i by Molmil](/molmil-images/mine/2y6i) | |
2Y3U
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![BU of 2y3u by Molmil](/molmil-images/mine/2y3u) | |
2Y50
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4AWA
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![BU of 4awa by Molmil](/molmil-images/mine/4awa) | Crystal structure of active legumain in complex with YVAD-CMK at pH 5.0 | Descriptor: | 2-acetamido-2-deoxy-beta-D-glucopyranose, LEGUMAIN, SULFATE ION, ... | Authors: | Dall, E, Brandstetter, H. | Deposit date: | 2012-06-01 | Release date: | 2013-06-26 | Last modified: | 2023-12-20 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Mechanistic and Structural Studies on Legumain Explain its Zymogenicity, Distinct Activation Pathways, and Regulation Proc.Natl.Acad.Sci.USA, 110, 2013
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4B9R
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![BU of 4b9r by Molmil](/molmil-images/mine/4b9r) | |
4AWB
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![BU of 4awb by Molmil](/molmil-images/mine/4awb) | Crystal structure of active legumain in complex with AAN-CMK | Descriptor: | 2-acetamido-2-deoxy-beta-D-glucopyranose, LEGUMAIN, MERCURY (II) ION, ... | Authors: | Dall, E, Brandstetter, H. | Deposit date: | 2012-06-01 | Release date: | 2013-06-26 | Last modified: | 2023-12-20 | Method: | X-RAY DIFFRACTION (2.7 Å) | Cite: | Mechanistic and Structural Studies on Legumain Explain its Zymogenicity, Distinct Activation Pathways, and Regulation Proc.Natl.Acad.Sci.USA, 110, 2013
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4BKC
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![BU of 4bkc by Molmil](/molmil-images/mine/4bkc) | |
4BK7
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![BU of 4bk7 by Molmil](/molmil-images/mine/4bk7) | |
4BK6
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![BU of 4bk6 by Molmil](/molmil-images/mine/4bk6) | |
4BKD
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![BU of 4bkd by Molmil](/molmil-images/mine/4bkd) | |
4BTZ
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![BU of 4btz by Molmil](/molmil-images/mine/4btz) | |
1JH1
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![BU of 1jh1 by Molmil](/molmil-images/mine/1jh1) | Crystal Structure of MMP-8 complexed with a 6H-1,3,4-thiadiazine derived inhibitor | Descriptor: | BUT-3-ENYL-[5-(4-CHLORO-PHENYL)-3,6-DIHYDRO-[1,3,4]THIADIAZIN-2-YLIDENE]-AMINE, CALCIUM ION, Matrix Metalloproteinase 8, ... | Authors: | Schroder, J, Henke, A, Wenzel, H, Brandstetter, H, Stammler, H.G, Stammler, A, Pfeiffer, W.D, Tschesche, H. | Deposit date: | 2001-06-27 | Release date: | 2001-12-27 | Last modified: | 2024-04-03 | Method: | X-RAY DIFFRACTION (2.7 Å) | Cite: | Structure-based design and synthesis of potent matrix metalloproteinase inhibitors derived from a 6H-1,3,4-thiadiazine scaffold. J.Med.Chem., 44, 2001
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1J2Q
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![BU of 1j2q by Molmil](/molmil-images/mine/1j2q) | 20S proteasome in complex with calpain-Inhibitor I from archaeoglobus fulgidus | Descriptor: | 2-ACETYLAMINO-4-METHYL-PENTANOIC ACID [1-(1-FORMYL-PENTYLCARBAMOYL)-3-METHYL-BUTYL]-AMIDE, Proteasome alpha subunit, Proteasome beta subunit | Authors: | Groll, M, Brandstetter, H, Bartunik, H, Bourenkow, G, Huber, R. | Deposit date: | 2003-01-08 | Release date: | 2003-03-18 | Last modified: | 2023-12-27 | Method: | X-RAY DIFFRACTION (2.83 Å) | Cite: | Investigations on the Maturation and Regulation of Archaebacterial Proteasomes J.MOL.BIOL., 327, 2003
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1ITV
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![BU of 1itv by Molmil](/molmil-images/mine/1itv) | Dimeric form of the haemopexin domain of MMP9 | Descriptor: | MMP9, SULFATE ION | Authors: | Cha, H, Kopetzki, E, Huber, R, Lanzendoerfer, M, Brandstetter, H. | Deposit date: | 2002-02-11 | Release date: | 2002-09-04 | Last modified: | 2023-12-27 | Method: | X-RAY DIFFRACTION (1.95 Å) | Cite: | Structural basis of the adaptive molecular recognition by MMP9. J.Mol.Biol., 320, 2002
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1J2P
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![BU of 1j2p by Molmil](/molmil-images/mine/1j2p) | alpha-ring from the proteasome from archaeoglobus fulgidus | Descriptor: | Proteasome alpha subunit | Authors: | Groll, M, Brandstetter, H, Bartunik, H, Bourenkow, G, Huber, R. | Deposit date: | 2003-01-08 | Release date: | 2003-03-18 | Last modified: | 2024-04-03 | Method: | X-RAY DIFFRACTION (2.6 Å) | Cite: | Investigations on the Maturation and Regulation of Archaebacterial Proteasomes J.MOL.BIOL., 327, 2003
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1RFN
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![BU of 1rfn by Molmil](/molmil-images/mine/1rfn) | HUMAN COAGULATION FACTOR IXA IN COMPLEX WITH P-AMINO BENZAMIDINE | Descriptor: | CALCIUM ION, P-AMINO BENZAMIDINE, PROTEIN (COAGULATION FACTOR IX), ... | Authors: | Hopfner, K.-P, Lang, A, Karcher, A, Sichler, K, Kopetzki, E, Brandstetter, H, Huber, R, Bode, W, Engh, R.A. | Deposit date: | 1999-04-19 | Release date: | 1999-09-01 | Last modified: | 2023-12-27 | Method: | X-RAY DIFFRACTION (2.8 Å) | Cite: | Coagulation factor IXa: the relaxed conformation of Tyr99 blocks substrate binding. Structure Fold.Des., 7, 1999
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1S0P
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![BU of 1s0p by Molmil](/molmil-images/mine/1s0p) | Structure of the N-Terminal Domain of the Adenylyl Cyclase-Associated Protein (CAP) from Dictyostelium discoideum. | Descriptor: | Adenylyl cyclase-associated protein, MAGNESIUM ION | Authors: | Ksiazek, D, Brandstetter, H, Israel, L, Bourenkov, G.P, Katchalova, G, Janssen, K.P, Bartunik, H.D, Noegel, A.A, Schleicher, M, Holak, T.A. | Deposit date: | 2004-01-01 | Release date: | 2004-01-27 | Last modified: | 2024-02-14 | Method: | X-RAY DIFFRACTION (1.4 Å) | Cite: | STRUCTURE OF THE N-TERMINAL DOMAIN OF THE ADENYLYL
CYCLASE-ASSOCIATED PROTEIN (CAP) FROM DICTYOSTELIUM DISCOIDEUM Structure, 11, 2003
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1ORW
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![BU of 1orw by Molmil](/molmil-images/mine/1orw) | Crystal Structure of Porcine Dipeptidyl Peptidase IV (CD26) in Complex with a Peptidomimetic Inhibitor | Descriptor: | (2S)-PYRROLIDIN-2-YLMETHYLAMINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | Authors: | Engel, M, Hoffmann, T, Wagner, L, Wermann, M, Heiser, U, Kiefersauer, R, Huber, R, Bode, W, Demuth, H.U, Brandstetter, H. | Deposit date: | 2003-03-16 | Release date: | 2003-05-06 | Last modified: | 2020-07-29 | Method: | X-RAY DIFFRACTION (2.84 Å) | Cite: | The Crystal Structure of Dipeptidyl Peptidase IV (CD26) Reveals its Functional Regulation and Enzymatic Mechanism Proc.Natl.Acad.Sci.USA, 100, 2003
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1N6E
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![BU of 1n6e by Molmil](/molmil-images/mine/1n6e) | tricorn protease in complex with a tridecapeptide chloromethyl ketone derivative | Descriptor: | DQTQKAAAELTFF, Tricorn protease | Authors: | Kim, J.-S, Groll, M, Huber, R, Brandstetter, H. | Deposit date: | 2002-11-10 | Release date: | 2002-12-30 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (2.6 Å) | Cite: | Navigation Inside a Protease: Substrate Selection and Product Exit in the Tricorn Protease
from Thermoplasma acidophilum J.Mol.Biol., 324, 2002
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1N6F
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![BU of 1n6f by Molmil](/molmil-images/mine/1n6f) | tricorn protease in complex with Z-Phe-diketo-Arg-Glu-Phe | Descriptor: | 4-[2-(3-BENZYLOXYCARBONYLAMINO-4-CYCLOHEXYL-1-HYDROXY-2-OXO-BUTYLAMINO)-5-GUANIDINO-PENTANOYLAMINO]-4-(1-CARBOXY-2-CYCLOHEXYL-ETHYLCARBAMOYL)-BUTYRIC ACID, tricorn protease | Authors: | Kim, J.-S, Groll, M, Huber, R, Brandstetter, H. | Deposit date: | 2002-11-10 | Release date: | 2002-12-30 | Last modified: | 2023-10-25 | Method: | X-RAY DIFFRACTION (2.7 Å) | Cite: | Navigation Inside a Protease: Substrate Selection and Product Exit in the Tricorn Protease
from Thermoplasma acidophilum J.Mol.Biol., 324, 2002
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