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Crystal structure of GlpG in complex with peptide boronate inhibitor
分子名称:	ACE-VAL-ARG-MET-B2A, Rhomboid family intramembrane serine protease GlpG
著者	Urban, S, Cho, S.
登録日	2020-01-15
公開日	2020-09-16
最終更新日	2023-11-15
実験手法	X-RAY DIFFRACTION (2.3 Å)
主引用文献	Designed Parasite-Selective Rhomboid Inhibitors Block Invasion and Clear Blood-Stage Malaria. Cell Chem Biol, 27, 2020

6PJQ

Time-resolved structural snapshot of proteolysis by GlpG inside the membrane
分子名称:	Peptide aldehyde inhibitor, Rhomboid protease GlpG
著者	Urban, S, Cho, S.
登録日	2019-06-28
公開日	2019-11-27
最終更新日	2023-10-11
実験手法	X-RAY DIFFRACTION (2.5 Å)
主引用文献	Ten catalytic snapshots of rhomboid intramembrane proteolysis from gate opening to peptide release. Nat.Struct.Mol.Biol., 26, 2019

6PJ7

Time-resolved structural snapshot of proteolysis by GlpG inside the membrane
分子名称:	Peptide aldehyde inhibitor, Rhomboid protease GlpG
著者	Urban, S, Cho, S.
登録日	2019-06-28
公開日	2019-10-02
最終更新日	2023-10-11
実験手法	X-RAY DIFFRACTION (2.3 Å)
主引用文献	Ten catalytic snapshots of rhomboid intramembrane proteolysis from gate opening to peptide release. Nat.Struct.Mol.Biol., 26, 2019

6PJ8

Time-resolved structural snapshot of proteolysis by GlpG inside the membrane
分子名称:	Peptide aldehyde inhibitor, Rhomboid protease GlpG
著者	Urban, S, Cho, S.
登録日	2019-06-28
公開日	2019-10-02
最終更新日	2023-10-11
実験手法	X-RAY DIFFRACTION (2.4 Å)
主引用文献	Ten catalytic snapshots of rhomboid intramembrane proteolysis from gate opening to peptide release. Nat.Struct.Mol.Biol., 26, 2019

6PJP

Time-resolved structural snapshot of proteolysis by GlpG inside the membrane
分子名称:	Peptide aldehyde inhibitor, Rhomboid protease GlpG
著者	Urban, S, Cho, S.
登録日	2019-06-28
公開日	2019-10-02
最終更新日	2023-10-11
実験手法	X-RAY DIFFRACTION (2.45 Å)
主引用文献	Ten catalytic snapshots of rhomboid intramembrane proteolysis from gate opening to peptide release. Nat.Struct.Mol.Biol., 26, 2019

6PJ4

Time-resolved structural snapshot of proteolysis by GlpG inside the membrane
分子名称:	Peptide aldehyde inhibitor, Rhomboid protease GlpG
著者	Urban, S, Cho, S.
登録日	2019-06-27
公開日	2019-10-02
最終更新日	2024-03-13
実験手法	X-RAY DIFFRACTION (2.3 Å)
主引用文献	Ten catalytic snapshots of rhomboid intramembrane proteolysis from gate opening to peptide release. Nat.Struct.Mol.Biol., 26, 2019

6VJ8

Crystal structure of GlpG in complex with peptide chloromethylketone inhibitor
分子名称:	Peptide chloromethylketone inhibitor, Rhomboid family intramembrane serine protease GlpG
著者	Urban, S, Cho, S.
登録日	2020-01-15
公開日	2020-09-16
最終更新日	2023-11-15
実験手法	X-RAY DIFFRACTION (2.3 Å)
主引用文献	Designed Parasite-Selective Rhomboid Inhibitors Block Invasion and Clear Blood-Stage Malaria. Cell Chem Biol, 27, 2020

6XRP

Crystal structure of GlpG in complex with peptide ketoamide inhibitor, Ac-RVWHA-ketoamide-phenylbutyl
分子名称:	N-(4-phenylbutyl)formamide, Rhomboid protease GlpG, peptide ketoamide inhibitor
著者	Urban, S, Cho, S.
登録日	2020-07-13
公開日	2020-09-16
最終更新日	2023-10-18
実験手法	X-RAY DIFFRACTION (2.4 Å)
主引用文献	Designed Parasite-Selective Rhomboid Inhibitors Block Invasion and Clear Blood-Stage Malaria. Cell Chem Biol, 27, 2020

6XRO

Crystal structure of GlpG in complex with peptide boronate inhibitor, Ac-KRFRSMQYSA-B(OH)2
分子名称:	CHLORIDE ION, Rhomboid protease GlpG, SODIUM ION, ...
著者	Urban, S, Cho, S.
登録日	2020-07-13
公開日	2020-09-16
最終更新日	2024-04-24
実験手法	X-RAY DIFFRACTION (2.3 Å)
主引用文献	Designed Parasite-Selective Rhomboid Inhibitors Block Invasion and Clear Blood-Stage Malaria. Cell Chem Biol, 27, 2020

6PJU

Time-resolved structural snapshot of proteolysis by GlpG inside the membrane
分子名称:	Peptide aldehyde inhibitor, Rhomboid protease GlpG
著者	Urban, S, Cho, S.
登録日	2019-06-28
公開日	2019-11-27
最終更新日	2023-10-11
実験手法	X-RAY DIFFRACTION (2.5 Å)
主引用文献	Ten catalytic snapshots of rhomboid intramembrane proteolysis from gate opening to peptide release. Nat.Struct.Mol.Biol., 26, 2019

6PJR

Time-resolved structural snapshot of proteolysis by GlpG inside the membrane
分子名称:	CHLORIDE ION, Peptide aldehyde inhibitor, Rhomboid protease GlpG
著者	Urban, S, Cho, S.
登録日	2019-06-28
公開日	2019-10-02
最終更新日	2023-10-11
実験手法	X-RAY DIFFRACTION (2.4 Å)
主引用文献	Ten catalytic snapshots of rhomboid intramembrane proteolysis from gate opening to peptide release. Nat.Struct.Mol.Biol., 26, 2019

6PJA

Time-resolved structural snapshot of proteolysis by GlpG inside the membrane
分子名称:	Peptide aldehyde inhibitor, Rhomboid protease GlpG
著者	Urban, S, Cho, S.
登録日	2019-06-28
公開日	2019-10-02
最終更新日	2024-03-13
実験手法	X-RAY DIFFRACTION (2.6 Å)
主引用文献	Ten catalytic snapshots of rhomboid intramembrane proteolysis from gate opening to peptide release. Nat.Struct.Mol.Biol., 26, 2019

6PJ5

Time-resolved structural snapshot of proteolysis by GlpG inside the membrane
分子名称:	Peptide aldehyde inhibitor, Rhomboid protease GlpG
著者	Urban, S, Cho, S.
登録日	2019-06-27
公開日	2019-10-02
最終更新日	2023-10-11
実験手法	X-RAY DIFFRACTION (2.4 Å)
主引用文献	Ten catalytic snapshots of rhomboid intramembrane proteolysis from gate opening to peptide release. Nat.Struct.Mol.Biol., 26, 2019

6PJ9

Time-resolved structural snapshot of proteolysis by GlpG inside the membrane
分子名称:	Peptide aldehyde inhibitor, Rhomboid protease GlpG
著者	Urban, S, Cho, S.
登録日	2019-06-28
公開日	2019-10-02
最終更新日	2023-10-11
実験手法	X-RAY DIFFRACTION (2.5 Å)
主引用文献	Ten catalytic snapshots of rhomboid intramembrane proteolysis from gate opening to peptide release. Nat.Struct.Mol.Biol., 26, 2019

5F5J

E.coli GlpG Y205F mutant complexed with aldehyde inhibitor in DMPC/CHAPSO bicelle
分子名称:	Rhomboid protease GlpG, peptidic derivative of Gurken: ACE-VAL-ARG-MET-ALA-aldehyde
著者	Urban, S, Cho, S, Dickey, S.
登録日	2015-12-04
公開日	2016-02-10
最終更新日	2024-07-10
実験手法	X-RAY DIFFRACTION (2.4 Å)
主引用文献	Crystal Structures and Inhibition Kinetics Reveal a Two-Stage Catalytic Mechanism with Drug Design Implications for Rhomboid Proteolysis. Mol.Cell, 61, 2016

5F5B

Structure of E.Coli GlpG complexed with peptidic inhibitor Ac-VRMA-CHO
分子名称:	Rhomboid protease GlpG, peptidic derivative of Gurken: ACE-VAL-ARG-MET-ALA-aldehyde
著者	Urban, S, Cho, S, Dickey, S.W.
登録日	2015-12-04
公開日	2016-02-17
最終更新日	2024-07-10
実験手法	X-RAY DIFFRACTION (2.3 Å)
主引用文献	Crystal Structures and Inhibition Kinetics Reveal a Two-Stage Catalytic Mechanism with Drug Design Implications for Rhomboid Proteolysis. Mol.Cell, 61, 2016

5F5D

Crystal structures and Inhibition kinetics reveal a two-state catalytic mechanism with drug design implications for rhomboid proteolysis
分子名称:	Rhomboid protease GlpG
著者	Urban, S, Cho, S, Dickey, S.W.
登録日	2015-12-04
公開日	2016-02-24
最終更新日	2023-09-27
実験手法	X-RAY DIFFRACTION (2.5 Å)
主引用文献	Crystal Structures and Inhibition Kinetics Reveal a Two-Stage Catalytic Mechanism with Drug Design Implications for Rhomboid Proteolysis. Mol.Cell, 61, 2016

5F5G

Structure of E.Coli GlpG Y205F mutant complexed with peptidic inhibitor Ac-RMA-CHO in the DMPC/CHAPSO bicelle
分子名称:	ACE-ARG-MET-ALA-aldehyde, Rhomboid protease GlpG
著者	Urban, S, Cho, S, Dickey, S.W.
登録日	2015-12-04
公開日	2016-04-06
最終更新日	2024-07-10
実験手法	X-RAY DIFFRACTION (2.3 Å)
主引用文献	Crystal Structures and Inhibition Kinetics Reveal a Two-Stage Catalytic Mechanism with Drug Design Implications for Rhomboid Proteolysis. Mol.Cell, 61, 2016

5F5K

E.Coli GlpG Y205F mutant complexed with aldehyde inhibitor in DMPC/CHAPSO bicelle
分子名称:	Peptidic derivative of Gurken: ACE-ARG-LYS-VAL-ARG-MET-ALA-aldehyde, Rhomboid protease GlpG
著者	Urban, S, Cho, S, Dickey, S.W.
登録日	2015-12-04
公開日	2016-02-10
最終更新日	2024-07-10
実験手法	X-RAY DIFFRACTION (2.4 Å)
主引用文献	Crystal Structures and Inhibition Kinetics Reveal a Two-Stage Catalytic Mechanism with Drug Design Implications for Rhomboid Proteolysis. Mol.Cell, 61, 2016

8RQF

Cryo-EM structure of human NTCP-Bulevirtide complex
分子名称:	Fab-specific nanobody, Heavy chain of Fab3, Light chain of Fab3, ...
著者	Liu, H, Zakrzewicz, D, Nosol, K, Irobalieva, R.N, Mukherjee, S, Bang-Soerensen, R, Goldmann, N, Kunz, S, Rossi, L, Kossiakoff, A.A, Urban, S, Glebe, D, Geyer, J, Locher, K.P.
登録日	2024-01-18
公開日	2024-03-27
実験手法	ELECTRON MICROSCOPY (3.41 Å)
主引用文献	Cryo-EM structure of human NTCP-Bulevirtide complex To Be Published

4NJN

Crystal Structure of E.coli GlpG at pH 4.5
分子名称:	Rhomboid protease GlpG
著者	Dickey, S.W, Baker, R.P, Cho, S, Urban, S.
登録日	2013-11-11
公開日	2013-12-25
最終更新日	2023-09-20
実験手法	X-RAY DIFFRACTION (2.4 Å)
主引用文献	Proteolysis inside the Membrane Is a Rate-Governed Reaction Not Driven by Substrate Affinity. Cell(Cambridge,Mass.), 155, 2013

4NJP

Proteolysis inside the membrane is a rate-governed reaction not Driven by substrate affinity
分子名称:	Rhomboid protease GlpG
著者	Dickey, S.W, Baker, R.P, Cho, S, Urban, S.
登録日	2013-11-11
公開日	2013-12-25
最終更新日	2023-09-20
実験手法	X-RAY DIFFRACTION (2.4 Å)
主引用文献	Proteolysis inside the Membrane Is a Rate-Governed Reaction Not Driven by Substrate Affinity. Cell(Cambridge,Mass.), 155, 2013

5AFW

Assembly of methylated LSD1 and CHD1 drives AR-dependent transcription and translocation
分子名称:	1,2-ETHANEDIOL, CHLORIDE ION, CHROMODOMAIN-HELICASE-DNA-BINDING PROTEIN 1, ...
著者	Metzger, E, Willmann, D, McMillan, J, Petroll, K, Metzger, P, Gerhardt, S, vonMaessenhausen, A, Schott, A.K, Espejo, A, Eberlin, A, Wohlwend, D, Schuele, K.M, Schleicher, M, Perner, S, Bedford, M.T, Dengjel, J, Flaig, R, Einsle, O, Schuele, R.
登録日	2015-01-26
公開日	2016-01-13
最終更新日	2024-01-10
実験手法	X-RAY DIFFRACTION (1.6 Å)
主引用文献	Assembly of Methylated Kdm1A and Chd1 Drives Androgen Receptor-Dependent Transcription and Translocation. Nat.Struct.Mol.Biol., 23, 2016

6H1E

Crystal structure of C21orf127-TRMT112 in complex with SAH and H4 peptide
分子名称:	HemK methyltransferase family member 2, Histone H4 peptide, Multifunctional methyltransferase subunit TRM112-like protein, ...
著者	Wang, S, Hermann, B, Metzger, E, Peng, L, Einsle, O, Schuele, R.
登録日	2018-07-11
公開日	2019-05-22
最終更新日	2024-01-17
実験手法	X-RAY DIFFRACTION (1.9 Å)
主引用文献	KMT9 monomethylates histone H4 lysine 12 and controls proliferation of prostate cancer cells. Nat.Struct.Mol.Biol., 26, 2019

6H1D

Crystal structure of C21orf127-TRMT112 in complex with SAH
分子名称:	HemK methyltransferase family member 2, Multifunctional methyltransferase subunit TRM112-like protein, S-ADENOSYL-L-HOMOCYSTEINE
著者	Wang, S, Hermann, B, Metzger, E, Peng, L, Einsle, O, Schuele, R.
登録日	2018-07-11
公開日	2019-05-22
最終更新日	2024-01-17
実験手法	X-RAY DIFFRACTION (1.94 Å)
主引用文献	KMT9 monomethylates histone H4 lysine 12 and controls proliferation of prostate cancer cells. Nat.Struct.Mol.Biol., 26, 2019

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全ヒット件数:	28
表示件数:	25
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