6VJ9
Crystal structure of GlpG in complex with peptide boronate inhibitor
Summary for 6VJ9
Entry DOI | 10.2210/pdb6vj9/pdb |
Related PRD ID | PRD_002373 |
Descriptor | Rhomboid family intramembrane serine protease GlpG, ACE-VAL-ARG-MET-B2A (3 entities in total) |
Functional Keywords | inhibitor, complex, glpg, rhomboid protease, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor |
Biological source | Escherichia coli More |
Total number of polymer chains | 2 |
Total formula weight | 22429.50 |
Authors | |
Primary citation | Gandhi, S.,Baker, R.P.,Cho, S.,Stanchev, S.,Strisovsky, K.,Urban, S. Designed Parasite-Selective Rhomboid Inhibitors Block Invasion and Clear Blood-Stage Malaria. Cell Chem Biol, 27:1410-1424.e6, 2020 Cited by PubMed: 32888502DOI: 10.1016/j.chembiol.2020.08.011 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.3 Å) |
Structure validation
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