7R8W
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7R8X
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8EXI
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8EXJ
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![BU of 8exj by Molmil](/molmil-images/mine/8exj) | Crystal structure of PTP1B D181A/Q262A phosphatase domain in complex with a JAK1 activation loop phosphopeptide | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, PHOSPHATE ION, Tyrosine-protein kinase JAK1 activation loop peptide, ... | 著者 | Morris, R, Kershaw, N.J, Babon, J.J. | 登録日 | 2022-10-25 | 公開日 | 2023-07-05 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.301 Å) | 主引用文献 | Structure guided studies of the interaction between PTP1B and JAK. Commun Biol, 6, 2023
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8EXM
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![BU of 8exm by Molmil](/molmil-images/mine/8exm) | Crystal structure of PTP1B D181A/Q262A phosphatase domain with a JAK3 activation loop phosphopeptide | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, PHOSPHATE ION, Tyrosine-protein kinase JAK3 activation loop peptide, ... | 著者 | Morris, R, Kershaw, N.J, Babon, J.J. | 登録日 | 2022-10-25 | 公開日 | 2023-07-05 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.349 Å) | 主引用文献 | Structure guided studies of the interaction between PTP1B and JAK. Commun Biol, 6, 2023
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8EXN
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![BU of 8exn by Molmil](/molmil-images/mine/8exn) | Crystal structure of PTP1B D181A/Q262A phosphatase domain with TYK2 activation loop phosphopeptide | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Non-receptor tyrosine-protein kinase TYK2 activation loop peptide, PHOSPHATE ION, ... | 著者 | Morris, R, Kershaw, N.J, Babon, J.J. | 登録日 | 2022-10-25 | 公開日 | 2023-07-05 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.151 Å) | 主引用文献 | Structure guided studies of the interaction between PTP1B and JAK. Commun Biol, 6, 2023
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8F88
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![BU of 8f88 by Molmil](/molmil-images/mine/8f88) | Crystal structure of PTP1B D181A/Q262A/C215A phosphatase domain with monophosphorylated JAK2 activation loop phosphopeptide | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein kinase JAK2, Tyrosine-protein phosphatase non-receptor type 1 | 著者 | Morris, R, Kershaw, N.J, Babon, J.J. | 登録日 | 2022-11-21 | 公開日 | 2023-07-05 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Structure guided studies of the interaction between PTP1B and JAK. Commun Biol, 6, 2023
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8EYA
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![BU of 8eya by Molmil](/molmil-images/mine/8eya) | Crystal structure of PTP1B D181A/Q262A/C215A phosphatase domain with a JAK2 activation loop phosphopeptide | 分子名称: | 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, ... | 著者 | Morris, R, Kershaw, N.J, Babon, J.J. | 登録日 | 2022-10-26 | 公開日 | 2023-07-05 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.099 Å) | 主引用文献 | Structure guided studies of the interaction between PTP1B and JAK. Commun Biol, 6, 2023
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8EYB
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![BU of 8eyb by Molmil](/molmil-images/mine/8eyb) | Crystal structure of PTP1B D181A/Q262A/C215A phosphatase domain with JAK2 activation loop phosphopeptide | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein kinase JAK2 activation loop phosphopeptide, Tyrosine-protein phosphatase non-receptor type 1 | 著者 | Morris, R, Kershaw, N.J, Babon, J.J. | 登録日 | 2022-10-26 | 公開日 | 2023-07-05 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.349 Å) | 主引用文献 | Structure guided studies of the interaction between PTP1B and JAK. Commun Biol, 6, 2023
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8EXK
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8EYC
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8CZ9
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6QQ3
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![BU of 6qq3 by Molmil](/molmil-images/mine/6qq3) | The room temperature structure of lysozyme via the acoustic levitation of a droplet | 分子名称: | ACETATE ION, CHLORIDE ION, Lysozyme C, ... | 著者 | Axford, D.N, Docker, P, Dye, E, Morris, R. | 登録日 | 2019-02-17 | 公開日 | 2019-03-06 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.53 Å) | 主引用文献 | Non-Contact Universal Sample Presentation for Room Temperature Macromolecular Crystallography Using Acoustic Levitation. Sci Rep, 9, 2019
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5W2O
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![BU of 5w2o by Molmil](/molmil-images/mine/5w2o) | Crystal structure of Mycobacterium tuberculosis KasA | 分子名称: | 3,3',3''-phosphanetriyltripropanoic acid, 3-oxoacyl-[acyl-carrier-protein] synthase 1, CHLORIDE ION, ... | 著者 | Capodagli, G.C, Neiditch, M.B. | 登録日 | 2017-06-06 | 公開日 | 2018-12-05 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Synergistic Lethality of a Binary Inhibitor of Mycobacterium tuberculosis KasA. MBio, 9, 2018
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5W2Q
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![BU of 5w2q by Molmil](/molmil-images/mine/5w2q) | Crystal structure of Mycobacterium tuberculosis KasA in complex with 6U5 | 分子名称: | 3,3',3''-phosphanetriyltripropanoic acid, 3-oxoacyl-[acyl-carrier-protein] synthase 1, GLYCEROL, ... | 著者 | Capodagli, G.C, Neiditch, M.B. | 登録日 | 2017-06-06 | 公開日 | 2018-12-05 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Synergistic Lethality of a Binary Inhibitor of Mycobacterium tuberculosis KasA. MBio, 9, 2018
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5W2S
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5W2P
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![BU of 5w2p by Molmil](/molmil-images/mine/5w2p) | Crystal structure of Mycobacterium tuberculosis KasA in complex with 6U5 | 分子名称: | 3,3',3''-phosphanetriyltripropanoic acid, 3-oxoacyl-[acyl-carrier-protein] synthase 1, GLYCEROL, ... | 著者 | Capodagli, G.C, Neiditch, M.B. | 登録日 | 2017-06-06 | 公開日 | 2018-12-05 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Synergistic Lethality of a Binary Inhibitor of Mycobacterium tuberculosis KasA. MBio, 9, 2018
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6CT5
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1SEN
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![BU of 1sen by Molmil](/molmil-images/mine/1sen) | Endoplasmic reticulum protein Rp19 O95881 | 分子名称: | CHLORIDE ION, PLATINUM (II) ION, Thioredoxin-like protein p19 | 著者 | Liu, Z.-J, Chen, L, Tempel, W, Shah, A, Lee, D, Dailey, T.A, Mayer, M.R, Rose, J.P, Richardson, D.C, Richardson, J.S, Dailey, H.A, Wang, B.-C, Southeast Collaboratory for Structural Genomics (SECSG) | 登録日 | 2004-02-17 | 公開日 | 2004-07-13 | 最終更新日 | 2017-10-11 | 実験手法 | X-RAY DIFFRACTION (1.199 Å) | 主引用文献 | Endoplasmic reticulum protein Rp19 To be Published
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3LON
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![BU of 3lon by Molmil](/molmil-images/mine/3lon) | HCV NS3-4a protease domain with ketoamide inhibitor narlaprevir | 分子名称: | (1R,2S,5S)-3-[N-({1-[(tert-butylsulfonyl)methyl]cyclohexyl}carbamoyl)-3-methyl-L-valyl]-N-{(1S)-1-[(1R)-2-(cyclopropylamino)-1-hydroxy-2-oxoethyl]pentyl}-6,6-dimethyl-3-azabicyclo[3.1.0]hexane-2-carboxamide, BETA-MERCAPTOETHANOL, Genome polyprotein, ... | 著者 | Prongay, A.J. | 登録日 | 2010-02-04 | 公開日 | 2011-01-19 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Candidate selection and preclinical evaluation culminating in the discovery of Narlaprevir (SCH 900518): A potent, selective and orally efficacious second generation HCV NS3 serine protease inhibitor To be Published
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