1UM4
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![BU of 1um4 by Molmil](/molmil-images/mine/1um4) | Catalytic Antibody 21H3 with hapten | 分子名称: | (1R)-1-PHENYLETHYL 4-(ACETYLAMINO)BENZYLPHOSPHONATE, Antibody 21H3 H chain, Antibody 21H3 L chain | 著者 | Beuscher IV, A.E, Reuter, J, Olson, A.J, Romesberg, F.E, Schultz, P.G, Wirsching, P, Janda, K.D, Lerner, R.A, Stevens, R.C. | 登録日 | 2003-09-23 | 公開日 | 2004-10-05 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structural Studies of an Efficient Catalytic Antibody Operating by Ping-Pong and Induced Fit Mechanisms To be Published
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1UM6
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![BU of 1um6 by Molmil](/molmil-images/mine/1um6) | catalytic antibody 21h3 | 分子名称: | antibody 21h3, H chain, L chain | 著者 | Beuscher IV, A.E, Reuter, J, Olson, A.J, Romesberg, F.E, Schultz, P.G, Wirsching, P, Janda, K.D, Lerner, R.A, Stevens, R.C. | 登録日 | 2003-09-23 | 公開日 | 2004-10-05 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structural Studies of an Efficient Catalytic Antibody Operating by Ping-Pong and Induced Fit Mechanisms To be Published
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1UM5
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![BU of 1um5 by Molmil](/molmil-images/mine/1um5) | Catalytic Antibody 21H3 with alcohol substrate | 分子名称: | 1-PHENYLETHANOL, Antibody 21H3 H chain, Antibody 21H3 L chain | 著者 | Beuscher IV, A.E, Reuter, J, Olson, A.J, Romesberg, F.E, Schultz, P.G, Wirsching, P, Janda, K.D, Lerner, R.A, Stevens, R.C. | 登録日 | 2003-09-23 | 公開日 | 2004-10-05 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Structural Studies of an Efficient Catalytic Antibody Operating by Ping-Pong and Induced Fit Mechanisms To be Published
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1CF8
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![BU of 1cf8 by Molmil](/molmil-images/mine/1cf8) | Convergence of catalytic antibody and terpene cyclase mechanisms: polyene cyclization directed by carbocation-pi interactions | 分子名称: | 4-{4-[2-(1A,7A-DIMETHYL-4-OXY-OCTAHYDRO-1-OXA-4-AZA-CYCLOPROPA[A]NAPHTHALEN-4-YL) -ACETYLAMINO]-PHENYLCARBAMOYL}-BUTYRIC ACID, CADMIUM ION, PROTEIN (CATALYTIC ANTIBODY 19A4 (HEAVY CHAIN)), ... | 著者 | Paschall, C.M, Hasserodt, J, Jones, T, Lerner, R.A, Janda, K.D, Christianson, D.W. | 登録日 | 1999-03-24 | 公開日 | 1999-07-28 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Convergence of Catalytic Antibody and Terpene Cyclase Mechanisms: Polyene Cyclization Directed by Carbocation-pi Interactions Angew.Chem.Int.Ed.Engl., 38, 1999
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5TTJ
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![BU of 5ttj by Molmil](/molmil-images/mine/5ttj) | |
5TTK
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![BU of 5ttk by Molmil](/molmil-images/mine/5ttk) | |
2G7N
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![BU of 2g7n by Molmil](/molmil-images/mine/2g7n) | Structure of the Light Chain of Botulinum Neurotoxin Serotype A Bound to small Molecule Inhibitors | 分子名称: | Botulinum neurotoxin type A, SILVER ION, ZINC ION | 著者 | Fu, Z, Baldwin, M.R, Boldt, G.E, Janda, K.D, Barbieri, J.T, Kim, J.-J.P. | 登録日 | 2006-02-28 | 公開日 | 2007-03-13 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure of the Light Chain of Botulinum Neurotoxin Serotype A bound to Small Molecule Inhibitors To be Published
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2G7P
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![BU of 2g7p by Molmil](/molmil-images/mine/2g7p) | Structure of the Light Chain of Botulinum Neurotoxin Serotype A Bound to Small Molecule Inhibitors | 分子名称: | Botulinum neurotoxin type A, ZINC ION | 著者 | Fu, Z, Baldwin, M.R, Boldt, G.E, Janda, K.D, Barbieri, J.T, Kim, J.-J.P. | 登録日 | 2006-02-28 | 公開日 | 2006-08-15 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Light chain of botulinum neurotoxin serotype A: structural resolution of a catalytic intermediate. Biochemistry, 45, 2006
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2G7K
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![BU of 2g7k by Molmil](/molmil-images/mine/2g7k) | Structure of the Light Chain of Botulinum Neurotoxin, Serotype A Bound to small Molecule Inhibitors | 分子名称: | Botulinum neurotoxin type A | 著者 | Fu, Z, Baldwin, M.R, Boldt, G.E, Crawford, A, Janda, K.D, Barbieri, J.T, Kim, J.-J.P. | 登録日 | 2006-02-28 | 公開日 | 2006-08-15 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Light chain of botulinum neurotoxin serotype A: structural resolution of a catalytic intermediate. Biochemistry, 45, 2006
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2G7Q
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![BU of 2g7q by Molmil](/molmil-images/mine/2g7q) | Structure of the Light Chain of Botulinum Neurotoxin Serotype A Bound to Small Molecule Inhibitors | 分子名称: | Botulinum neurotoxin type A, N-HYDROXY-L-ARGININAMIDE, ZINC ION | 著者 | Fu, Z, Baldwin, M.R, Boldt, G.E, Janda, K.D, Barbieri, J.T, Kim, J.-J.P. | 登録日 | 2006-02-28 | 公開日 | 2006-08-15 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.41 Å) | 主引用文献 | Light chain of botulinum neurotoxin serotype A: structural resolution of a catalytic intermediate. Biochemistry, 45, 2006
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3QG7
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![BU of 3qg7 by Molmil](/molmil-images/mine/3qg7) | Structural Basis for Ligand Recognition and Discrimination of a Quorum Quenching Antibody | 分子名称: | AP4-24H11 Antibody Heavy Chain, AP4-24H11 Antibody Light Chain, HEXAETHYLENE GLYCOL, ... | 著者 | Kirchdoerfer, R.K, Kaufmann, G.F, Janda, J.D, Wilson, I.A. | 登録日 | 2011-01-24 | 公開日 | 2011-03-23 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.78 Å) | 主引用文献 | Structural Basis for Ligand Recognition and Discrimination of a Quorum-quenching Antibody. J.Biol.Chem., 286, 2011
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3QG6
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![BU of 3qg6 by Molmil](/molmil-images/mine/3qg6) | Structural Basis for Ligand Recognition and Discrimination of a Quorum Quenching Antibody | 分子名称: | AP4-24H11 Heavy Chain, AP4-24H11 Light Chain, Agr autoinducing peptide, ... | 著者 | Kirchdoerfer, R.N, Janda, J.D, Kaufmann, G.F, Wilson, I.A. | 登録日 | 2011-01-24 | 公開日 | 2011-03-23 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structural Basis for Ligand Recognition and Discrimination of a Quorum-quenching Antibody. J.Biol.Chem., 286, 2011
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8TFR
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![BU of 8tfr by Molmil](/molmil-images/mine/8tfr) | Apo Fab from C10-S66K antibody | 分子名称: | Heavy chain from Fab of C10_S66K antibody, Immunoglobulin G-binding protein G, Light chain from Fab of C10_S66K antibody | 著者 | Pholcharee, T, Wilson, I.A. | 登録日 | 2023-07-11 | 公開日 | 2023-08-16 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.99 Å) | 主引用文献 | An Engineered Human-Antibody Fragment with Fentanyl Pan-Specificity That Reverses Carfentanil-Induced Respiratory Depression. Acs Chem Neurosci, 14, 2023
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8TFP
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![BU of 8tfp by Molmil](/molmil-images/mine/8tfp) | Fab from C10-S66K antibody in complex with carfentanil | 分子名称: | Carfentanil, Heavy chain of Fab from C10-S66K antibody, Light chain of Fab from C10-S66K antibody | 著者 | Pholcharee, T, Wilson, I.A. | 登録日 | 2023-07-11 | 公開日 | 2023-08-16 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.78 Å) | 主引用文献 | An Engineered Human-Antibody Fragment with Fentanyl Pan-Specificity That Reverses Carfentanil-Induced Respiratory Depression. Acs Chem Neurosci, 14, 2023
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8TFQ
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![BU of 8tfq by Molmil](/molmil-images/mine/8tfq) | Fab from C10-S66K antibody in complex with fentanyl | 分子名称: | Heavy chain from Fab of C10_S66K antibody, Light chain from Fab of C10_S66K antibody, N-phenyl-N-[1-(2-phenylethyl)piperidin-4-yl]propanamide | 著者 | Pholcharee, T, Wilson, I.A. | 登録日 | 2023-07-11 | 公開日 | 2023-08-16 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | An Engineered Human-Antibody Fragment with Fentanyl Pan-Specificity That Reverses Carfentanil-Induced Respiratory Depression. Acs Chem Neurosci, 14, 2023
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1A3L
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![BU of 1a3l by Molmil](/molmil-images/mine/1a3l) | |
7N18
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![BU of 7n18 by Molmil](/molmil-images/mine/7n18) | Clostridium botulinum Neurotoxin Serotype A Light Chain Inhibited by a Chiral Hydroxamic Acid | 分子名称: | (3R)-3-(4-chlorophenyl)-N,5-dihydroxypentanamide, (3S)-3-(4-chlorophenyl)-N,5-dihydroxypentanamide, Botulinum neurotoxin type A, ... | 著者 | Silvaggi, N.R, Allen, K.N. | 登録日 | 2021-05-27 | 公開日 | 2022-07-06 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.03 Å) | 主引用文献 | Use of Crystallography and Molecular Modeling for the Inhibition of the Botulinum Neurotoxin A Protease. Acs Med.Chem.Lett., 12, 2021
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6C71
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![BU of 6c71 by Molmil](/molmil-images/mine/6c71) | Nicotine Oxidoreductase in Complex with S-nicotine | 分子名称: | (S)-3-(1-METHYLPYRROLIDIN-2-YL)PYRIDINE, Amine oxidase, FLAVIN-ADENINE DINUCLEOTIDE | 著者 | Tararina, M.A, Allen, K.N. | 登録日 | 2018-01-19 | 公開日 | 2018-07-11 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.649 Å) | 主引用文献 | Crystallography Coupled with Kinetic Analysis Provides Mechanistic Underpinnings of a Nicotine-Degrading Enzyme. Biochemistry, 57, 2018
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1NCW
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![BU of 1ncw by Molmil](/molmil-images/mine/1ncw) | |
4HEV
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![BU of 4hev by Molmil](/molmil-images/mine/4hev) | Clostridium Botulinum Serotype A Light Chain Inhibited By Adamantane Hydroxamate | 分子名称: | Botulinum neurotoxin type A light chain, N-hydroxy-2-[(3S,5S,7S)-tricyclo[3.3.1.1~3,7~]dec-1-yl]acetamide, ZINC ION | 著者 | Silvaggi, N.R, Allen, K.N. | 登録日 | 2012-10-04 | 公開日 | 2013-01-23 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Evaluation of adamantane hydroxamates as botulinum neurotoxin inhibitors: synthesis, crystallography, modeling, kinetic and cellular based studies. Bioorg.Med.Chem., 21, 2013
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1ND0
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![BU of 1nd0 by Molmil](/molmil-images/mine/1nd0) | |
1I7Z
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![BU of 1i7z by Molmil](/molmil-images/mine/1i7z) | ANTIBODY GNC92H2 BOUND TO LIGAND | 分子名称: | CHIMERA OF IG GAMMA-1 CHAIN: HUMAN CONSTANT REGION AND MOUSE VARIABLE REGION, CHIMERA OF IG KAPPA CHAIN: HUMAN CONSTANT REGION AND MOUSE VARIABLE REGION, COCAINE | 著者 | Larsen, N.A, Wilson, I.A. | 登録日 | 2001-03-12 | 公開日 | 2001-08-08 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal structure of a cocaine-binding antibody. J.Mol.Biol., 311, 2001
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1FL3
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![BU of 1fl3 by Molmil](/molmil-images/mine/1fl3) | |
3CFC
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![BU of 3cfc by Molmil](/molmil-images/mine/3cfc) | |
3CFE
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![BU of 3cfe by Molmil](/molmil-images/mine/3cfe) | Crystal structure of purple-fluorescent antibody EP2-25C10 | 分子名称: | GLYCEROL, PURPLE-FLUORESCENT ANTIBODY EP2-25C10-IGG2B HEAVY CHAIN, PURPLE-FLUORESCENT ANTIBODY EP2-25C10-KAPPA LIGHT CHAIN, ... | 著者 | Debler, E.W, Heine, A, Wilson, I.A. | 登録日 | 2008-03-03 | 公開日 | 2008-03-18 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.99 Å) | 主引用文献 | Deeply inverted electron-hole recombination in a luminescent antibody-stilbene complex. Science, 319, 2008
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