3HD6
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![BU of 3hd6 by Molmil](/molmil-images/mine/3hd6) | Crystal Structure of the Human Rhesus Glycoprotein RhCG | 分子名称: | Ammonium transporter Rh type C, octyl beta-D-glucopyranoside | 著者 | Gruswitz, F, Chaudhary, S, Ho, J.D, Pezeshki, B, Ho, C.-M, Stroud, R.M, Center for Structures of Membrane Proteins (CSMP) | 登録日 | 2009-05-06 | 公開日 | 2009-09-01 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Function of human Rh based on structure of RhCG at 2.1 A. Proc.Natl.Acad.Sci.USA, 107, 2010
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3K8N
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![BU of 3k8n by Molmil](/molmil-images/mine/3k8n) | |
2TSC
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![BU of 2tsc by Molmil](/molmil-images/mine/2tsc) | STRUCTURE, MULTIPLE SITE BINDING, AND SEGMENTAL ACCOMODATION IN THYMIDYLATE SYNTHASE ON BINDING D/UMP AND AN ANTI-FOLATE | 分子名称: | 10-PROPARGYL-5,8-DIDEAZAFOLIC ACID, 2'-DEOXYURIDINE 5'-MONOPHOSPHATE, THYMIDYLATE SYNTHASE | 著者 | Montfort, W.R, Stroud, R.M. | 登録日 | 1991-07-03 | 公開日 | 1991-10-15 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.97 Å) | 主引用文献 | Structure, multiple site binding, and segmental accommodation in thymidylate synthase on binding dUMP and an anti-folate. Biochemistry, 29, 1990
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2TGD
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![BU of 2tgd by Molmil](/molmil-images/mine/2tgd) | |
3R1F
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![BU of 3r1f by Molmil](/molmil-images/mine/3r1f) | Crystal structure of a key regulator of virulence in Mycobacterium tuberculosis | 分子名称: | ESX-1 secretion-associated regulator EspR | 著者 | Rosenberg, O.S, Dovey, C, Finer-Moore, J, Stroud, R.M, Cox, J.S. | 登録日 | 2011-03-10 | 公開日 | 2011-08-03 | 最終更新日 | 2011-08-31 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | EspR, a key regulator of Mycobacterium tuberculosis virulence, adopts a unique dimeric structure among helix-turn-helix proteins. Proc.Natl.Acad.Sci.USA, 108, 2011
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2NG1
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![BU of 2ng1 by Molmil](/molmil-images/mine/2ng1) | N AND GTPASE DOMAINS OF THE SIGNAL SEQUENCE RECOGNITION PROTEIN FFH FROM THERMUS AQUATICUS | 分子名称: | 1,2-ETHANEDIOL, 1,4-DIETHYLENE DIOXIDE, GUANOSINE-5'-DIPHOSPHATE, ... | 著者 | Freymann, D.M, Stroud, R.M, Walter, P. | 登録日 | 1998-09-11 | 公開日 | 1999-07-30 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.02 Å) | 主引用文献 | Functional changes in the structure of the SRP GTPase on binding GDP and Mg2+GDP. Nat.Struct.Biol., 6, 1999
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4GGM
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![BU of 4ggm by Molmil](/molmil-images/mine/4ggm) | Structure of LpxI | 分子名称: | (R)-((2R,3S,4R,5R,6R)-3-HYDROXY-2-(HYDROXYMETHYL)-5-((R)-3-HYDROXYTETRADECANAMIDO)-6-(PHOSPHONOOXY)TETRAHYDRO-2H-PYRAN-4-YL) 3-HYDROXYTETRADECANOATE, MAGNESIUM ION, UDP-2,3-diacylglucosamine pyrophosphatase LpxI | 著者 | Metzger IV, L.E, Lee, J.K, Finer-Moore, J.S, Raetz, C.R.H, Stroud, R.M, Center for Structures of Membrane Proteins (CSMP) | 登録日 | 2012-08-06 | 公開日 | 2012-10-03 | 最終更新日 | 2017-10-25 | 実験手法 | X-RAY DIFFRACTION (2.897 Å) | 主引用文献 | LpxI structures reveal how a lipid A precursor is synthesized. Nat.Struct.Mol.Biol., 19, 2012
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4HB1
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![BU of 4hb1 by Molmil](/molmil-images/mine/4hb1) | A DESIGNED FOUR HELIX BUNDLE PROTEIN. | 分子名称: | DHP1, UNKNOWN ATOM OR ION | 著者 | Schafmeister, C.E, Laporte, S.L, Miercke, L.J.W, Stroud, R.M. | 登録日 | 1997-11-10 | 公開日 | 1998-03-04 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | A designed four helix bundle protein with native-like structure. Nat.Struct.Biol., 4, 1997
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4ISK
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![BU of 4isk by Molmil](/molmil-images/mine/4isk) | Crystal structure of E.coli thymidylate synthase with dUMP and the BGC 945 inhibitor | 分子名称: | 2'-DEOXYURIDINE 5'-MONOPHOSPHATE, 2'-deoxy-5'-uridylic acid, MAGNESIUM ION, ... | 著者 | Tochowicz, A, Finer-Moore, J, Stroud, R.M. | 登録日 | 2013-01-16 | 公開日 | 2013-12-25 | 最終更新日 | 2014-02-12 | 実験手法 | X-RAY DIFFRACTION (1.752 Å) | 主引用文献 | Development and Binding Mode Assessment of N-[4-[2-Propyn-1-yl[(6S)-4,6,7,8-tetrahydro-2-(hydroxymethyl)-4-oxo-3H-cyclopenta[g]quinazolin-6-yl]amino]benzoyl]-l-gamma-glutamyl-d-glutamic Acid (BGC 945), a Novel Thymidylate Synthase Inhibitor That Targets Tumor Cells. J.Med.Chem., 56, 2013
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4ITS
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![BU of 4its by Molmil](/molmil-images/mine/4its) | Crystal structure of the catalytic domain of human Pus1 with MES in the active site | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, SULFATE ION, tRNA pseudouridine synthase A, ... | 著者 | Czudnochowski, N, Finer-Moore, J.S, Stroud, R.M. | 登録日 | 2013-01-18 | 公開日 | 2013-06-05 | 最終更新日 | 2013-10-23 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | In Human Pseudouridine Synthase 1 (hPus1), a C-Terminal Helical Insert Blocks tRNA from Binding in the Same Orientation as in the Pus1 Bacterial Homologue TruA, Consistent with Their Different Target Selectivities. J.Mol.Biol., 425, 2013
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1TGN
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![BU of 1tgn by Molmil](/molmil-images/mine/1tgn) | |
4ZYR
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![BU of 4zyr by Molmil](/molmil-images/mine/4zyr) | Crystal structure of E. coli Lactose permease G46W/G262W bound to p-nitrophenyl alpha-D-galactopyranoside (alpha-NPG) | 分子名称: | 4-nitrophenyl alpha-D-galactopyranoside, Lactose permease, nonyl beta-D-glucopyranoside | 著者 | Kumar, H, Finer-Moore, J.S, Kaback, H.R, Stroud, R.M. | 登録日 | 2015-05-22 | 公開日 | 2015-07-29 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (3.312 Å) | 主引用文献 | Structure of LacY with an alpha-substituted galactoside: Connecting the binding site to the protonation site. Proc.Natl.Acad.Sci.USA, 112, 2015
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1NG1
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![BU of 1ng1 by Molmil](/molmil-images/mine/1ng1) | N AND GTPASE DOMAINS OF THE SIGNAL SEQUENCE RECOGNITION PROTEIN FFH FROM THERMUS AQUATICUS | 分子名称: | 1,2-ETHANEDIOL, ACETIC ACID, CADMIUM ION, ... | 著者 | Freymann, D.M, Stroud, R.M, Walter, P. | 登録日 | 1998-04-30 | 公開日 | 1999-07-30 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.03 Å) | 主引用文献 | Functional changes in the structure of the SRP GTPase on binding GDP and Mg2+GDP. Nat.Struct.Biol., 6, 1999
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3LNN
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![BU of 3lnn by Molmil](/molmil-images/mine/3lnn) | Crystal structure of ZneB from Cupriavidus metallidurans | 分子名称: | Membrane fusion protein (MFP) heavy metal cation efflux ZneB (CzcB-like), ZINC ION | 著者 | Lee, J.K, De Angelis, F, Miercke, L.J, Stroud, R.M, Vandenbussche, G, Center for Structures of Membrane Proteins (CSMP) | 登録日 | 2010-02-02 | 公開日 | 2010-06-30 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.796 Å) | 主引用文献 | Metal-induced conformational changes in ZneB suggest an active role of membrane fusion proteins in efflux resistance systems. Proc.Natl.Acad.Sci.USA, 107, 2010
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2IST
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![BU of 2ist by Molmil](/molmil-images/mine/2ist) | |
3NK5
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![BU of 3nk5 by Molmil](/molmil-images/mine/3nk5) | Crystal structure of AqpZ mutant F43W | 分子名称: | Aquaporin Z, octyl beta-D-glucopyranoside | 著者 | Savage, D.F, O'Connell, J.D, Stroud, R.M, Finer-Moore, J.S. | 登録日 | 2010-06-18 | 公開日 | 2010-08-11 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structural context shapes the aquaporin selectivity filter. Proc.Natl.Acad.Sci.USA, 107, 2010
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3MP7
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![BU of 3mp7 by Molmil](/molmil-images/mine/3mp7) | |
1NN6
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![BU of 1nn6 by Molmil](/molmil-images/mine/1nn6) | Human Pro-Chymase | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Chymase | 著者 | Reiling, K.K, Krucinski, J, Miercke, L.J.W, Raymond, W.W, Caughey, G.H, Stroud, R.M. | 登録日 | 2003-01-12 | 公開日 | 2003-03-04 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Structure of human pro-chymase: a model for the activating transition of granule-associated proteases. Biochemistry, 42, 2003
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3NKC
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![BU of 3nkc by Molmil](/molmil-images/mine/3nkc) | Crystal structure of AqpZ F43W,H174G,T183F | 分子名称: | Aquaporin Z, octyl beta-D-glucopyranoside | 著者 | Savage, D.F, O'Connell III, J.D, Finer-Moore, J, Stroud, R.M. | 登録日 | 2010-06-18 | 公開日 | 2010-11-03 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Structural context shapes the aquaporin selectivity filter. Proc.Natl.Acad.Sci.USA, 107, 2010
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3NE2
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![BU of 3ne2 by Molmil](/molmil-images/mine/3ne2) | |
3NKA
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![BU of 3nka by Molmil](/molmil-images/mine/3nka) | Crystal structure of AqpZ H174G,T183F | 分子名称: | Aquaporin Z, GLYCEROL, octyl beta-D-glucopyranoside | 著者 | Savage, D.F, O'Connell III, J.D, Finer-Moore, J, Stroud, R.M. | 登録日 | 2010-06-18 | 公開日 | 2010-11-03 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structural context shapes the aquaporin selectivity filter. Proc.Natl.Acad.Sci.USA, 107, 2010
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3P5S
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![BU of 3p5s by Molmil](/molmil-images/mine/3p5s) | Structural insights into the catalytic mechanism of CD38: Evidence for a conformationally flexible covalent enzyme-substrate complex | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, CD38 molecule, SULFATE ION, ... | 著者 | Egea, P.F, Muller-Stauffler, H, Kohn, I, Cakou-Kefir, C, Stroud, R.M, Kellenberburger, E, Schuber, F. | 登録日 | 2010-10-10 | 公開日 | 2011-10-19 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Insights into the mechanism of bovine CD38/NAD+glycohydrolase from the X-ray structures of its Michaelis complex and covalently-trapped intermediates. Plos One, 7, 2012
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1ZPR
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![BU of 1zpr by Molmil](/molmil-images/mine/1zpr) | E. COLI THYMIDYLATE SYNTHASE MUTANT E58Q IN COMPLEX WITH CB3717 AND 2'-DEOXYURIDINE 5'-MONOPHOSPHATE (DUMP) | 分子名称: | 10-PROPARGYL-5,8-DIDEAZAFOLIC ACID, 2'-DEOXYURIDINE 5'-MONOPHOSPHATE, THYMIDYLATE SYNTHASE | 著者 | Sage, C.R, Stout, T.J, Rutenber, E.E, Stroud, R.M. | 登録日 | 1996-10-15 | 公開日 | 1997-07-07 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | An essential role for water in an enzyme reaction mechanism: the crystal structure of the thymidylate synthase mutant E58Q. Biochemistry, 35, 1996
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2G86
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![BU of 2g86 by Molmil](/molmil-images/mine/2g86) | |
2G8D
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![BU of 2g8d by Molmil](/molmil-images/mine/2g8d) | |