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4IOR
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BU of 4ior by Molmil
Crystal Structure of the first bromodomain of BRD4 in complex with DMSO
分子名称: 1,2-ETHANEDIOL, Bromodomain-containing protein 4, DIMETHYL SULFOXIDE
著者Lolli, G, Battistutta, R.
登録日2013-01-08
公開日2013-10-02
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Different orientations of low-molecular-weight fragments in the binding pocket of a BRD4 bromodomain.
Acta Crystallogr.,Sect.D, 69, 2013
1ZOF
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BU of 1zof by Molmil
Crystal structure of alkyl hydroperoxide-reductase (AhpC) from Helicobacter Pylori
分子名称: alkyl hydroperoxide-reductase
著者Papinutto, E, Windle, H.J, Cendron, L, Battistutta, R, Kelleher, D, Zanotti, G.
登録日2005-05-13
公開日2005-11-29
最終更新日2024-10-30
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Crystal structure of alkyl hydroperoxide-reductase (AhpC) from Helicobacter pylori.
Biochim.Biophys.Acta, 1753, 2005
4KWP
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BU of 4kwp by Molmil
Crystal Structure of Human CK2-alpha in complex with a benzimidazole inhibitor (K164) at 1.25 A resolution
分子名称: 1,2-ETHANEDIOL, 4,5,6,7-tetrabromo-1-(2-deoxy-beta-D-erythro-pentofuranosyl)-1H-benzimidazole, Casein kinase II subunit alpha, ...
著者Ranchio, A, Lolli, G, Battistutta, R.
登録日2013-05-24
公開日2014-04-09
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献Cell-permeable dual inhibitors of protein kinases CK2 and PIM-1: structural features and pharmacological potential.
Cell.Mol.Life Sci., 71, 2014
1S2X
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BU of 1s2x by Molmil
Crystal structure of Cag-Z from Helicobacter pylori
分子名称: Cag-Z, ISOPROPYL ALCOHOL
著者Cendron, L, Seydel, A, Angelini, A, Battistutta, R, Zanotti, G.
登録日2004-01-12
公開日2004-07-27
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structure of CagZ, a protein from the Helicobacter pylori pathogenicity island that encodes for a type IV secretion system
J.Mol.Biol., 340, 2004
6QS5
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BU of 6qs5 by Molmil
Crystal Structure of maize CK2 in complex with tyrphostin AG99
分子名称: (~{E})-3-[3,4-bis(oxidanyl)phenyl]-2-cyano-prop-2-enamide, Casein kinase II subunit alpha
著者Lolli, G, Mazzorana, M, Battistutta, R.
登録日2019-02-20
公開日2019-02-27
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.961 Å)
主引用文献Inhibition of protein kinase CK2 by flavonoids and tyrphostins. A structural insight.
Biochemistry, 51, 2012
6RFE
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BU of 6rfe by Molmil
Human protein kinase CK2 alpha in complex with 2-cyano-2-propenamide compound 4
分子名称: (~{E})-~{N}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamide, 1,2-ETHANEDIOL, Casein kinase II subunit alpha, ...
著者Dalle Vedove, A, Zanforlin, E, Ribaudo, G, Zagotto, G, Battistutta, R, Lolli, G.
登録日2019-04-13
公開日2020-04-08
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.54 Å)
主引用文献A novel class of selective CK2 inhibitors targeting its open hinge conformation.
Eur.J.Med.Chem., 195, 2020
6RFF
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BU of 6rff by Molmil
Human protein kinase CK2 alpha in complex with 2-cyano-2-propenamide compound 7
分子名称: (~{E})-~{N}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-nitro-4-oxidanyl-phenyl)prop-2-enamide, 1,2-ETHANEDIOL, Casein kinase II subunit alpha, ...
著者Dalle Vedove, A, Zanforlin, E, Ribaudo, G, Zagotto, G, Battistutta, R, Lolli, G.
登録日2019-04-14
公開日2020-04-08
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献A novel class of selective CK2 inhibitors targeting its open hinge conformation.
Eur.J.Med.Chem., 195, 2020
6RCM
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BU of 6rcm by Molmil
Human protein kinase CK2 alpha in complex with 2-cyano-2-propenamide compound 3
分子名称: (~{E})-~{N}-(5-~{tert}-butyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamide, 1,2-ETHANEDIOL, Casein kinase II subunit alpha, ...
著者Dalle Vedove, A, Zanforlin, E, Ribaudo, G, Zagotto, G, Battistutta, R, Lolli, G.
登録日2019-04-11
公開日2020-04-08
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献A novel class of selective CK2 inhibitors targeting its open hinge conformation.
Eur.J.Med.Chem., 195, 2020
1NZE
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BU of 1nze by Molmil
Crystal structure of PsbQ polypeptide of photosystem II from higher plants
分子名称: Oxygen-evolving enhancer protein 3, ZINC ION
著者Calderone, V, Trabucco, M, Vujicic, A, Battistutta, R, Giacometti, G.M, Andreucci, F, Barbato, R, Zanotti, G.
登録日2003-02-17
公開日2003-08-26
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Crystal structure of the PsbQ protein of photosystem II from higher plants
Embo Rep., 4, 2003
1OO2
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BU of 1oo2 by Molmil
Crystal structure of transthyretin from Sparus aurata
分子名称: CADMIUM ION, transthyretin
著者Pasquato, N, Ramazzina, I, Folli, C, Battistutta, R, Berni, R, Zanotti, G.
登録日2003-03-03
公開日2004-01-20
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献Distinctive binding and structural properties of piscine transthyretin.
Febs Lett., 555, 2003
1M2P
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BU of 1m2p by Molmil
Crystal structure of 1,8-di-hydroxy-4-nitro-anthraquinone/CK2 kinase complex
分子名称: 1,8-DI-HYDROXY-4-NITRO-ANTHRAQUINONE, Casein kinase II, alpha chain
著者De Moliner, E, Moro, S, Sarno, S, Zagotto, G, Zanotti, G, Pinna, L.A, Battistutta, R.
登録日2002-06-25
公開日2003-06-17
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Inhibition of protein kinase CK2 by anthraquinone-related compounds. A structural insight
J.Biol.Chem., 278, 2003
1M2R
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BU of 1m2r by Molmil
Crystal structure of 5,8-di-amino-1,4-di-hydroxy-anthraquinone/CK2 kinase complex
分子名称: 5,8-DI-AMINO-1,4-DIHYDROXY-ANTHRAQUINONE, CASEIN kinase II, alpha chain
著者De Moliner, E, Moro, S, Sarno, S, Zagotto, G, Zanotti, G, Pinna, L.A, Battistutta, R.
登録日2002-06-25
公開日2003-06-17
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Inhibition of protein kinase CK2 by anthraquinone-related compounds. A structural insight
J.Biol.Chem., 278, 2003
1M2Q
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BU of 1m2q by Molmil
Crystal structure of 1,8-di-hydroxy-4-nitro-xanten-9-one/CK2 kinase complex
分子名称: 1,8-DI-HYDROXY-4-NITRO-XANTHEN-9-ONE, Casein kinase II, alpha chain
著者De Moliner, E, Sarno, S, Moro, S, Zagotto, G, Zanotti, G, Pinna, L.A, Battistutta, R.
登録日2002-06-25
公開日2003-06-17
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.79 Å)
主引用文献Inhibition of protein kinase CK2 by anthraquinone-related compounds. A structural insight
J.Biol.Chem., 278, 2003
3PVG
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BU of 3pvg by Molmil
Crystal structure of Z. mays CK2 alpha subunit in complex with the inhibitor 4,5,6,7-tetrabromo-1-carboxymethylbenzimidazole (K68)
分子名称: (4,5,6,7-tetrabromo-1H-benzimidazol-1-yl)acetic acid, Casein kinase II subunit alpha
著者Papinutto, E, Franchin, C, Battistutta, R.
登録日2010-12-07
公開日2010-12-15
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献ATP site-directed inhibitors of protein kinase CK2: an update.
Curr Top Med Chem, 11, 2011
3CWY
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BU of 3cwy by Molmil
Structure of CagD from H. pylori pathogenicity island crystallized in the presence of Cu(II) ions
分子名称: COPPER (II) ION, protein CagD
著者Cendron, L, Zanotti, G, Angelini, A, Barison, N, Couturier, M, Stein, M.
登録日2008-04-23
公開日2008-12-30
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献The Helicobacter pylori CagD (HP0545, Cag24) protein is essential for CagA translocation and maximal induction of interleukin-8 secretion.
J.Mol.Biol., 386, 2009
3CWX
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BU of 3cwx by Molmil
Crystal structure of cagd from helicobacter pylori pathogenicity island
分子名称: protein CagD
著者Cendron, L, Zanotti, G, Angelini, A, Barison, N, Couturier, M, Stein, M.
登録日2008-04-23
公開日2008-12-30
最終更新日2024-10-30
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献The Helicobacter pylori CagD (HP0545, Cag24) protein is essential for CagA translocation and maximal induction of interleukin-8 secretion.
J.Mol.Biol., 386, 2009
1O9R
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BU of 1o9r by Molmil
The X-ray crystal structure of Agrobacterium tumefaciens Dps, a member of the family that protect DNA without binding
分子名称: 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, AGROBACTERIUM TUMEFACIENS DPS, ...
著者Ilari, A, Ceci, P, Chiancone, E.
登録日2002-12-18
公開日2003-05-29
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献The Dps Protein of Agrobacterium Tumefaciens Does not Bind to DNA But Protects It Toward Oxidative Cleavage: X-Ray Crystal Structure, Iron Binding, and Hydroxyl-Radical Scavenging Properties
J.Biol.Chem., 278, 2003
2PNC
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BU of 2pnc by Molmil
Crystal Structure of Bovine Plasma Copper-Containing Amine Oxidase in Complex with Clonidine
分子名称: 2,6-DICHLORO-N-IMIDAZOLIDIN-2-YLIDENEANILINE, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Cendron, L, Holt, A, Smith, D.J, Zanotti, G, Rigo, A, Di Paolo, M.L.
登録日2007-04-24
公開日2008-02-26
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Multiple binding sites for substrates and modulators of semicarbazide-sensitive amine oxidases: kinetic consequences
Mol.Pharmacol., 73, 2008
6RCB
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BU of 6rcb by Molmil
Human protein kinase CK2 alpha in complex with 2-cyano-2-propenamide compound 14
分子名称: (~{E})-2-cyano-~{N}-(2-hydroxyphenyl)-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamide, Casein kinase II subunit alpha, SULFATE ION
著者Dalle Vedove, A, Lolli, G.
登録日2019-04-11
公開日2020-04-08
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献A novel class of selective CK2 inhibitors targeting its open hinge conformation.
Eur.J.Med.Chem., 195, 2020
6HOV
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BU of 6hov by Molmil
Crystal Structure of BRD4 first bromodomain in complex with ferulic acid
分子名称: 1,2-ETHANEDIOL, 3-(4-HYDROXY-3-METHOXYPHENYL)-2-PROPENOIC ACID, Bromodomain-containing protein 4
著者Dalle Vedove, A, Lolli, G.
登録日2018-09-18
公開日2019-10-09
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Biochemical and cellular mechanism of protein kinase CK2 inhibition by deceptive curcumin.
Febs J., 287, 2020
1LTR
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BU of 1ltr by Molmil
CRYSTAL STRUCTURE OF THE B SUBUNIT OF HUMAN HEAT-LABILE ENTEROTOXIN FROM E. COLI CARRYING A PEPTIDE WITH ANTI-HSV ACTIVITY
分子名称: HEAT-LABILE ENTEROTOXIN, SULFATE ION
著者Matkovic-Calogovic, D, Loreggian, A, Palu, G, Zanotti, G.
登録日1998-07-31
公開日1999-02-09
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (3.04 Å)
主引用文献Crystal structure of the B subunit of Escherichia coli heat-labile enterotoxin carrying peptides with anti-herpes simplex virus type 1 activity.
J.Biol.Chem., 274, 1999
2PYB
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BU of 2pyb by Molmil
Napa protein from borrelia burgdorferi
分子名称: FE (III) ION, Neutrophil activating protein
著者Zanotti, G, Papinutto, E, De Bernard, M.
登録日2007-05-16
公開日2008-08-12
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structure and immunomodulatory property relationship in NapA of Borrelia burgdorferi.
Biochim.Biophys.Acta, 1804, 2010
6ISJ
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BU of 6isj by Molmil
Crystal structure of CX-4945 bound CK2 alpha from C. neoformans
分子名称: 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid, Casein kinase II subunit alpha, SULFATE ION
著者Cho, H.S.
登録日2018-11-16
公開日2019-11-20
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of CX-4945 bound CK2 alpha from C. neoformans
To be published
1NA7
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BU of 1na7 by Molmil
Crystal structure of the catalytic subunit of human protein kinase CK2
分子名称: Casein kinase II, alpha chain
著者Pechkova, E, Zanotti, G, Nicolini, C.
登録日2002-11-27
公開日2003-08-26
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Three-dimensional atomic structure of a catalytic subunit mutant of human protein kinase CK2.
Acta Crystallogr.,Sect.D, 59, 2003
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