3JSM
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![BU of 3jsm by Molmil](/molmil-images/mine/3jsm) | K65R mutant HIV-1 reverse transcriptase cross-linked to DS-DNA and complexed with tenofovir-diphosphate as the incoming nucleotide substrate | 分子名称: | DNA (5'-D(*A*CP*AP*GP*TP*CP*CP*CP*TP*GP*TP*TP*CP*GP*GP*(MRG)P*CP*GP*CP*CP*(DDG))-3'), DNA (5'-D(*A*TP*GP*GP*TP*CP*GP*GP*CP*GP*CP*CP*CP*GP*AP*AP*CP*AP*GP*GP*GP*AP*CP*TP*GP*TP*G)-3'), HIV-1 REVERSE TRANSCRIPTASE P51 SUBUNIT, ... | 著者 | Das, K, Arnold, E. | 登録日 | 2009-09-10 | 公開日 | 2009-09-29 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structural basis for the role of the K65r mutation in HIV-1 reverse transcriptase polymerization, excision antagonism, and tenofovir resistance. J.Biol.Chem., 284, 2009
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1ARJ
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![BU of 1arj by Molmil](/molmil-images/mine/1arj) | ARG-BOUND TAR RNA, NMR | 分子名称: | ARGININE, TAR RNA | 著者 | Aboul-Ela, F, Varani, G, Karn, J. | 登録日 | 1995-08-30 | 公開日 | 1996-11-08 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | The structure of the human immunodeficiency virus type-1 TAR RNA reveals principles of RNA recognition by Tat protein. J.Mol.Biol., 253, 1995
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5V91
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![BU of 5v91 by Molmil](/molmil-images/mine/5v91) | Crystal structure of fosfomycin resistance protein from Klebsiella pneumoniae | 分子名称: | Fosfomycin resistance protein, ZINC ION | 著者 | Klontz, E, Guenther, S, Silverstein, Z, Sundberg, E. | 登録日 | 2017-03-22 | 公開日 | 2017-08-30 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Structure and Dynamics of FosA-Mediated Fosfomycin Resistance in Klebsiella pneumoniae and Escherichia coli. Antimicrob. Agents Chemother., 61, 2017
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5V3D
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![BU of 5v3d by Molmil](/molmil-images/mine/5v3d) | Crystal structure of fosfomycin resistance protein from Klebsiella pneumoniae with bound fosfomycin | 分子名称: | 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, FOSFOMYCIN, ... | 著者 | Klontz, E, Guenther, S, Silverstein, Z, Sundberg, E. | 登録日 | 2017-03-07 | 公開日 | 2017-08-30 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.539 Å) | 主引用文献 | Structure and Dynamics of FosA-Mediated Fosfomycin Resistance in Klebsiella pneumoniae and Escherichia coli. Antimicrob. Agents Chemother., 61, 2017
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5VB0
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![BU of 5vb0 by Molmil](/molmil-images/mine/5vb0) | Crystal structure of fosfomycin resistance protein FosA3 | 分子名称: | Fosfomycin resistance protein FosA3, MANGANESE (II) ION, NICKEL (II) ION | 著者 | Klontz, E, Guenther, S, Silverstein, Z, Sundberg, E. | 登録日 | 2017-03-28 | 公開日 | 2017-08-30 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.689 Å) | 主引用文献 | Structure and Dynamics of FosA-Mediated Fosfomycin Resistance in Klebsiella pneumoniae and Escherichia coli. Antimicrob. Agents Chemother., 61, 2017
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1EDS
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![BU of 1eds by Molmil](/molmil-images/mine/1eds) | SOLUTION STRUCTURE OF INTRADISKAL LOOP 1 OF BOVINE RHODOPSIN (RHODOPSIN RESIDUES 92-123) | 分子名称: | RHODOPSIN | 著者 | Yeagle, P.L, Salloum, A, Chopra, A, Bhawsar, N, Ali, L. | 登録日 | 2000-01-28 | 公開日 | 2000-08-09 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Structures of the intradiskal loops and amino terminus of the G-protein receptor, rhodopsin. J.Pept.Res., 55, 2000
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1EDW
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![BU of 1edw by Molmil](/molmil-images/mine/1edw) | SOLUTION STRUCTURE OF THIRD INTRADISKAL LOOP OF BOVINE RHODOPSIN (RESIDUES 268-293) | 分子名称: | RHODOPSIN | 著者 | Yeagle, P.L, Salloum, A, Chopra, A, Bhawsar, N, Ali, L. | 登録日 | 2000-01-28 | 公開日 | 2000-08-09 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Structures of the intradiskal loops and amino terminus of the G-protein receptor, rhodopsin. J.Pept.Res., 55, 2000
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4ZXR
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![BU of 4zxr by Molmil](/molmil-images/mine/4zxr) | Structure of Thaumatin wrapped in graphene within vacuum | 分子名称: | GLYCEROL, L(+)-TARTARIC ACID, Thaumatin-1 | 著者 | Aller, P, Warren, A.J, Trincao, J, Evans, G. | 登録日 | 2015-05-20 | 公開日 | 2015-10-14 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.92 Å) | 主引用文献 | In vacuo X-ray data collection from graphene-wrapped protein crystals. Acta Crystallogr.,Sect.D, 71, 2015
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1EDX
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![BU of 1edx by Molmil](/molmil-images/mine/1edx) | SOLUTION STRUCTURE OF AMINO TERMINUS OF BOVINE RHODOPSIN (RESIDUES 1-40) | 分子名称: | RHODOPSIN | 著者 | Yeagle, P.L, Salloum, A, Chopra, A, Bhawsar, N, Ali, L. | 登録日 | 2000-01-28 | 公開日 | 2000-08-09 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Structures of the intradiskal loops and amino terminus of the G-protein receptor, rhodopsin. J.Pept.Res., 55, 2000
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5A5Q
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![BU of 5a5q by Molmil](/molmil-images/mine/5a5q) | Crystal structure of human ATAD2 bromodomain in complex with 3-methyl- 8-piperidin-4-ylamino-1,2-dihydro-1,7-naphthyridin-2-one hydrochloride | 分子名称: | 1,2-ETHANEDIOL, 3-methyl-8-[(piperidin-4-yl)amino]-1,2-dihydro-1,7-naphthyridin-2-one, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2, ... | 著者 | Chung, C, Bamborough, P, Demont, E. | 登録日 | 2015-06-20 | 公開日 | 2015-07-22 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.97 Å) | 主引用文献 | Fragment-Based Discovery of Low-Micromolar Atad2 Bromodomain Inhibitors. J.Med.Chem., 58, 2015
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1EDV
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![BU of 1edv by Molmil](/molmil-images/mine/1edv) | SOLUTION STRUCTURE OF 2ND INTRADISKAL LOOP OF BOVINE RHODOPSIN (RESIDUES 172-205) | 分子名称: | RHODOPSIN | 著者 | Yeagle, P.L, Salloum, A, Chopra, A, Bhawsar, N, Ali, L. | 登録日 | 2000-01-28 | 公開日 | 2000-08-09 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Structures of the intradiskal loops and amino terminus of the G-protein receptor, rhodopsin. J.Pept.Res., 55, 2000
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4FXI
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5A4C
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![BU of 5a4c by Molmil](/molmil-images/mine/5a4c) | FGFR1 ligand complex | 分子名称: | 1,2-ETHANEDIOL, 1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]urea, FIBROBLAST GROWTH FACTOR RECEPTOR 1 (FMS-RELATED TYROSINE KINASE 2, ... | 著者 | Klein, T, Vajpai, N, Phillips, J.J, Davies, G, Holdgate, G.A, Phillips, C, Tucker, J.A, Norman, R.A, Scott, A.S, Higazi, D.R, Lowe, D, Thompson, G.S, Breeze, A.L. | 登録日 | 2015-06-05 | 公開日 | 2015-08-05 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.09 Å) | 主引用文献 | Structural and Dynamic Insights Into the Energetics of Activation Loop Rearrangement in Fgfr1 Kinase. Nat.Commun., 6, 2015
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4H1J
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![BU of 4h1j by Molmil](/molmil-images/mine/4h1j) | Crystal structure of PYK2 with the pyrazole 13a | 分子名称: | 1-[3-tert-butyl-1-(4-methylphenyl)-1H-pyrazol-5-yl]-3-[3-(4-methoxy-2-methylphenyl)-1H-pyrazol-5-yl]urea, Protein-tyrosine kinase 2-beta | 著者 | Han, S. | 登録日 | 2012-09-10 | 公開日 | 2012-11-28 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Identification of novel series of pyrazole and indole-urea based DFG-out PYK2 inhibitors. Bioorg.Med.Chem.Lett., 22, 2012
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3MYG
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![BU of 3myg by Molmil](/molmil-images/mine/3myg) | Aurora A Kinase complexed with SCH 1473759 | 分子名称: | 2-{ethyl[(5-{[6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}isothiazol-3-yl)methyl]amino}-2-methylpropan-1-ol, Serine/threonine-protein kinase 6, TETRAETHYLENE GLYCOL | 著者 | Hruza, A, Prosis, W, Ramanathan, L. | 登録日 | 2010-05-10 | 公開日 | 2010-07-21 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Discovery of a Potent, Injectable Inhibitor of Aurora Kinases Based on the Imidazo-[1,2-a]-Pyrazine Core. ACS Med Chem Lett, 1, 2010
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1RPV
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![BU of 1rpv by Molmil](/molmil-images/mine/1rpv) | HIV-1 REV PROTEIN (RESIDUES 34-50) | 分子名称: | HIV-1 REV PROTEIN | 著者 | Scanlon, M.J, Fairlie, D.P, Craik, D.J, Englebretsen, D.R, West, M.L. | 登録日 | 1995-05-04 | 公開日 | 1995-10-15 | 最終更新日 | 2022-03-02 | 実験手法 | SOLUTION NMR | 主引用文献 | NMR solution structure of the RNA-binding peptide from human immunodeficiency virus (type 1) Rev. Biochemistry, 34, 1995
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5VWZ
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![BU of 5vwz by Molmil](/molmil-images/mine/5vwz) | Bak in complex with Bim-h3Pc | 分子名称: | 2-(2-{2-[2-(2-METHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHANOL, AMMONIUM ION, Bcl-2 homologous antagonist/killer, ... | 著者 | Brouwer, J.M, Colman, P.M, Czabotar, P.E. | 登録日 | 2017-05-23 | 公開日 | 2017-11-15 | 最終更新日 | 2020-01-08 | 実験手法 | X-RAY DIFFRACTION (1.622 Å) | 主引用文献 | Conversion of Bim-BH3 from Activator to Inhibitor of Bak through Structure-Based Design. Mol. Cell, 68, 2017
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5VWY
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![BU of 5vwy by Molmil](/molmil-images/mine/5vwy) | |
3V7S
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![BU of 3v7s by Molmil](/molmil-images/mine/3v7s) | Crystal structure of Staphylococcus aureus biotin protein ligase in complex with inhibitor 0364 | 分子名称: | 5-methyl-3-[4-(4-{5-[(3aS,4S,6aR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl]pentyl}-1H-1,2,3-triazol-1-yl)butyl]-1,3-benzoxazol-2(3H)-one, Biotin ligase | 著者 | Yap, M.Y, Pendini, N.R. | 登録日 | 2011-12-21 | 公開日 | 2012-04-25 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Selective inhibition of biotin protein ligase from Staphylococcus aureus. J.Biol.Chem., 287, 2012
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3VVP
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5VWX
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![BU of 5vwx by Molmil](/molmil-images/mine/5vwx) | Bak core latch dimer in complex with Bim-h0-h3Glt | 分子名称: | 1,2-ETHANEDIOL, Bcl-2 homologous antagonist/killer, Bcl-2-like protein 11 | 著者 | Brouwer, J.M, Lan, P, Lessene, G, Colman, P.M, Czabotar, P.E. | 登録日 | 2017-05-23 | 公開日 | 2017-11-15 | 最終更新日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (2.489 Å) | 主引用文献 | Conversion of Bim-BH3 from Activator to Inhibitor of Bak through Structure-Based Design. Mol. Cell, 68, 2017
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5WH8
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![BU of 5wh8 by Molmil](/molmil-images/mine/5wh8) | Cellulase Cel5C_n | 分子名称: | 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, PENTAETHYLENE GLYCOL, ... | 著者 | Koropatkin, N.M, Pope, P.B, Naas, A.E. | 登録日 | 2017-07-15 | 公開日 | 2018-03-14 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.57 Å) | 主引用文献 | "Candidatus Paraporphyromonas polyenzymogenes" encodes multi-modular cellulases linked to the type IX secretion system. Microbiome, 6, 2018
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3V8K
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3V7R
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![BU of 3v7r by Molmil](/molmil-images/mine/3v7r) | Crystal structure of Staphylococcus aureus biotin protein ligase in complex with inhibitor | 分子名称: | (3aS,4S,6aR)-4-(5-{1-[4-(6-amino-9H-purin-9-yl)butyl]-1H-1,2,3-triazol-4-yl}pentyl)tetrahydro-1H-thieno[3,4-d]imidazol-2(3H)-one, Biotin ligase | 著者 | Yap, M.Y, Pendini, N.R. | 登録日 | 2011-12-21 | 公開日 | 2012-12-26 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.61 Å) | 主引用文献 | Selective inhibition of biotin protein ligase from Staphylococcus aureus. J.Biol.Chem., 287, 2012
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3V8L
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![BU of 3v8l by Molmil](/molmil-images/mine/3v8l) | |