Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
Search by PDB author
5ITD
DownloadVisualize
BU of 5itd by Molmil
Crystal structure of PI3K alpha with PI3K delta inhibitor
分子名称: 5-{4-[3-(4-acetylpiperazine-1-carbonyl)phenyl]quinazolin-6-yl}-2-methoxypyridine-3-carbonitrile, Phosphatidylinositol 3-kinase regulatory subunit alpha, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
著者Knapp, M.S, Elling, R.A.
登録日2016-03-16
公開日2016-09-07
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (3.02 Å)
主引用文献Discovery and Pharmacological Characterization of Novel Quinazoline-Based PI3K Delta-Selective Inhibitors.
Acs Med.Chem.Lett., 7, 2016
5IGJ
DownloadVisualize
BU of 5igj by Molmil
Macrolide 2'-phosphotransferase type I - complex with guanosine and clarithromycin
分子名称: CLARITHROMYCIN, GUANOSINE, ISOPROPYL ALCOHOL, ...
著者Berghuis, A.M, Fong, D.H.
登録日2016-02-28
公開日2017-04-26
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Structural Basis for Kinase-Mediated Macrolide Antibiotic Resistance.
Structure, 25, 2017
5IGW
DownloadVisualize
BU of 5igw by Molmil
Macrolide 2'-phosphotransferase type II - complex with GDP and clarithromycin
分子名称: CLARITHROMYCIN, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
著者Berghuis, A.M, Fong, D.H.
登録日2016-02-28
公開日2017-04-26
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.096 Å)
主引用文献Structural Basis for Kinase-Mediated Macrolide Antibiotic Resistance.
Structure, 25, 2017
5IGI
DownloadVisualize
BU of 5igi by Molmil
Macrolide 2'-phosphotransferase type I - complex with guanosine and azithromycin
分子名称: AZITHROMYCIN, GUANOSINE, ISOPROPYL ALCOHOL, ...
著者Berghuis, A.M, Fong, D.H.
登録日2016-02-28
公開日2017-04-26
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Structural Basis for Kinase-Mediated Macrolide Antibiotic Resistance.
Structure, 25, 2017
5IGT
DownloadVisualize
BU of 5igt by Molmil
Macrolide 2'-phosphotransferase type I - complex with guanosine and erythromycin
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ERYTHROMYCIN A, GUANOSINE, ...
著者Berghuis, A.M, Fong, D.H.
登録日2016-02-28
公開日2017-04-26
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.39 Å)
主引用文献Structural Basis for Kinase-Mediated Macrolide Antibiotic Resistance.
Structure, 25, 2017
5IS5
DownloadVisualize
BU of 5is5 by Molmil
Discovery and Pharmacological Characterization of Novel Quinazoline-based PI3K delta-selective Inhibitors
分子名称: 5-{4-[3-(4-acetylpiperazine-1-carbonyl)phenyl]quinazolin-6-yl}-2-methoxypyridine-3-carbonitrile, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
著者Gutmann, S, Rummel, G, Shrestha, B.
登録日2016-03-15
公開日2016-08-10
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Discovery and Pharmacological Characterization of Novel Quinazoline-Based PI3K Delta-Selective Inhibitors.
Acs Med.Chem.Lett., 7, 2016
5IGP
DownloadVisualize
BU of 5igp by Molmil
Macrolide 2'-phosphotransferase type I - complex with GDP and erythromycin
分子名称: ERYTHROMYCIN A, GUANOSINE-5'-DIPHOSPHATE, ISOPROPYL ALCOHOL, ...
著者Berghuis, A.M, Fong, D.H.
登録日2016-02-28
公開日2017-04-26
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural Basis for Kinase-Mediated Macrolide Antibiotic Resistance.
Structure, 25, 2017
5IGZ
DownloadVisualize
BU of 5igz by Molmil
Macrolide 2'-phosphotransferase type II - complex with GDP and spiramycin
分子名称: GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Macrolide 2'-phosphotransferase II, ...
著者Berghuis, A.M, Fong, D.H.
登録日2016-02-28
公開日2017-04-26
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural Basis for Kinase-Mediated Macrolide Antibiotic Resistance.
Structure, 25, 2017
5IWU
DownloadVisualize
BU of 5iwu by Molmil
Macrolide 2'-phosphotransferase type II complexed with erythromycin
分子名称: ACETATE ION, CALCIUM ION, ERYTHROMYCIN A, ...
著者Berghuis, A.M, Fong, D.H.
登録日2016-03-22
公開日2017-04-26
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Structural Basis for Kinase-Mediated Macrolide Antibiotic Resistance.
Structure, 25, 2017
6HG4
DownloadVisualize
BU of 6hg4 by Molmil
Crystal Structure of the human IL-17RC ECD in complex with human IL-17F
分子名称: Interleukin-17 receptor C, Interleukin-17F
著者Rondeau, J.M, Goepfert, A.
登録日2018-08-22
公開日2020-03-18
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (3.32 Å)
主引用文献Structural Analysis Reveals that the Cytokine IL-17F Forms a Homodimeric Complex with Receptor IL-17RC to Drive IL-17RA-Independent Signaling.
Immunity, 52, 2020
6HGA
DownloadVisualize
BU of 6hga by Molmil
Crystal Structure of the human IL-17RC D2-D3-D4 domains in complex with an anti-APP tag Fab
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Interleukin-17 receptor C, anti-APP-tag Fab heavy-chain, ...
著者Rondeau, J.M, Goepfert, A.
登録日2018-08-23
公開日2020-03-18
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structural Analysis Reveals that the Cytokine IL-17F Forms a Homodimeric Complex with Receptor IL-17RC to Drive IL-17RA-Independent Signaling.
Immunity, 52, 2020
6HGO
DownloadVisualize
BU of 6hgo by Molmil
Crystal Structure of human IL-17F
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Interleukin-17F, ...
著者Rondeau, J.M, Goepfert, A.
登録日2018-08-23
公開日2019-11-20
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structural Analysis Reveals that the Cytokine IL-17F Forms a Homodimeric Complex with Receptor IL-17RC to Drive IL-17RA-Independent Signaling.
Immunity, 52, 2020
5IGY
DownloadVisualize
BU of 5igy by Molmil
Macrolide 2'-phosphotransferase type II - complex with GDP and erythromycin
分子名称: CALCIUM ION, ERYTHROMYCIN A, GUANOSINE-5'-DIPHOSPHATE, ...
著者Berghuis, A.M, Fong, D.H.
登録日2016-02-28
公開日2017-04-26
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Structural Basis for Kinase-Mediated Macrolide Antibiotic Resistance.
Structure, 25, 2017
5IGS
DownloadVisualize
BU of 5igs by Molmil
Macrolide 2'-phosphotransferase type I - complex with guanosine and oleandomycin
分子名称: (3S,5R,6S,7R,8R,11R,12S,13R,14S,15S)-6-HYDROXY-5,7,8,11,13,15-HEXAMETHYL-4,10-DIOXO-14-{[3,4,6-TRIDEOXY-3-(DIMETHYLAMINO)-BETA-D-XYLO-HEXOPYRANOSYL]OXY}-1,9-DIOXASPIRO[2.13]HEXADEC-12-YL 2,6-DIDEOXY-3-O-METHYL-ALPHA-L-ARABINO-HEXOPYRANOSIDE, GUANOSINE, ISOPROPYL ALCOHOL, ...
著者Berghuis, A.M, Fong, D.H.
登録日2016-02-28
公開日2017-04-26
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.38 Å)
主引用文献Structural Basis for Kinase-Mediated Macrolide Antibiotic Resistance.
Structure, 25, 2017
5BNC
DownloadVisualize
BU of 5bnc by Molmil
Structure of heme binding protein MSMEG_6519 from Mycobacterium smegmatis
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, MAGNESIUM ION, NICKEL (II) ION, ...
著者Ahmed, F.H, Carr, P.D, Jackson, C.J.
登録日2015-05-26
公開日2015-10-21
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Sequence-Structure-Function Classification of a Catalytically Diverse Oxidoreductase Superfamily in Mycobacteria.
J.Mol.Biol., 427, 2015
5IGU
DownloadVisualize
BU of 5igu by Molmil
Macrolide 2'-phosphotransferase type II
分子名称: Macrolide 2'-phosphotransferase II
著者Berghuis, A.M, Fong, D.H.
登録日2016-02-28
公開日2017-04-26
最終更新日2020-01-08
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structural Basis for Kinase-Mediated Macrolide Antibiotic Resistance.
Structure, 25, 2017
5IH0
DownloadVisualize
BU of 5ih0 by Molmil
Macrolide 2'-phosphotransferase type II Y92M mutant - complex with GDP and erythromycin
分子名称: ACETATE ION, ERYTHROMYCIN A, GUANOSINE-5'-DIPHOSPHATE, ...
著者Berghuis, A.M, Fong, D.H.
登録日2016-02-28
公開日2017-04-26
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Structural Basis for Kinase-Mediated Macrolide Antibiotic Resistance.
Structure, 25, 2017
4MUH
DownloadVisualize
BU of 4muh by Molmil
Crystal structure of pantothenate synthetase in complex with 2-(2-(5-acetamido-1,3,4-thiadiazol-2-ylsulfonylcarbamoyl)-5-methoxy-1H-indol-1-yl)acetic acid
分子名称: 1,2-ETHANEDIOL, ETHANOL, Pantothenate synthetase, ...
著者Silvestre, H.L, Blundell, T.L.
登録日2013-09-21
公開日2014-08-27
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.72 Å)
主引用文献Optimization of Inhibitors of Mycobacterium tuberculosis Pantothenate Synthetase Based on Group Efficiency Analysis.
Chemmedchem, 11, 2016
4MQ6
DownloadVisualize
BU of 4mq6 by Molmil
Pantothenate synthase in complex with 2-(5-methoxy-2-(tosylcarbamoyl)-1H-indol-1-yl)acetic acid
分子名称: (5-methoxy-2-{[(4-methylphenyl)sulfonyl]carbamoyl}-1H-indol-1-yl)acetic acid, 1,2-ETHANEDIOL, ETHANOL, ...
著者Silvestre, H.L, Blundell, T.L.
登録日2013-09-15
公開日2014-08-27
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Optimization of Inhibitors of Mycobacterium tuberculosis Pantothenate Synthetase Based on Group Efficiency Analysis.
Chemmedchem, 11, 2016
4MUE
DownloadVisualize
BU of 4mue by Molmil
Crystal strcture of pantothenate synthetase in complex with 2-(5-methoxy-2-(4-(trifluoromethyl)phenylsulfonylcarbamoyl)-1H-indol-1-yl)acetic acid
分子名称: 1,2-ETHANEDIOL, ETHANOL, Pantothenate synthetase, ...
著者Silvestre, H.L, Blundell, T.L.
登録日2013-09-21
公開日2014-08-27
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.06 Å)
主引用文献Optimization of Inhibitors of Mycobacterium tuberculosis Pantothenate Synthetase Based on Group Efficiency Analysis.
Chemmedchem, 11, 2016
4MUF
DownloadVisualize
BU of 4muf by Molmil
Crystal structure of pantothenate synthetase in complex with 2-(2-(4-tert-butylphenylsulfonylcarbamoyl)-5-methoxy-1H-indol-1-yl)acetic acid
分子名称: (2-{[(4-tert-butylphenyl)sulfonyl]carbamoyl}-5-methoxy-1H-indol-1-yl)acetic acid, ETHANOL, Pantothenate synthetase
著者Silvestre, H.L, Blundell, T.L.
登録日2013-09-21
公開日2014-08-27
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Optimization of Inhibitors of Mycobacterium tuberculosis Pantothenate Synthetase Based on Group Efficiency Analysis.
Chemmedchem, 11, 2016
1M8Z
DownloadVisualize
BU of 1m8z by Molmil
Crystal Structure Of A Pumilio-Homology Domain
分子名称: BETA-MERCAPTOETHANOL, PUMILIO 1
著者Wang, X, Zamore, P.D, Hall, T.M.T.
登録日2002-07-26
公開日2002-09-04
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structure of a Pumilio homology domain.
Mol.Cell, 7, 2001
4PRU
DownloadVisualize
BU of 4pru by Molmil
Crystal structure of dimethyllysine hen egg-white lysozyme in complex with sclx4 at 2.2 A resolution
分子名称: 25,26,27,28-tetrahydroxypentacyclo[19.3.1.1~3,7~.1~9,13~.1~15,19~]octacosa-1(25),3(28),4,6,9(27),10,12,15(26),16,18,21,23-dodecaene-5,11,17,23-tetrasulfonic acid, GLYCEROL, Lysozyme C
著者McGovern, R.E, Lyons, J.A, Crowley, P.B.
登録日2014-03-06
公開日2014-11-12
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural study of a small molecule receptor bound to dimethyllysine in lysozyme.
Chem Sci, 6, 2015
4HB4
DownloadVisualize
BU of 4hb4 by Molmil
Crystal structure of CRM1 inhibitor Leptomycin B in complex with CRM1(537DLTVK541/GLCEQ)-Ran-RanBP1
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, Exportin-1, ...
著者Sun, Q, Chook, Y.M.
登録日2012-09-27
公開日2013-01-09
最終更新日2017-07-26
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Nuclear export inhibition through covalent conjugation and hydrolysis of Leptomycin B by CRM1.
Proc.Natl.Acad.Sci.USA, 110, 2013
4HCX
DownloadVisualize
BU of 4hcx by Molmil
Structure of ICDH-1 from M.tuberculosis complexed with NADPH & Mn2+
分子名称: CHLORIDE ION, Isocitrate dehydrogenase [NADP], MANGANESE (II) ION, ...
著者Hazra, S, Blanchard, J.
登録日2012-10-01
公開日2013-02-27
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献Structural, Kinetic and Chemical Mechanism of Isocitrate Dehydrogenase-1 from Mycobacterium tuberculosis.
Biochemistry, 52, 2013

222926

件を2024-07-24に公開中

PDB statisticsPDBj update infoContact PDBjnumon