8ABP
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4GNK
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7ABP
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2RGN
| Crystal Structure of p63RhoGEF complex with Galpha-q and RhoA | 分子名称: | GUANOSINE-5'-DIPHOSPHATE, Guanine nucleotide-binding protein G(i) subunit alpha-1,Guanine nucleotide-binding protein G(q) subunit alpha, MAGNESIUM ION, ... | 著者 | Shankaranarayanan, A, Nance, M.R, Tesmer, J.J.G. | 登録日 | 2007-10-04 | 公開日 | 2008-01-15 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | Structure of Galphaq-p63RhoGEF-RhoA complex reveals a pathway for the activation of RhoA by GPCRs. Science, 318, 2007
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3UZT
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3UZS
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3C4W
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3C4Z
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3NYO
| Crystal Structure of G Protein-Coupled Receptor Kinase 6 in Complex with AMP | 分子名称: | (R,R)-2,3-BUTANEDIOL, ADENOSINE MONOPHOSPHATE, G protein-coupled receptor kinase 6, ... | 著者 | Tesmer, J.J.G, Singh, P. | 登録日 | 2010-07-15 | 公開日 | 2010-09-22 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.92 Å) | 主引用文献 | Molecular basis for activation of G protein-coupled receptor kinases. Embo J., 29, 2010
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3NYN
| Crystal Structure of G Protein-Coupled Receptor Kinase 6 in Complex with Sangivamycin | 分子名称: | (R,R)-2,3-BUTANEDIOL, G protein-coupled receptor kinase 6, SANGIVAMYCIN, ... | 著者 | Tesmer, J.J.G, Singh, P. | 登録日 | 2010-07-15 | 公開日 | 2010-09-22 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.72 Å) | 主引用文献 | Molecular basis for activation of G protein-coupled receptor kinases. Embo J., 29, 2010
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4L9I
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4MK0
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4EKD
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4EKC
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6MVD
| Crystal structure of Lecithin:cholesterol acyltransferase (LCAT) in complex with isopropyl dodec-11-enylfluorophosphonate (IDFP) and a small molecule activator | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 6-{4-[(4R)-4-hydroxy-6-oxo-4-(trifluoromethyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]pyridin-3-yl]piperidin-1-yl}-4-(trifluoromethyl)pyridine-3-carbonitrile, NICKEL (II) ION, ... | 著者 | Manthei, K.A, Chang, L, Tesmer, J.J.G. | 登録日 | 2018-10-25 | 公開日 | 2018-12-05 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Molecular basis for activation of lecithin:cholesterol acyltransferase by a compound that increases HDL cholesterol. Elife, 7, 2018
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2I1K
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2I1J
| Moesin from Spodoptera frugiperda at 2.1 angstroms resolution | 分子名称: | CHLORIDE ION, GLYCEROL, Moesin, ... | 著者 | Li, Q, Nance, M.R, Tesmer, J.J.G. | 登録日 | 2006-08-14 | 公開日 | 2006-12-19 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Self-masking in an Intact ERM-merlin Protein: An Active Role for the Central alpha-Helical Domain. J.Mol.Biol., 365, 2007
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3V5W
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3QR0
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3QR1
| Crystal Structure of L. pealei PLC21 | 分子名称: | CALCIUM ION, PHOSPHOLIPASE C-BETA (PLC-BETA) | 著者 | Lyon, A.M, Suddala, K.C, Northup, J.K, Tesmer, J.J.G. | 登録日 | 2011-02-16 | 公開日 | 2011-08-10 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | An autoinhibitory helix in the C-terminal region of phospholipase C-beta mediates Galphaq activation. Nat.Struct.Mol.Biol., 18, 2011
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4WBO
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4X94
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4WNK
| Crystal Structure of Bovine G Protein Coupled-Receptor Kinase 5 in Complex with CCG215022 | 分子名称: | (4S)-4-{4-fluoro-3-[(pyridin-2-ylmethyl)carbamoyl]phenyl}-N-(1H-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide, G protein-coupled receptor kinase 5, SULFATE ION | 著者 | Homan, K.T, Tesmer, J.J.G. | 登録日 | 2014-10-13 | 公開日 | 2015-06-10 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.42 Å) | 主引用文献 | Crystal Structure of G Protein-coupled Receptor Kinase 5 in Complex with a Rationally Designed Inhibitor. J.Biol.Chem., 290, 2015
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4X90
| Crystal structure of Lysosomal Phospholipase A2 | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ... | 著者 | Glukhova, A, Tesmer, J.J.G. | 登録日 | 2014-12-11 | 公開日 | 2015-03-11 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.84 Å) | 主引用文献 | Structure and function of lysosomal phospholipase A2 and lecithin:cholesterol acyltransferase. Nat Commun, 6, 2015
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4X91
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