3ACA
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3W3M
| Crystal structure of human TLR8 in complex with Resiquimod (R848) crystal form 2 | 分子名称: | 1-[4-amino-2-(ethoxymethyl)-1H-imidazo[4,5-c]quinolin-1-yl]-2-methylpropan-2-ol, 2-acetamido-2-deoxy-beta-D-glucopyranose, SULFATE ION, ... | 著者 | Tanji, H, Ohto, U, Shimizu, T. | 登録日 | 2012-12-22 | 公開日 | 2013-04-03 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Structural reorganization of the Toll-like receptor 8 dimer induced by agonistic ligands Science, 339, 2013
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3WPF
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3W3K
| Crystal structure of human TLR8 in complex with CL075 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-propyl[1,3]thiazolo[4,5-c]quinolin-4-amine, ... | 著者 | Tanji, H, Ohto, U, Shimizu, T. | 登録日 | 2012-12-22 | 公開日 | 2013-04-03 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural reorganization of the Toll-like receptor 8 dimer induced by agonistic ligands Science, 339, 2013
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3WPD
| Crystal structure of horse TLR9 in complex with inhibitory DNA4084 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, DNA (5'-D(*CP*CP*TP*GP*GP*AP*TP*GP*GP*G)-3'), ... | 著者 | Ohto, U, Tanji, H, Shimizu, T. | 登録日 | 2014-01-11 | 公開日 | 2015-02-11 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.75 Å) | 主引用文献 | Structural basis of CpG and inhibitory DNA recognition by Toll-like receptor 9 Nature, 520, 2015
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3W3J
| Crystal structure of human TLR8 in complex with CL097 | 分子名称: | 2-(ethoxymethyl)-1H-imidazo[4,5-c]quinolin-4-amine, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Tanji, H, Ohto, U, Shimizu, T. | 登録日 | 2012-12-22 | 公開日 | 2013-04-03 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structural reorganization of the Toll-like receptor 8 dimer induced by agonistic ligands Science, 339, 2013
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3WPG
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3WPI
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3W3L
| Crystal structure of human TLR8 in complex with Resiquimod (R848) crystal form 1 | 分子名称: | 1-[4-amino-2-(ethoxymethyl)-1H-imidazo[4,5-c]quinolin-1-yl]-2-methylpropan-2-ol, 2-acetamido-2-deoxy-beta-D-glucopyranose, SULFATE ION, ... | 著者 | Tanji, H, Ohto, U, Shimizu, T. | 登録日 | 2012-12-22 | 公開日 | 2013-04-03 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.33 Å) | 主引用文献 | Structural reorganization of the Toll-like receptor 8 dimer induced by agonistic ligands Science, 339, 2013
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3WPE
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3W3N
| Crystal structure of human TLR8 in complex with Resiquimod (R848) crystal form 3 | 分子名称: | 1-[4-amino-2-(ethoxymethyl)-1H-imidazo[4,5-c]quinolin-1-yl]-2-methylpropan-2-ol, 2-acetamido-2-deoxy-beta-D-glucopyranose, GLYCEROL, ... | 著者 | Tanji, H, Ohto, U, Shimizu, T. | 登録日 | 2012-12-22 | 公開日 | 2013-04-03 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structural reorganization of the Toll-like receptor 8 dimer induced by agonistic ligands Science, 339, 2013
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3WPB
| Crystal structure of horse TLR9 (unliganded form) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, SULFATE ION, ... | 著者 | Ohto, U, Tanji, H, Shimizu, T. | 登録日 | 2014-01-11 | 公開日 | 2015-02-11 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structural basis of CpG and inhibitory DNA recognition by Toll-like receptor 9 Nature, 520, 2015
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3WPH
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3WPC
| Crystal structure of horse TLR9 in complex with agonistic DNA1668_12mer | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, DNA (5'-D(*CP*AP*TP*GP*AP*CP*GP*TP*TP*CP*CP*T)-3'), ... | 著者 | Ohto, U, Tanji, H, Shimizu, T. | 登録日 | 2014-01-11 | 公開日 | 2015-02-11 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Structural basis of CpG and inhibitory DNA recognition by Toll-like receptor 9 Nature, 520, 2015
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3AC9
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1AY4
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1AY5
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1AY8
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2DDQ
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1VHR
| HUMAN VH1-RELATED DUAL-SPECIFICITY PHOSPHATASE | 分子名称: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, HUMAN VH1-RELATED DUAL-SPECIFICITY PHOSPHATASE VHR, SULFATE ION | 著者 | Yuvaniyama, J, Denu, J.M, Dixon, J.E, Saper, M.A. | 登録日 | 1996-02-20 | 公開日 | 1996-06-20 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Crystal structure of the dual specificity protein phosphatase VHR. Science, 272, 1996
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3A73
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1VDH
| Structure-based functional identification of a novel heme-binding protein from thermus thermophilus HB8 | 分子名称: | muconolactone isomerase-like protein | 著者 | Ebihara, A, Okamoto, A, Kousumi, Y, Yamamoto, H, Masui, R, Ueyama, N, Shibata, T, Inoue, Y, Yokoyama, S, Kuramitsu, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2004-03-22 | 公開日 | 2004-09-22 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure-based functional identification of a novel heme-binding protein from Thermus thermophilus HB8. J.STRUCT.FUNCT.GENOM., 6, 2005
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2AY3
| AROMATIC AMINO ACID AMINOTRANSFERASE WITH 3-(3,4-DIMETHOXYPHENYL)PROPIONIC ACID | 分子名称: | 3-(3,4-DIMETHOXYPHENYL)PROPIONIC ACID, AROMATIC AMINO ACID AMINOTRANSFERASE, PYRIDOXAL-5'-PHOSPHATE | 著者 | Okamoto, A, Hirotsu, K, Kagamiyama, H. | 登録日 | 1998-08-06 | 公開日 | 1999-02-02 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | The active site of Paracoccus denitrificans aromatic amino acid aminotransferase has contrary properties: flexibility and rigidity. Biochemistry, 38, 1999
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2AY9
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2AY6
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