6GR7
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![BU of 6gr7 by Molmil](/molmil-images/mine/6gr7) | Crystal Structure Of Human Transthyretin in complex with 2,4,5-trichlorophenoxyacetic acid (2,4,5-T) | 分子名称: | 2-[2,4,5-tris(chloranyl)phenoxy]ethanoic acid, Transthyretin | 著者 | Grundstrom, C, Zhang, J, Olofsson, A, Andersson, P.L, Sauer-Eriksson, A.E. | 登録日 | 2018-06-09 | 公開日 | 2018-07-11 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Interspecies Variation between Fish and Human Transthyretins in Their Binding of Thyroid-Disrupting Chemicals. Environ. Sci. Technol., 52, 2018
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7U8C
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![BU of 7u8c by Molmil](/molmil-images/mine/7u8c) | Crystal structure of Mesothelin C-terminal peptide-MORAb 15B6 FAB complex | 分子名称: | MORab 15B6 Fab heavy chain, MORab 15B6 Fab light chain, Mesothelin, ... | 著者 | Zhan, J, Esser, L, Xia, D. | 登録日 | 2022-03-08 | 公開日 | 2022-06-08 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Highly active CAR T cells that bind to a juxtamembrane region of mesothelin and are not blocked by shed mesothelin. Proc.Natl.Acad.Sci.USA, 119, 2022
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6CUR
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![BU of 6cur by Molmil](/molmil-images/mine/6cur) | Ras:SOS:Ras in complex with a small molecule activator | 分子名称: | FORMIC ACID, GLYCEROL, GTPase HRas, ... | 著者 | Phan, J, Abbott, J, Fesik, S.W. | 登録日 | 2018-03-26 | 公開日 | 2019-02-06 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.73 Å) | 主引用文献 | Discovery of Quinazolines That Activate SOS1-Mediated Nucleotide Exchange on RAS. ACS Med Chem Lett, 9, 2018
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6CUO
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![BU of 6cuo by Molmil](/molmil-images/mine/6cuo) | Ras:SOS:Ras in complex with a small molecule activator | 分子名称: | FORMIC ACID, GLYCEROL, GTPase HRas, ... | 著者 | Phan, J, Abbott, J, Fesik, S.W. | 登録日 | 2018-03-26 | 公開日 | 2019-02-06 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.73 Å) | 主引用文献 | Discovery of Quinazolines That Activate SOS1-Mediated Nucleotide Exchange on RAS. ACS Med Chem Lett, 9, 2018
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6E1Z
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6DAI
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![BU of 6dai by Molmil](/molmil-images/mine/6dai) | Discovery of Potent 2-Aryl-6,7-Dihydro-5HPyrrolo[ 1,2-a]imidazoles as WDR5 WIN-site Inhibitors Using Fragment-Based Methods and Structure-Based Design | 分子名称: | 6-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-2-yl)-1-methylindoline, DIMETHYL SULFOXIDE, WD repeat-containing protein 5 | 著者 | Phan, J, Fesik, S.W. | 登録日 | 2018-05-01 | 公開日 | 2018-09-05 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.63 Å) | 主引用文献 | Discovery of Potent 2-Aryl-6,7-dihydro-5 H-pyrrolo[1,2- a]imidazoles as WDR5-WIN-Site Inhibitors Using Fragment-Based Methods and Structure-Based Design. J. Med. Chem., 61, 2018
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5JRE
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7U8H
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![BU of 7u8h by Molmil](/molmil-images/mine/7u8h) | Discovery of a KRAS G12V Inhibitor in vivo Tool Compound starting from an HSQC-NMR based Fragment Hit | 分子名称: | 1H-benzimidazol-2-ylmethanethiol, 2-amino-4,5,6,7-tetrahydro-1-benzothiophene-3-carbonitrile, GTPase KRas, ... | 著者 | Phan, J, Fesik, S.W. | 登録日 | 2022-03-08 | 公開日 | 2022-11-09 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.702 Å) | 主引用文献 | Fragment Optimization of Reversible Binding to the Switch II Pocket on KRAS Leads to a Potent, In Vivo Active KRAS G12C Inhibitor. J.Med.Chem., 65, 2022
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4WUJ
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![BU of 4wuj by Molmil](/molmil-images/mine/4wuj) | Structural Biochemistry of a Fungal LOV Domain Photoreceptor Reveals an Evolutionarily Conserved Pathway Integrating Blue-Light and Oxidative Stress | 分子名称: | FLAVIN MONONUCLEOTIDE, Glycoside hydrolase family 15, cellulose signaling associated protein envoy, ... | 著者 | Hopkins, H.C, Lokhandwala, J, Zoltowski, B.D. | 登録日 | 2014-10-31 | 公開日 | 2015-01-14 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.23 Å) | 主引用文献 | Structural Biochemistry of a Fungal LOV Domain Photoreceptor Reveals an Evolutionarily Conserved Pathway Integrating Light and Oxidative Stress. Structure, 23, 2015
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7V3P
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![BU of 7v3p by Molmil](/molmil-images/mine/7v3p) | Cryo-EM structure of the IGF1R/insulin complex | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Insulin A chain, Insulin B chain, ... | 著者 | Zhang, J, Liu, C, Zhang, X, Wei, T, Wu, C. | 登録日 | 2021-08-11 | 公開日 | 2022-08-17 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Cryo-EM structure of the IGF1R/insulin complex To Be Published
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6UJH
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6UJL
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8DSG
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![BU of 8dsg by Molmil](/molmil-images/mine/8dsg) | P411-PFA carbene transferase | 分子名称: | 1,2-ETHANEDIOL, 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Cytochrome P450-BM3 variant P411-PFA, ... | 著者 | Maggiolo, A.O, Porter, N.J, Zhang, J, Arnold, F.H. | 登録日 | 2022-07-22 | 公開日 | 2023-03-08 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | Chemodivergent C(sp 3 )-H and C(sp 2 )-H Cyanomethylation Using Engineered Carbene Transferases. Nat Catal, 6, 2023
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6V9J
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6UJJ
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6V9M
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![BU of 6v9m by Molmil](/molmil-images/mine/6v9m) | |
6V9N
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6V9L
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6V9F
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5JID
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![BU of 5jid by Molmil](/molmil-images/mine/5jid) | Crystal Structure of Human Transthyretin in Complex with Perfluorooctanoic acid (PFOA) | 分子名称: | SODIUM ION, Transthyretin, pentadecafluorooctanoic acid | 著者 | Begum, A, Zhang, J, Olofsson, A, Andersson, P, Sauer-Eriksson, A.E. | 登録日 | 2016-04-22 | 公開日 | 2016-10-05 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.2 Å) | 主引用文献 | Structure-Based Virtual Screening Protocol for in Silico Identification of Potential Thyroid Disrupting Chemicals Targeting Transthyretin. Environ. Sci. Technol., 50, 2016
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5JIQ
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![BU of 5jiq by Molmil](/molmil-images/mine/5jiq) | Crystal Structure of Human Transthyretin in Complex with 2,2',4,4'-tetrahydroxybenzophenone (BP2) | 分子名称: | GLYCEROL, SODIUM ION, Transthyretin, ... | 著者 | Begum, A, Zhang, J, Olofsson, A, Andersson, P, Sauer-Eriksson, A.E. | 登録日 | 2016-04-22 | 公開日 | 2016-10-05 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Structure-Based Virtual Screening Protocol for in Silico Identification of Potential Thyroid Disrupting Chemicals Targeting Transthyretin. Environ. Sci. Technol., 50, 2016
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5JIM
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![BU of 5jim by Molmil](/molmil-images/mine/5jim) | Crystal Structure of Human Transthyretin in Complex with Perfluoroktansulfonsyra (PFOS) | 分子名称: | SODIUM ION, Transthyretin, heptadecafluoro-1-octanesulfonic acid | 著者 | Begum, A, Zhang, J, Olofsson, A, Andersson, P, Sauer-Eriksson, A.E. | 登録日 | 2016-04-22 | 公開日 | 2016-10-05 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.26 Å) | 主引用文献 | Structure-Based Virtual Screening Protocol for in Silico Identification of Potential Thyroid Disrupting Chemicals Targeting Transthyretin. Environ. Sci. Technol., 50, 2016
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7KGB
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6TC6
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6TC9
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![BU of 6tc9 by Molmil](/molmil-images/mine/6tc9) | Crystal structure of MutM from Neisseria meningitidis | 分子名称: | DNA, DNA containing abasic site analogue, Formamidopyrimidine-DNA glycosylase, ... | 著者 | Silhan, J, Landova, B, Boura, E. | 登録日 | 2019-11-05 | 公開日 | 2020-09-16 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.175 Å) | 主引用文献 | Conformational changes of DNA repair glycosylase MutM triggered by DNA binding. Febs Lett., 594, 2020
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