5H36
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![BU of 5h36 by Molmil](/molmil-images/mine/5h36) | Crystal structures of the TRIC trimeric intracellular cation channel orthologue from Rhodobacter sphaeroides | Descriptor: | 1,2-DIMYRISTOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, Uncharacterized protein TRIC | Authors: | Kasuya, G, Hiraizumi, M, Hattori, M, Nureki, O. | Deposit date: | 2016-10-20 | Release date: | 2017-01-11 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (3.409 Å) | Cite: | Crystal structures of the TRIC trimeric intracellular cation channel orthologues Cell Res., 26, 2016
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6NAD
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5Z66
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![BU of 5z66 by Molmil](/molmil-images/mine/5z66) | Structure of periplasmic trehalase from Diamondback moth gut bacteria complexed with validoxylamine | Descriptor: | (1S,2S,3R,6S)-4-(HYDROXYMETHYL)-6-{[(1S,2S,3S,4R,5R)-2,3,4-TRIHYDROXY-5-(HYDROXYMETHYL)CYCLOHEXYL]AMINO}CYCLOHEX-4-ENE-1,2,3-TRIOL, GLYCEROL, Periplasmic trehalase, ... | Authors: | Harne, S.R, Adhav, A.S, Joshi, R.S, Gayathri, P. | Deposit date: | 2018-01-22 | Release date: | 2019-01-23 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Mechanistic insights into enzymatic catalysis by trehalase from the insect gut endosymbiont Enterobacter cloacae. Febs J., 286, 2019
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5ZTF
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![BU of 5ztf by Molmil](/molmil-images/mine/5ztf) | Structure of Ca2+ ATPase | Descriptor: | CALCIUM ION, MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, ... | Authors: | Inoue, M, Watanabe, S, Inaba, K. | Deposit date: | 2018-05-03 | Release date: | 2019-05-22 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (3.45 Å) | Cite: | Structural Basis of Sarco/Endoplasmic Reticulum Ca2+-ATPase 2b Regulation via Transmembrane Helix Interplay. Cell Rep, 27, 2019
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5Z6H
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![BU of 5z6h by Molmil](/molmil-images/mine/5z6h) | Structure of periplasmic trehalase from Diamondback moth gut bacteria in the apo form | Descriptor: | GLYCEROL, Periplasmic trehalase, SULFATE ION | Authors: | Harne, S.R, Adhav, A.S, Joshi, R.S, Gayathri, P. | Deposit date: | 2018-01-22 | Release date: | 2019-01-23 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Mechanistic insights into enzymatic catalysis by trehalase from the insect gut endosymbiont Enterobacter cloacae. Febs J., 286, 2019
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8FSL
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7FH2
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![BU of 7fh2 by Molmil](/molmil-images/mine/7fh2) | Crystal structure of the first bromodomain of BRD4 in complex with 16D10 | Descriptor: | Bromodomain-containing protein 4, CHLORIDE ION, N-[2-[2-[(E)-3-(2,5-dimethoxyphenyl)prop-2-enoyl]-4,5-dimethoxy-phenyl]ethyl]ethanamide | Authors: | Yokoyama, T, Hirasawa, N. | Deposit date: | 2021-07-29 | Release date: | 2022-08-03 | Last modified: | 2023-11-29 | Method: | X-RAY DIFFRACTION (2.492 Å) | Cite: | A chalcone derivative suppresses TSLP induction in mice and human keratinocytes through binding to BET family proteins. Biochem Pharmacol, 194, 2021
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6JJU
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![BU of 6jju by Molmil](/molmil-images/mine/6jju) | Structure of Ca2+ ATPase | Descriptor: | CALCIUM ION, MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, ... | Authors: | Inoue, M, Sakuta, N, Watanabe, S, Inaba, K. | Deposit date: | 2019-02-27 | Release date: | 2019-05-22 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (3.2 Å) | Cite: | Structural Basis of Sarco/Endoplasmic Reticulum Ca2+-ATPase 2b Regulation via Transmembrane Helix Interplay. Cell Rep, 27, 2019
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3CD8
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![BU of 3cd8 by Molmil](/molmil-images/mine/3cd8) | X-ray Structure of c-Met with triazolopyridazine Inhibitor. | Descriptor: | 7-methoxy-4-[(6-phenyl[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methoxy]quinoline, Hepatocyte growth factor receptor | Authors: | Bellon, S.F, Albrecht, B.K, Harmange, J.-C, Bauer, D, Choquette, D, Dussault, I. | Deposit date: | 2008-02-26 | Release date: | 2008-04-29 | Last modified: | 2023-08-30 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Discovery and Optimization of Triazolopyridazines as Potent and Selective Inhibitors of the c-Met Kinase. J.Med.Chem., 51, 2008
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7NMZ
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5GHK
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![BU of 5ghk by Molmil](/molmil-images/mine/5ghk) | Crystal Structure Analysis of Canine serum albumin | Descriptor: | Serum albumin | Authors: | Kihira, K, Yamada, K, Kureishi, M, Yokomaku, K, Shinohara, R, Akiyama, M, Komatsu, T. | Deposit date: | 2016-06-20 | Release date: | 2016-11-23 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (3.2 Å) | Cite: | Artificial Blood for Dogs Sci Rep, 6, 2016
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3APQ
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3CCN
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![BU of 3ccn by Molmil](/molmil-images/mine/3ccn) | X-ray structure of c-Met with triazolopyridazine inhibitor. | Descriptor: | 4-[(6-phenyl[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methyl]phenol, Hepatocyte growth factor receptor | Authors: | Abrecht, B.K, Harmange, J.-C, Bauer, D, Dussault, I, long, A, Bellon, S.F. | Deposit date: | 2008-02-26 | Release date: | 2008-04-29 | Last modified: | 2023-08-30 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Discovery and Optimization of Triazolopyridazines as Potent and Selective Inhibitors of the c-Met Kinase. J.Med.Chem., 51, 2008
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3APO
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![BU of 3apo by Molmil](/molmil-images/mine/3apo) | Crystal structure of full-length ERdj5 | Descriptor: | DnaJ homolog subfamily C member 10 | Authors: | Inaba, K, Suzuki, M, Nagata, K. | Deposit date: | 2010-10-20 | Release date: | 2011-04-20 | Last modified: | 2011-07-13 | Method: | X-RAY DIFFRACTION (2.4 Å) | Cite: | Structural basis of an ERAD pathway mediated by the ER-resident protein disulfide reductase ERdj5. Mol.Cell, 41, 2011
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3APS
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![BU of 3aps by Molmil](/molmil-images/mine/3aps) | Crystal structure of Trx4 domain of ERdj5 | Descriptor: | DnaJ homolog subfamily C member 10, GLYCEROL, SULFATE ION | Authors: | Inaba, K, Suzuki, M, Nagata, K. | Deposit date: | 2010-10-20 | Release date: | 2011-04-20 | Last modified: | 2011-07-13 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Structural basis of an ERAD pathway mediated by the ER-resident protein disulfide reductase ERdj5. Mol.Cell, 41, 2011
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1A0K
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3LH0
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3LM5
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![BU of 3lm5 by Molmil](/molmil-images/mine/3lm5) | Crystal Structure of human Serine/Threonine Kinase 17B (STK17B) in complex with Quercetin | Descriptor: | 3,5,7,3',4'-PENTAHYDROXYFLAVONE, Serine/threonine-protein kinase 17B | Authors: | Ugochukwu, E, Soundararajan, M, Rellos, P, Fedorov, O, Phillips, C, Wang, J, Hapka, E, Filippakopoulos, P, Chaikuad, A, Pike, A.C.W, Carpenter, L, Vollmar, M, von Delft, F, Bountra, C, Arrowsmith, C.H, Weigelt, J, Edwards, A, Knapp, S, Structural Genomics Consortium (SGC) | Deposit date: | 2010-01-29 | Release date: | 2010-03-16 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (2.29 Å) | Cite: | A Chemical Probe for Dark Kinase STK17B Derives Its Potency and High Selectivity through a Unique P-Loop Conformation. J.Med.Chem., 63, 2020
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5X9H
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3LGF
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3LGL
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5X9G
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5XQN
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![BU of 5xqn by Molmil](/molmil-images/mine/5xqn) | Crystal structure of Notched-fin eelpout type III antifreeze protein (NFE6, AFP), C2221 form. | Descriptor: | Ice-structuring protein, SULFATE ION | Authors: | Adachi, M, Kondo, H, Tsuda, S. | Deposit date: | 2017-06-07 | Release date: | 2018-05-16 | Last modified: | 2024-03-27 | Method: | X-RAY DIFFRACTION (1.19 Å) | Cite: | Polypentagonal ice-like water networks emerge solely in an activity-improved variant of ice-binding protein Proc. Natl. Acad. Sci. U.S.A., 115, 2018
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5GW9
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![BU of 5gw9 by Molmil](/molmil-images/mine/5gw9) | Crystal structure of C163, a backbone circularized G-CSF | Descriptor: | Granulocyte colony-stimulating factor | Authors: | Miyafusa, T, Honda, S. | Deposit date: | 2016-09-09 | Release date: | 2017-09-13 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (1.65 Å) | Cite: | Structural insights into the backbone-circularized granulocyte colony-stimulating factor containing a short connector. Biochem. Biophys. Res. Commun., 500, 2018
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5GMT
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