5UVV
BRD4 Bromodomain 2 with A-1457066
Summary for 5UVV
Entry DOI | 10.2210/pdb5uvv/pdb |
Related | 5UVS 5UVT 5UVU 5UVW 5UVX 5UVY 5UVZ |
Descriptor | Bromodomain-containing protein 4, 7-(cyclopropylmethyl)-10-(ethylsulfonyl)-2-methyl-2,4,6,7-tetrahydro-3H-2,4,7-triazadibenzo[cd,f]azulen-3-one (3 entities in total) |
Functional Keywords | helix bundle, signaling protein-inhibitor complex, signaling protein/inhibitor |
Biological source | Homo sapiens (Human) |
Cellular location | Nucleus: O60885 |
Total number of polymer chains | 2 |
Total formula weight | 26408.85 |
Authors | Park, C.H. (deposition date: 2017-02-20, release date: 2017-06-21, Last modification date: 2024-03-06) |
Primary citation | Park, C.H. BRD4 Bromodomain 2 with A-1457066 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.99 Å) |
Structure validation
Download full validation report