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5UVV

BRD4 Bromodomain 2 with A-1457066

Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue 8NS A 501
ChainResidue
ATRP374
APRO375
APRO379
AVAL380
AASP381
ALEU385
AASN433
AVAL439
AHOH610

site_idAC2
Number of Residues9
Detailsbinding site for residue 8NS B 501
ChainResidue
BTRP374
BPRO375
BLYS378
BPRO379
BVAL380
BASP381
BLEU385
BASN433
BHOH611

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsSite: {"description":"Acetylated histone binding","evidences":[{"source":"PubMed","id":"22464331","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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