5UVV

BRD4 Bromodomain 2 with A-1457066

Summary for 5UVV

• Entry DOI: 10.2210/pdb5uvv/pdb
• Related: 5UVS 5UVT 5UVU 5UVW 5UVX 5UVY 5UVZ
• Descriptor: Bromodomain-containing protein 4, 7-(cyclopropylmethyl)-10-(ethylsulfonyl)-2-methyl-2,4,6,7-tetrahydro-3H-2,4,7-triazadibenzo[cd,f]azulen-3-one (3 entities in total)
• Functional Keywords: helix bundle, signaling protein-inhibitor complex, signaling protein/inhibitor
• Biological source: Homo sapiens (Human)
• Cellular location: Nucleus: O60885
• Total number of polymer chains: 2
• Total formula weight: 26408.85

Authors

Park, C.H. (deposition date: 2017-02-20, release date: 2017-06-21, Last modification date: 2024-03-06)

• Primary citation: Park, C.H.; BRD4 Bromodomain 2 with A-1457066; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.99 Å)