5UVX
BRD4 Bromodomain 2 with A-1359643
Summary for 5UVX
Entry DOI | 10.2210/pdb5uvx/pdb |
Related | 5UVS 5UVT 5UVU 5UVV 5UVW 5UVY 5UVZ |
Descriptor | Bromodomain-containing protein 4, N-[3-(6-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl)-4-phenoxyphenyl]methanesulfonamide (3 entities in total) |
Functional Keywords | helix bundle, signaling protein-inhibitor complex, signaling protein/inhibitor |
Biological source | Homo sapiens (Human) |
Cellular location | Nucleus: O60885 |
Total number of polymer chains | 2 |
Total formula weight | 26432.78 |
Authors | Park, C.H. (deposition date: 2017-02-20, release date: 2017-06-21, Last modification date: 2024-03-06) |
Primary citation | Park, C.H. BRD4 Bromodomain 2 with A-1359643 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.53 Å) |
Structure validation
Download full validation report