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5UVW

BRD4_Bromodomain1-A1376855

Summary for 5UVW
Entry DOI10.2210/pdb5uvw/pdb
Related5UVS 5UVT 5UVU 5UVV 5UVX 5UVY 5UVZ
DescriptorBromodomain-containing protein 4, N-[4-(2,4-difluorophenoxy)-3-(6-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl)phenyl]ethanesulfonamide, SULFATE ION, ... (4 entities in total)
Functional Keywordshelix bundle brd4 bromodomain 1 - inhibitor complex three complexes per asymmetric unit, signaling protein-inhibitor complex, signaling protein/inhibitor
Biological sourceHomo sapiens (Human)
Cellular locationNucleus: O60885
Total number of polymer chains3
Total formula weight41021.42
Authors
Park, C.H. (deposition date: 2017-02-20, release date: 2017-06-21, Last modification date: 2024-03-06)
Primary citationPark, C.H.
BRD4_Bromodomain1-A1376855
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.14 Å)
Structure validation

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PDB entries from 2024-04-17

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