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5UVY

BRD4 Bromodomain 2 with A-1349391

Summary for 5UVY
Entry DOI10.2210/pdb5uvy/pdb
Related5UVS 5UVT 5UVU 5UVV 5UVW 5UVX 5UVZ
DescriptorBromodomain-containing protein 4, 6-methyl-4-(2-phenoxyphenyl)-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one (3 entities in total)
Functional Keywordshelix bundle, signaling protein-inhibitor complex, signaling protein/inhibitor
Biological sourceHomo sapiens (Human)
Cellular locationNucleus: O60885
Total number of polymer chains1
Total formula weight13123.29
Authors
Park, C.H. (deposition date: 2017-02-20, release date: 2017-06-14, Last modification date: 2024-03-06)
Primary citationPark, C.H.
BRD4 Bromodomain 2 with A-1349391
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.25 Å)
Structure validation

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PDB entries from 2024-04-17

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