5UVT
BRD4_BD2_A-1454056
Summary for 5UVT
Entry DOI | 10.2210/pdb5uvt/pdb |
Related | 5UVS 5UVU 5UVV 5UVW 5UVX 5UVY 5UVZ |
Descriptor | Bromodomain-containing protein 4, 7-(cyclopropylmethyl)-2-methyl-10-[(propan-2-yl)sulfonyl]-2,4,6,7-tetrahydro-3H-2,4,7-triazadibenzo[cd,f]azulen-3-one (3 entities in total) |
Functional Keywords | helix bundle, signaling protein-inhibitor complex, signaling protein/inhibitor |
Biological source | Homo sapiens (Human) |
Cellular location | Nucleus: O60885 |
Total number of polymer chains | 1 |
Total formula weight | 13218.45 |
Authors | Park, C.H. (deposition date: 2017-02-20, release date: 2017-06-21, Last modification date: 2024-04-03) |
Primary citation | Park, C.H. Complex structure of BRD4_BD2_A-1454056 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.67 Å) |
Structure validation
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