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4A51

Crystal structure of human kinesin Eg5 in complex with 1-(3-(((2-Aminoethyl)thio)diphenylmethyl)phenyl)ethanone hydrochloride

Summary for 4A51
Entry DOI10.2210/pdb4a51/pdb
Related1II6 1Q0B 1X88 1YRS 2FKY 2FL2 2FL6 2G1Q 2GM1 2UYI 2UYM 2WOG 2X2R 2X7C 2X7D 2X7E 2XAE 4A1Z 4A28 4A2T 4A50
DescriptorKINESIN-LIKE PROTEIN KIF11, ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ... (7 entities in total)
Functional Keywordscell cycle, mitosis, inhibitor, ksp
Biological sourceHOMO SAPIENS (HUMAN)
Cellular locationCytoplasm: P52732
Total number of polymer chains7
Total formula weight293672.52
Authors
Kaan, H.Y.K.,Kozielski, F. (deposition date: 2011-10-24, release date: 2012-10-31, Last modification date: 2023-12-20)
Primary citationWang, F.,Good, J.A.D.,Rath, O.,Kaan, H.Y.K.,Sutcliffe, O.B.,Mackay, S.P.,Kozielski, F.
Triphenylbutanamines: Kinesin Spindle Protein Inhibitors with in Vivo Antitumor Activity.
J.Med.Chem., 55:1511-, 2012
Cited by
PubMed: 22248262
DOI: 10.1021/JM201195M
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.75 Å)
Structure validation

217157

건을2024-03-13부터공개중

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