4A1Z
Eg5-1
Summary for 4A1Z
Entry DOI | 10.2210/pdb4a1z/pdb |
Related | 1II6 1Q0B 1X88 1YRS 2FKY 2FL2 2FL6 2G1Q 2GM1 2UYI 2UYM 2WOG 2X2R 2X7C 2X7D 2X7E 2XAE |
Descriptor | KINESIN-LIKE PROTEIN KIF11, MAGNESIUM ION, NITRATE ION, ... (5 entities in total) |
Functional Keywords | motor protein |
Biological source | HOMO SAPIENS (HUMAN) |
Cellular location | Cytoplasm: P52732 |
Total number of polymer chains | 2 |
Total formula weight | 83106.27 |
Authors | Talapatra, S.K.,Kozielski, F. (deposition date: 2011-09-20, release date: 2012-10-31, Last modification date: 2023-12-20) |
Primary citation | Talapatra, S.K.,Anthony, N.G.,Mackay, S.P.,Kozielski, F. The Mitotic Kinesin Eg5 Overcomes Inhibition to the Phase I/II Clinical Candidate Sb743921 by an Allosteric Resistance Mechanism. J.Med.Chem., 56:6317-, 2013 Cited by PubMed: 23875972DOI: 10.1021/JM4006274 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.8 Å) |
Structure validation
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