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1F88
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BU of 1f88 by Molmil
CRYSTAL STRUCTURE OF BOVINE RHODOPSIN
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, MERCURY (II) ION, RETINAL, ...
Authors:Okada, T, Palczewski, K, Stenkamp, R.E, Miyano, M.
Deposit date:2000-06-29
Release date:2000-08-04
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:Crystal structure of rhodopsin: A G protein-coupled receptor.
Science, 289, 2000
4CJ6
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BU of 4cj6 by Molmil
Crystal structure of the complex of the Cellular Retinal Binding Protein Mutant R234W with 9-cis-retinal
Descriptor: RETINAL, RETINALDEHYDE-BINDING PROTEIN 1
Authors:Bolze, C.S, Helbling, R.E, Owen, R.L, Pearson, A.R, Pompidor, G, Dworkowski, F, Fuchs, M.R, Furrer, J, Golczak, M, Palczewski, K, Cascella, M, Stocker, A.
Deposit date:2013-12-19
Release date:2014-01-08
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (1.896 Å)
Cite:Human Cellular Retinaldehyde-Binding Protein Has Secondary Thermal 9-Cis-Retinal Isomerase Activity.
J.Am.Chem.Soc., 136, 2014
4CIZ
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BU of 4ciz by Molmil
Crystal structure of the complex of the Cellular Retinal Binding Protein with 9-cis-retinal
Descriptor: L(+)-TARTARIC ACID, RETINAL, RETINALDEHYDE-BINDING PROTEIN 1
Authors:Bolze, C.S, Helbling, R.E, Owen, R.L, Pearson, A.R, Pompidor, G, Dworkowski, F, Fuchs, M.R, Furrer, J, Golczak, M, Palczewski, K, Cascella, M, Stocker, A.
Deposit date:2013-12-18
Release date:2014-01-08
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (3.403 Å)
Cite:Human Cellular Retinaldehyde-Binding Protein Has Secondary Thermal 9-Cis-Retinal Isomerase Activity.
J.Am.Chem.Soc., 136, 2014
8FD1
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BU of 8fd1 by Molmil
Crystal structure of photoactivated rhodopsin in complex with a nanobody
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Nanobody Nb2, ...
Authors:Salom, D, Palczewski, K, Kiser, P.D.
Deposit date:2022-12-01
Release date:2023-08-30
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (4.25 Å)
Cite:Structural basis for the allosteric modulation of rhodopsin by nanobody binding to its extracellular domain.
Nat Commun, 14, 2023
8FD0
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BU of 8fd0 by Molmil
Crystal structure of bovine rod opsin in complex with a nanobody
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Nanobody Nb2, ...
Authors:Salom, D, Palczewski, K, Kiser, P.D.
Deposit date:2022-12-01
Release date:2023-08-30
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (3.71 Å)
Cite:Structural basis for the allosteric modulation of rhodopsin by nanobody binding to its extracellular domain.
Nat Commun, 14, 2023
8FCZ
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BU of 8fcz by Molmil
Crystal structure of ground-state rhodopsin in complex with a nanobody
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Nanobody Nb2, ...
Authors:Salom, D, Palczewski, K, Kiser, P.D.
Deposit date:2022-12-01
Release date:2023-08-30
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (3.7 Å)
Cite:Structural basis for the allosteric modulation of rhodopsin by nanobody binding to its extracellular domain.
Nat Commun, 14, 2023
4ZHK
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BU of 4zhk by Molmil
Crystal structure of RPE65 in complex with MB-002
Descriptor: (1R)-1-[3-(cyclohexylmethoxy)phenyl]propane-1,3-diol, (1S)-1-[3-(cyclohexylmethoxy)phenyl]propane-1,3-diol, FE (II) ION, ...
Authors:Kiser, P.D, Palczewski, K.
Deposit date:2015-04-25
Release date:2015-05-27
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.09 Å)
Cite:Molecular pharmacodynamics of emixustat in protection against retinal degeneration.
J.Clin.Invest., 125, 2015
2NWC
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BU of 2nwc by Molmil
A 3.02 angstrom crystal structure of wild-type apo GroEL in a monoclinic space group
Descriptor: 60 kDa chaperonin
Authors:Kiser, P.D, Lodowski, D.T, Palczewski, K.
Deposit date:2006-11-14
Release date:2007-05-22
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (3.02 Å)
Cite:Purification, crystallization and structure determination of native GroEL from Escherichia coli lacking bound potassium ions
Acta Crystallogr.,Sect.F, 63, 2007
6B20
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BU of 6b20 by Molmil
Crystal structure of a complex between G protein beta gamma dimer and an inhibitory Nanobody regulator
Descriptor: CHLORIDE ION, Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1, Guanine nucleotide-binding protein G(T) subunit gamma-T1, ...
Authors:Gulati, S, Kiser, P.D, Palczewski, K.
Deposit date:2017-09-19
Release date:2018-05-30
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.34 Å)
Cite:Targeting G protein-coupled receptor signaling at the G protein level with a selective nanobody inhibitor.
Nat Commun, 9, 2018
6MZB
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BU of 6mzb by Molmil
Cryo-EM structure of phosphodiesterase 6
Descriptor: GUANOSINE-3',5'-MONOPHOSPHATE, MAGNESIUM ION, Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma, ...
Authors:Gulati, S, Palczewski, K.
Deposit date:2018-11-04
Release date:2019-03-06
Last modified:2021-05-19
Method:ELECTRON MICROSCOPY (3.4 Å)
Cite:Cryo-EM structure of phosphodiesterase 6 reveals insights into the allosteric regulation of type I phosphodiesterases.
Sci Adv, 5, 2019
6OFJ
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BU of 6ofj by Molmil
Cryo-EM structure of the native rhodopsin dimer from rod photoreceptor cells
Descriptor: Rhodopsin
Authors:Zhao, D.Y, Gulati, S, Ernst, O.P, Palczewski, K.
Deposit date:2019-03-30
Release date:2019-08-21
Last modified:2019-12-18
Method:ELECTRON MICROSCOPY (4.5 Å)
Cite:Cryo-EM structure of the native rhodopsin dimer in nanodiscs.
J.Biol.Chem., 294, 2019
3KVC
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BU of 3kvc by Molmil
Crystal structure of bovine RPE65 at 1.9 angstrom resolution
Descriptor: FE (II) ION, Retinoid isomerohydrolase
Authors:Kiser, P.D, Lodowski, D.T, Golczak, M, Palczewski, K.
Deposit date:2009-11-29
Release date:2010-02-02
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Importance of membrane structural integrity for RPE65 retinoid isomerization activity.
J.Biol.Chem., 285, 2010
3LM1
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BU of 3lm1 by Molmil
Crystal Structure Analysis of Maclura pomifera agglutinin complex with p-nitrophenyl-GalNAc
Descriptor: 4-nitrophenyl 2-acetamido-2-deoxy-beta-D-glucopyranoside, Agglutinin alpha chain, Agglutinin beta-2 chain
Authors:Huang, J, Xu, Z, Wang, D, Ogato, C, Hirama, T, Palczewski, K, Hazen, S.L, Lee, X, Young, N.M.
Deposit date:2010-01-29
Release date:2010-09-22
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Characterization of the secondary binding sites of Maclura pomifera agglutinin by glycan array and crystallographic analyses.
Glycobiology, 20, 2010
3LLZ
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BU of 3llz by Molmil
Crystal Structure Analysis of Maclura pomifera agglutinin complex with Gal-beta-1,3-GalNAc
Descriptor: Agglutinin alpha chain, Agglutinin beta-2 chain, beta-D-galactopyranose-(1-3)-2-acetamido-2-deoxy-beta-D-galactopyranose
Authors:Huang, J, Xu, Z, Wang, D, Ogato, C, Hirama, T, Palczewski, K, Hazen, S.L, Lee, X, Young, N.M.
Deposit date:2010-01-29
Release date:2010-09-22
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.55 Å)
Cite:Characterization of the secondary binding sites of Maclura pomifera agglutinin by glycan array and crystallographic analyses.
Glycobiology, 20, 2010
3LLY
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BU of 3lly by Molmil
Crystal Structure Analysis of Maclura pomifera agglutinin
Descriptor: Agglutinin alpha chain, Agglutinin beta-2 chain
Authors:Huang, J, Xu, Z, Wang, D, Ogato, C, Hirama, T, Palczewski, K, Hazen, S.L, Lee, X, Young, N.M.
Deposit date:2010-01-29
Release date:2010-09-22
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (2.25 Å)
Cite:Characterization of the secondary binding sites of Maclura pomifera agglutinin by glycan array and crystallographic analyses.
Glycobiology, 20, 2010
3VAT
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BU of 3vat by Molmil
Crystal structure of DNPEP, ZnMg form
Descriptor: Aspartyl aminopeptidase, MAGNESIUM ION, ZINC ION
Authors:Kiser, P.D, Chen, Y, Palczewski, K.
Deposit date:2011-12-29
Release date:2012-02-29
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Insights into substrate specificity and metal activation of Mammalian tetrahedral aspartyl aminopeptidase.
J.Biol.Chem., 287, 2012
3VAR
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BU of 3var by Molmil
Crystal structure of DNPEP, ZnZn form
Descriptor: Aspartyl aminopeptidase, ZINC ION
Authors:Kiser, P.D, Chen, Y, Palczewski, K.
Deposit date:2011-12-29
Release date:2012-02-29
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (2.25 Å)
Cite:Insights into substrate specificity and metal activation of Mammalian tetrahedral aspartyl aminopeptidase.
J.Biol.Chem., 287, 2012
1HZX
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BU of 1hzx by Molmil
CRYSTAL STRUCTURE OF BOVINE RHODOPSIN
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, HEPTANE-1,2,3-TRIOL, MERCURY (II) ION, ...
Authors:Teller, D.C, Okada, T, Behnke, C.A, Palczewski, K, Stenkamp, R.E.
Deposit date:2001-01-26
Release date:2001-07-04
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:Advances in determination of a high-resolution three-dimensional structure of rhodopsin, a model of G-protein-coupled receptors (GPCRs).
Biochemistry, 40, 2001
1JBA
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BU of 1jba by Molmil
UNMYRISTOYLATED GCAP-2 WITH THREE CALCIUM IONS BOUND
Descriptor: CALCIUM ION, PROTEIN (GUANYLATE CYCLASE ACTIVATING PROTEIN 2)
Authors:Ames, J.B, Dizhoor, A.M, Ikura, M, Palczewski, K, Stryer, L.
Deposit date:1999-04-03
Release date:1999-12-10
Last modified:2023-12-27
Method:SOLUTION NMR
Cite:Three-dimensional structure of guanylyl cyclase activating protein-2, a calcium-sensitive modulator of photoreceptor guanylyl cyclases.
J.Biol.Chem., 274, 1999
7MOR
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BU of 7mor by Molmil
CRYSTAL STRUCTURE OF NATIVE BOVINE ARRESTIN 1 IN COMPLEX WITH 5-METHYLENEBIPHOSPHONATE INOSITOL PENTAKISPHAOPHATE (5-PCP IP5)
Descriptor: Methylenebisphosphonate inositol pentakisphosphate, S-arrestin
Authors:Sander, C.L, Palczewski, K, Kiser, P.D.
Deposit date:2021-05-03
Release date:2021-10-13
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:Structural evidence for visual arrestin priming via complexation of phosphoinositols.
Structure, 30, 2022
7MP2
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BU of 7mp2 by Molmil
CRYSTAL STRUCTURE OF NATIVE BOVINE ARRESTIN 1 IN COMPLEX WITH 1D-MYO-INOSITOL 1,5-BISDIPHOSPHATE TETRAKISPHOSPHATE (1,5-PP IP4)
Descriptor: (1R,3S,4R,5S,6R)-2,4,5,6-tetrakis(phosphonooxy)cyclohexane-1,3-diyl bis[trihydrogen (diphosphate)], S-arrestin
Authors:Sander, C.L, Palczewski, K, Kiser, P.D.
Deposit date:2021-05-04
Release date:2021-10-13
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (3 Å)
Cite:Structural evidence for visual arrestin priming via complexation of phosphoinositols.
Structure, 30, 2022
7MP0
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BU of 7mp0 by Molmil
CRYSTAL STRUCTURE OF NATIVE BOVINE ARRESTIN 1 IN COMPLEX WITH 1D-MYO-INOSITOL 5-DIPHOSPHATE PENTAKISPHOSPHATE (5-PP IP5)
Descriptor: (1r,2R,3S,4s,5R,6S)-2,3,4,5,6-pentakis(phosphonooxy)cyclohexyl trihydrogen diphosphate, 2-ETHOXYETHANOL, S-arrestin
Authors:Sander, C.L, Palczewski, K, Kiser, P.D.
Deposit date:2021-05-04
Release date:2021-10-13
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Structural evidence for visual arrestin priming via complexation of phosphoinositols.
Structure, 30, 2022
7MP1
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BU of 7mp1 by Molmil
CRYSTAL STRUCTURE OF NATIVE BOVINE ARRESTIN 1 IN COMPLEX WITH 1,5-DI-METHYLENEBISPHOSPHONATE INOSITOL TETRAKISPHOSPHATE (1,5-PCP-IP4)
Descriptor: S-arrestin, {[(1R,3S,4S,5R,6S)-2,4,5,6-tetrakis(phosphonooxy)cyclohexane-1,3-diyl]bis[oxy(hydroxyphosphoryl)methanediyl]}bis(phosphonic acid)
Authors:Sander, C.L, Palczewski, K, Kiser, P.D.
Deposit date:2021-05-04
Release date:2021-10-13
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.66 Å)
Cite:Structural evidence for visual arrestin priming via complexation of phosphoinositols.
Structure, 30, 2022
5KJD
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BU of 5kjd by Molmil
Synechocystis apocarotenoid oxygenase (ACO) mutant - Glu150Gln
Descriptor: Apocarotenoid-15,15'-oxygenase, FE (II) ION
Authors:Sui, X, Kiser, P.D, Palczewski, K.
Deposit date:2016-06-18
Release date:2016-08-03
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.75 Å)
Cite:Key Residues for Catalytic Function and Metal Coordination in a Carotenoid Cleavage Dioxygenase.
J.Biol.Chem., 291, 2016
5KK0
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Synechocystis ACO mutant - T136A
Descriptor: Apocarotenoid-15,15'-oxygenase, CHLORIDE ION, FE (II) ION
Authors:Sui, X, Kiser, P.D, Palczewski, K.
Deposit date:2016-06-20
Release date:2016-07-13
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:Utilization of Dioxygen by Carotenoid Cleavage Oxygenases.
J.Biol.Chem., 290, 2015

 

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