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PDB: 214 件

6FAU
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BU of 6fau by Molmil
Crystal structure of C-terminal modified Tau peptide-hybrid 4.2e-I with 14-3-3sigma
分子名称: (2~{R})-2-[(~{R})-(2-methoxyphenyl)-phenyl-methyl]pyrrolidine, 14-3-3 protein sigma, ACE-ARG-THR-PRO-SEP-LEU-PRO-GLY, ...
著者Andrei, S.A, Meijer, F.A, Ottmann, C, Milroy, L.G.
登録日2017-12-18
公開日2018-05-16
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献Inhibition of 14-3-3/Tau by Hybrid Small-Molecule Peptides Operating via Two Different Binding Modes.
ACS Chem Neurosci, 9, 2018
6FI4
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BU of 6fi4 by Molmil
Crystal structure of C-terminal modified Tau peptide-hybrid 3.2e with 14-3-3sigma
分子名称: (2~{S})-2-(diphenylmethyl)pyrrolidine, 14-3-3 protein sigma, CALCIUM ION, ...
著者Andrei, S.A, Meijer, F.A, Ottmann, C, Milroy, L.G.
登録日2018-01-17
公開日2018-05-16
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Inhibition of 14-3-3/Tau by Hybrid Small-Molecule Peptides Operating via Two Different Binding Modes.
ACS Chem Neurosci, 9, 2018
6FAV
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BU of 6fav by Molmil
Crystal structure of C-terminal modified Tau peptide-hybrid 4.2f-I with 14-3-3sigma
分子名称: (2~{R})-2-[(~{R})-(3-methoxyphenyl)-phenyl-methyl]pyrrolidine, 14-3-3 protein sigma, ACE-ARG-THR-PRO-SEP-LEU-PRO-GLY, ...
著者Andrei, S.A, Meijer, F.A, Ottmann, C, Milroy, L.G.
登録日2017-12-18
公開日2018-05-16
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Inhibition of 14-3-3/Tau by Hybrid Small-Molecule Peptides Operating via Two Different Binding Modes.
ACS Chem Neurosci, 9, 2018
6FBY
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BU of 6fby by Molmil
Crystal structure of C-terminal modified Tau peptide-hybrid 4.2b with 14-3-3sigma
分子名称: (2~{R})-2-[(~{S})-(3-methylphenyl)-phenyl-methyl]pyrrolidine, 14-3-3 protein sigma, ACE-ARG-THR-PRO-SEP-LEU-PRO-GLY, ...
著者Andrei, S.A, Meijer, F.A, Ottmann, C, Milroy, L.G.
登録日2017-12-20
公開日2018-05-16
最終更新日2019-02-27
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Inhibition of 14-3-3/Tau by Hybrid Small-Molecule Peptides Operating via Two Different Binding Modes.
ACS Chem Neurosci, 9, 2018
6FI5
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BU of 6fi5 by Molmil
Crystal structure of C-terminal modified Tau peptide-hybrid 3.2d with 14-3-3sigma
分子名称: (2~{S})-2-(diphenylmethyl)pyrrolidine, 14-3-3 protein sigma, CHLORIDE ION, ...
著者Andrei, S.A, Meijer, F.A, Ottmann, C, Milroy, L.G.
登録日2018-01-17
公開日2018-05-16
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Inhibition of 14-3-3/Tau by Hybrid Small-Molecule Peptides Operating via Two Different Binding Modes.
ACS Chem Neurosci, 9, 2018
6FAW
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BU of 6faw by Molmil
Crystal structure of C-terminal modified Tau peptide-hybrid 4.2c-I with 14-3-3sigma
分子名称: (2~{R})-2-[(~{R})-[2-(2-methoxyethoxy)phenyl]-phenyl-methyl]pyrrolidine, 14-3-3 protein sigma, ACE-ARG-THR-PRO-SEP-LEU-PRO-GLY, ...
著者Andrei, S.A, Meijer, F.A, Ottmann, C, Milroy, L.G.
登録日2017-12-18
公開日2018-05-16
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Inhibition of 14-3-3/Tau by Hybrid Small-Molecule Peptides Operating via Two Different Binding Modes.
ACS Chem Neurosci, 9, 2018
6FBW
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BU of 6fbw by Molmil
Crystal structure of C-terminal modified Tau peptide-hybrid 4.2f-II with 14-3-3sigma
分子名称: (2~{R})-2-[(~{S})-(3-methoxyphenyl)-phenyl-methyl]pyrrolidine, 14-3-3 protein sigma, ARG-THR-PRO-SEP-LEU-PRO-GLY, ...
著者Andrei, S.A, Meijer, F.A, Ottmann, C, Milroy, L.G.
登録日2017-12-20
公開日2018-05-16
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Inhibition of 14-3-3/Tau by Hybrid Small-Molecule Peptides Operating via Two Different Binding Modes.
ACS Chem Neurosci, 9, 2018
4TQE
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BU of 4tqe by Molmil
Structure of tau peptide in complex with Tau5 antibody Fab fragment
分子名称: Fab heavy chain, If kappa light chain, Microtubule-associated protein tau, ...
著者Cehlar, O, Skrabana, R, Novak, M.
登録日2014-06-11
公開日2015-07-29
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structure of tau peptide in complex with Tau5 antibody Fab fragment
To Be Published
4Y5I
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BU of 4y5i by Molmil
Crystal structure of C-terminal modified Tau peptide-hybrid 126B with 14-3-3sigma
分子名称: 14-3-3 protein sigma, CHLORIDE ION, Microtubule-associated protein tau
著者Leysen, S, Bartel, M, Milroy, L, Brunsveld, L, Ottmann, C.
登録日2015-02-11
公開日2016-01-13
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Stabilizer-Guided Inhibition of Protein-Protein Interactions.
Angew.Chem.Int.Ed.Engl., 54, 2015
6PXR
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BU of 6pxr by Molmil
Anti-TAU BIIB092 FAB with TAU peptide
分子名称: Microtubule-associated protein tau, gosuranemab Fab, heavy chain, ...
著者Arndt, J.W, Quan, C.
登録日2019-07-26
公開日2020-07-29
最終更新日2021-02-10
実験手法X-RAY DIFFRACTION (1.556 Å)
主引用文献Characterization of tau binding by gosuranemab.
Neurobiol.Dis., 146, 2020
4FL5
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BU of 4fl5 by Molmil
Crystal structure of human 14-3-3 sigma in complex with a Tau-protein peptide surrounding pS214
分子名称: 14-3-3 protein sigma, CALCIUM ION, CHLORIDE ION, ...
著者Schumacher, B, Ottmann, C.
登録日2012-06-14
公開日2013-12-11
最終更新日2017-06-07
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Involvement of 14-3-3 in tubulin instability and impaired axon development is mediated by Tau.
FASEB J., 29, 2015
8KDX
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BU of 8kdx by Molmil
Tau-S214 Phosphorylation Inhibits Fyn Kinase Interaction and Increases the Decay Time of NMDAR-mediated Current
分子名称: Microtubule-associated protein tau, Tyrosine-protein kinase Fyn
著者Padavattan, S, Jos, S.
登録日2023-08-10
公開日2024-02-28
実験手法X-RAY DIFFRACTION (1.01 Å)
主引用文献Tau-S214 Phosphorylation Inhibits Fyn Kinase Interaction and Increases the Decay Time of NMDAR-mediated Current.
J.Mol.Biol., 436, 2024
7PQP
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BU of 7pqp by Molmil
tau-microtubule structural ensemble based on CryoEM data
分子名称: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, Isoform Tau-F of Microtubule-associated protein tau, ...
著者Brotzakis, Z.F, Vendruscolo, M.
登録日2021-09-18
公開日2021-12-15
最終更新日2022-01-12
実験手法ELECTRON MICROSCOPY (4.1 Å)
主引用文献A Structural Ensemble of a Tau-Microtubule Complex Reveals Regulatory Tau Phosphorylation and Acetylation Mechanisms.
Acs Cent.Sci., 7, 2021
7PQC
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BU of 7pqc by Molmil
tau-microtubule structural ensemble based on CryoEM data
分子名称: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, Isoform Tau-F of Microtubule-associated protein tau, ...
著者Brotzakis, Z.F, Vendruscolo, M.
登録日2021-09-16
公開日2021-12-15
最終更新日2022-01-12
実験手法ELECTRON MICROSCOPY (4.1 Å)
主引用文献A Structural Ensemble of a Tau-Microtubule Complex Reveals Regulatory Tau Phosphorylation and Acetylation Mechanisms.
Acs Cent.Sci., 7, 2021

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件を2024-05-15に公開中

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