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PDB: 8 results

8PSY
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BU of 8psy by Molmil
ERK2 covelently bound to RU68 cyclohexenone based inhibitor
Descriptor: AMP PHOSPHORAMIDATE, Mitogen-activated protein kinase 1, ~{O}3-~{tert}-butyl ~{O}1-methyl (1~{S},3~{R})-4-oxidanylidene-1-(phenylmethyl)cyclohexane-1,3-dicarboxylate
Authors:Sok, P, Poti, A, Remenyi, A, Gogl, G.
Deposit date:2023-07-13
Release date:2024-07-24
Last modified:2024-10-16
Method:X-RAY DIFFRACTION (2.55 Å)
Cite:Targeting a key protein-protein interaction surface on mitogen-activated protein kinases by a precision-guided warhead scaffold.
Nat Commun, 15, 2024
8PSW
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BU of 8psw by Molmil
ERK2 covalently bound to RU67 cyclohexenone based inhibitor
Descriptor: AMP PHOSPHORAMIDATE, Mitogen-activated protein kinase 1, ~{O}3-~{tert}-butyl ~{O}1-methyl (1~{R},3~{R})-4-oxidanylidene-1-(phenylmethyl)cyclohexane-1,3-dicarboxylate
Authors:Sok, P, Poti, A, Remenyi, A, Gogl, G.
Deposit date:2023-07-13
Release date:2024-07-24
Last modified:2024-10-16
Method:X-RAY DIFFRACTION (2 Å)
Cite:Targeting a key protein-protein interaction surface on mitogen-activated protein kinases by a precision-guided warhead scaffold.
Nat Commun, 15, 2024
8PT1
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BU of 8pt1 by Molmil
ERK2 covelently bound to RU76 cyclohexenone based inhibitor
Descriptor: Mitogen-activated protein kinase 1, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ~{O}1-methyl ~{O}3-(phenylmethyl) (1~{S},3~{R})-1-methyl-4-oxidanylidene-cyclohexane-1,3-dicarboxylate
Authors:Sok, P, Poti, A, Remenyi, A, Gogl, G.
Deposit date:2023-07-13
Release date:2024-07-24
Last modified:2024-10-16
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Targeting a key protein-protein interaction surface on mitogen-activated protein kinases by a precision-guided warhead scaffold.
Nat Commun, 15, 2024
8PT3
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BU of 8pt3 by Molmil
ERK2 covelently bound to RU77 cyclohexenone based inhibitor
Descriptor: GLYCEROL, Mitogen-activated protein kinase 1, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ...
Authors:Sok, P, Poti, A, Remenyi, A.
Deposit date:2023-07-13
Release date:2024-07-24
Last modified:2024-10-16
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Targeting a key protein-protein interaction surface on mitogen-activated protein kinases by a precision-guided warhead scaffold.
Nat Commun, 15, 2024
8PST
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BU of 8pst by Molmil
ERK2 covelently bound to RU60 cyclohexenone based inhibitor
Descriptor: AMP PHOSPHORAMIDATE, Mitogen-activated protein kinase 1, ~{O}3-~{tert}-butyl ~{O}1-methyl (1~{R},3~{S})-1-methyl-4-oxidanylidene-cyclohexane-1,3-dicarboxylate
Authors:Sok, P, Poti, A, Remenyi, A, Gogl, G.
Deposit date:2023-07-13
Release date:2024-07-24
Last modified:2024-10-16
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Targeting a key protein-protein interaction surface on mitogen-activated protein kinases by a precision-guided warhead scaffold.
Nat Commun, 15, 2024
8PSR
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BU of 8psr by Molmil
ERK2 covalently bound to SynthRevD-12-opt artificial peptide
Descriptor: GLYCEROL, Mitogen-activated protein kinase 1, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ...
Authors:Sok, P, Poti, A, Gogl, G, Remenyi, A.
Deposit date:2023-07-13
Release date:2024-07-24
Last modified:2024-10-16
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Targeting a key protein-protein interaction surface on mitogen-activated protein kinases by a precision-guided warhead scaffold.
Nat Commun, 15, 2024
8PT0
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BU of 8pt0 by Molmil
ERK2 covelently bound to RU75 cyclohexenone based inhibitor
Descriptor: GLYCEROL, Mitogen-activated protein kinase 1, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ...
Authors:Sok, P, Poti, A, Remenyi, A, Gogl, G.
Deposit date:2023-07-13
Release date:2024-07-24
Last modified:2024-10-16
Method:X-RAY DIFFRACTION (1.65 Å)
Cite:Targeting a key protein-protein interaction surface on mitogen-activated protein kinases by a precision-guided warhead scaffold.
Nat Commun, 15, 2024
8PT5
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BU of 8pt5 by Molmil
ERK2 covelently bound to RU187 cyclohexenone based inhibitor
Descriptor: GLYCEROL, Mitogen-activated protein kinase 1, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ...
Authors:Sok, P, Poti, A, Remenyi, A.
Deposit date:2023-07-13
Release date:2024-07-24
Last modified:2024-10-16
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:Targeting a key protein-protein interaction surface on mitogen-activated protein kinases by a precision-guided warhead scaffold.
Nat Commun, 15, 2024

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