4HAT
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![BU of 4hat by Molmil](/molmil-images/mine/4hat) | |
7CND
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![BU of 7cnd by Molmil](/molmil-images/mine/7cnd) | NCI-1 in complex with CRM1-Ran-RanBP1 | Descriptor: | 3[N-MORPHOLINO]PROPANE SULFONIC ACID, CHLORIDE ION, CRM1 isoform 1, ... | Authors: | Sun, Q, Lei, Y. | Deposit date: | 2020-07-31 | Release date: | 2021-06-09 | Last modified: | 2023-11-29 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Structure-Guided Design of the First Noncovalent Small-Molecule Inhibitor of CRM1. J.Med.Chem., 64, 2021
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4HB2
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![BU of 4hb2 by Molmil](/molmil-images/mine/4hb2) | Crystal structure of CRM1-Ran-RanBP1 | Descriptor: | 1,2-ETHANEDIOL, CHLORIDE ION, Exportin-1, ... | Authors: | Sun, Q, Chook, Y.M. | Deposit date: | 2012-09-27 | Release date: | 2013-01-09 | Last modified: | 2024-02-28 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Nuclear export inhibition through covalent conjugation and hydrolysis of Leptomycin B by CRM1. Proc.Natl.Acad.Sci.USA, 110, 2013
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4HAZ
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![BU of 4haz by Molmil](/molmil-images/mine/4haz) | Crystal structure of CRM1 inhibitor Leptomycin B in complex with CRM1(R543S,K548E,K579Q)-Ran-RanBP1 | Descriptor: | CHLORIDE ION, Exportin-1, GTP-binding nuclear protein Ran, ... | Authors: | Sun, Q, Chook, Y.M. | Deposit date: | 2012-09-27 | Release date: | 2013-01-09 | Last modified: | 2017-07-26 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Nuclear export inhibition through covalent conjugation and hydrolysis of Leptomycin B by CRM1. Proc.Natl.Acad.Sci.USA, 110, 2013
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4HAW
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![BU of 4haw by Molmil](/molmil-images/mine/4haw) | |
6XJR
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![BU of 6xjr by Molmil](/molmil-images/mine/6xjr) | |
6XJS
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![BU of 6xjs by Molmil](/molmil-images/mine/6xjs) | |
7L5E
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![BU of 7l5e by Molmil](/molmil-images/mine/7l5e) | |
5OWU
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![BU of 5owu by Molmil](/molmil-images/mine/5owu) | Kap95:Nup1 complex | Descriptor: | Importin subunit beta-1, Nucleoporin NUP1 | Authors: | Stewart, M. | Deposit date: | 2017-09-04 | Release date: | 2017-10-25 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Structural basis for the high-affinity binding of nucleoporin Nup1p to the Saccharomyces cerevisiae importin-beta homologue, Kap95p. J. Mol. Biol., 349, 2005
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3M1I
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![BU of 3m1i by Molmil](/molmil-images/mine/3m1i) | |
4HAV
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![BU of 4hav by Molmil](/molmil-images/mine/4hav) | |
4HAU
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![BU of 4hau by Molmil](/molmil-images/mine/4hau) | |
1WA5
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![BU of 1wa5 by Molmil](/molmil-images/mine/1wa5) | Structure of the Cse1:Imp-alpha:RanGTP complex | Descriptor: | GTP-binding nuclear protein Ran, GUANOSINE-5'-TRIPHOSPHATE, Importin alpha re-exporter, ... | Authors: | Stewart, M. | Deposit date: | 2004-10-23 | Release date: | 2004-12-13 | Last modified: | 2023-12-13 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Structural basis for the assembly of a nuclear export complex. Nature, 432, 2004
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6CIT
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![BU of 6cit by Molmil](/molmil-images/mine/6cit) | |
8HQ6
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![BU of 8hq6 by Molmil](/molmil-images/mine/8hq6) | KL2 in complex with CRM1-Ran-RanBP1 | Descriptor: | CHLORIDE ION, CRM1 isoform 1, DIMETHYL SULFOXIDE, ... | Authors: | Sun, Q, Jian, L. | Deposit date: | 2022-12-13 | Release date: | 2023-10-25 | Method: | X-RAY DIFFRACTION (2.03 Å) | Cite: | Discovery of Aminoratjadone Derivatives as Potent Noncovalent CRM1 Inhibitors. J.Med.Chem., 66, 2023
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5YST
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![BU of 5yst by Molmil](/molmil-images/mine/5yst) | RanM189D in complex with RanBP1-CRM1 | Descriptor: | 1,2-ETHANEDIOL, CHLORIDE ION, Exportin-1,Exportin-1, ... | Authors: | Sun, Q, Zhang, Y. | Deposit date: | 2017-11-15 | Release date: | 2018-11-21 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (2.04 Å) | Cite: | RanM189D in complex with RanBP1-CRM1 To Be Published
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4XRI
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![BU of 4xri by Molmil](/molmil-images/mine/4xri) | Crystal Structure of Importin Beta in an Ammonium Sulfate Condition | Descriptor: | GLYCEROL, Putative uncharacterized protein, SULFATE ION | Authors: | Tauchert, M.J, Neumann, P, Ficner, R, Dickmanns, A. | Deposit date: | 2015-01-21 | Release date: | 2016-01-27 | Last modified: | 2024-01-10 | Method: | X-RAY DIFFRACTION (2.05 Å) | Cite: | Impact of the crystallization condition on importin-beta conformation. Acta Crystallogr D Struct Biol, 72, 2016
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4HB4
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![BU of 4hb4 by Molmil](/molmil-images/mine/4hb4) | |
5UWP
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![BU of 5uwp by Molmil](/molmil-images/mine/5uwp) | |
7DBG
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![BU of 7dbg by Molmil](/molmil-images/mine/7dbg) | Yeast CRM1e (apo) in complex with Ran-RanBP1 | Descriptor: | 3[N-MORPHOLINO]PROPANE SULFONIC ACID, CHLORIDE ION, CRM1 isoform 1, ... | Authors: | Sun, Q, Lei, Y. | Deposit date: | 2020-10-20 | Release date: | 2021-09-29 | Last modified: | 2023-11-29 | Method: | X-RAY DIFFRACTION (2.06 Å) | Cite: | Novel Mechanistic Observations and NES-Binding Groove Features Revealed by the CRM1 Inhibitors Plumbagin and Oridonin. J.Nat.Prod., 84, 2021
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5DIF
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![BU of 5dif by Molmil](/molmil-images/mine/5dif) | |
8HQ3
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![BU of 8hq3 by Molmil](/molmil-images/mine/8hq3) | KL1 in complex with CRM1-Ran-RanBP1 | Descriptor: | CHLORIDE ION, CRM1 isoform 1, DIMETHYL SULFOXIDE, ... | Authors: | Sun, Q, Jian, L. | Deposit date: | 2022-12-13 | Release date: | 2023-10-25 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | Discovery of Aminoratjadone Derivatives as Potent Noncovalent CRM1 Inhibitors. J.Med.Chem., 66, 2023
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4GMX
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![BU of 4gmx by Molmil](/molmil-images/mine/4gmx) | |
3VYC
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![BU of 3vyc by Molmil](/molmil-images/mine/3vyc) | |
8HQ4
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![BU of 8hq4 by Molmil](/molmil-images/mine/8hq4) | B27 in complex with CRM1-Ran-RanBP1 | Descriptor: | 3-[(4-fluorophenyl)carbonylamino]-4-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]benzoic acid, CHLORIDE ION, CRM1 isoform 1, ... | Authors: | Lei, Y, Sun, Q. | Deposit date: | 2022-12-13 | Release date: | 2023-12-20 | Method: | X-RAY DIFFRACTION (2.12 Å) | Cite: | B27 in complex with CRM1-Ran-RanBP1 To Be Published
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