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6O9I
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BU of 6o9i by Molmil
Ternary complex of mouse ECD with Fab1 and Fab2
分子名称: 1,2-ETHANEDIOL, Fab 2 heavy chain, Fab1 heavy chain, ...
著者Min, X, Wang, Z.
登録日2019-03-13
公開日2020-01-22
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Molecular mechanism of an antagonistic antibody against glucose-dependent insulinotropic polypeptide receptor.
Mabs, 12, 2020
7P8X
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Crystal Structure of leukotoxin LukE from Staphylococcus aureus in complex with a doubly sulfated CCR2 N-terminal peptide
分子名称: C-C chemokine receptor type 2, IMIDAZOLE, Leucotoxin LukEv, ...
著者Lambey, P, Hoh, F, Peysson, F, Granier, S, Leyrat, C.
登録日2021-07-23
公開日2022-04-06
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Structural insights into recognition of chemokine receptors by Staphylococcus aureus leukotoxins.
Elife, 11, 2022
7P8U
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Crystal Structure of leukotoxin LukE from Staphylococcus aureus in complex with p-cresyl sulfate
分子名称: (4-methylphenyl) hydrogen sulfate, DI(HYDROXYETHYL)ETHER, IMIDAZOLE, ...
著者Lambey, P, Hoh, F, Peysson, F, Granier, S, Leyrat, C.
登録日2021-07-23
公開日2022-04-06
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural insights into recognition of chemokine receptors by Staphylococcus aureus leukotoxins.
Elife, 11, 2022
7P93
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Crystal Structure of leukotoxin LukE from Staphylococcus aureus in complex with a sulfated ACKR1 N-terminal peptide
分子名称: Atypical chemokine receptor 1, Leucotoxin LukEv
著者Lambey, P, Hoh, F, Peysson, F, Granier, S, Leyrat, C.
登録日2021-07-23
公開日2022-04-06
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Structural insights into recognition of chemokine receptors by Staphylococcus aureus leukotoxins.
Elife, 11, 2022
7P8T
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BU of 7p8t by Molmil
Crystal Structure of leukotoxin LukE from Staphylococcus aureus at 1.5 Angstrom resolution
分子名称: CHLORIDE ION, Leucotoxin LukEv
著者Lambey, P, Hoh, F, Granier, S, Leyrat, C.
登録日2021-07-23
公開日2022-04-06
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.459 Å)
主引用文献Structural insights into recognition of chemokine receptors by Staphylococcus aureus leukotoxins.
Elife, 11, 2022
7P8S
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BU of 7p8s by Molmil
Crystal Structure of leukotoxin LukE from Staphylococcus aureus at 1.9 Angstrom resolution
分子名称: (CARBAMOYLMETHYL-CARBOXYMETHYL-AMINO)-ACETIC ACID, HEXAETHYLENE GLYCOL, Leucotoxin LukEv, ...
著者Lambey, P, Hoh, F, Granier, S, Leyrat, C.
登録日2021-07-23
公開日2022-04-06
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural insights into recognition of chemokine receptors by Staphylococcus aureus leukotoxins.
Elife, 11, 2022
6O9H
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BU of 6o9h by Molmil
Mouse ECD with Fab1
分子名称: Gastric inhibitory polypeptide receptor, Heavy chain, Light chain, ...
著者Min, X, Wang, Z.
登録日2019-03-13
公開日2020-01-22
最終更新日2020-04-01
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Molecular mechanism of an antagonistic antibody against glucose-dependent insulinotropic polypeptide receptor.
Mabs, 12, 2020
5KQE
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BU of 5kqe by Molmil
Solution structure of P2a-J2a/b-P2b of medaka telomerase RNA
分子名称: Telomerase RNA P2ab
著者Wang, Y, Feigon, J.
登録日2016-07-06
公開日2016-08-24
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Structural conservation in the template/pseudoknot domain of vertebrate telomerase RNA from teleost fish to human.
Proc.Natl.Acad.Sci.USA, 113, 2016
5BJ3
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BU of 5bj3 by Molmil
THERMUS THERMOPHILUS ASPARTATE AMINOTRANSFERASE TETRA MUTANT 1
分子名称: PROTEIN (ASPARTATE AMINOTRANSFERASE), PYRIDOXAL-5'-PHOSPHATE
著者Ura, H, Nakai, T, Kawaguchi, S.I, Miyahara, I, Hirotsu, K, Kuramitsu, S.
登録日1999-01-11
公開日2003-09-02
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Substrate recognition mechanism of thermophilic dual-substrate enzyme
J.BIOCHEM.(TOKYO), 130, 2001
5F87
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Crystal structure of Drosophila Poglut1 (Rumi) complexed with UDP
分子名称: GLYCEROL, O-glucosyltransferase rumi, URIDINE-5'-DIPHOSPHATE
著者Yu, H.J, Li, H.L.
登録日2015-12-09
公開日2016-07-20
最終更新日2018-04-18
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structural analysis of Notch-regulating Rumi reveals basis for pathogenic mutations.
Nat. Chem. Biol., 12, 2016
5F84
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BU of 5f84 by Molmil
Crystal structure of Drosophila Poglut1 (Rumi) complexed with its glycoprotein product (glucosylated EGF repeat) and UDP
分子名称: Coagulation factor IX, O-glucosyltransferase rumi, SULFATE ION, ...
著者Yu, H.J, Li, H.L.
登録日2015-12-09
公開日2016-07-20
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural analysis of Notch-regulating Rumi reveals basis for pathogenic mutations.
Nat. Chem. Biol., 12, 2016
1CS4
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BU of 1cs4 by Molmil
COMPLEX OF GS-ALPHA WITH THE CATALYTIC DOMAINS OF MAMMALIAN ADENYLYL CYCLASE: COMPLEX WITH 2'-DEOXY-ADENOSINE 3'-MONOPHOSPHATE, PYROPHOSPHATE AND MG
分子名称: 2'-DEOXY-ADENOSINE 3'-MONOPHOSPHATE, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 5'-GUANOSINE-DIPHOSPHATE-MONOTHIOPHOSPHATE, ...
著者Tesmer, J.J.G, Dessauer, C.A, Sunahara, R.K, Johnson, R.A, Gilman, A.G, Sprang, S.R.
登録日1999-08-16
公開日2001-01-10
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Molecular basis for P-site inhibition of adenylyl cyclase.
Biochemistry, 39, 2000
5NUN
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BU of 5nun by Molmil
Engineered beta-lactoglobulin: variant F105L-L39A-M107F in complex with chlorpromazine (LG-LAF-CLP)
分子名称: 3-(2-chloro-10H-phenothiazin-10-yl)-N,N-dimethylpropan-1-amine, Beta-lactoglobulin
著者Loch, J.I, Bonarek, P, Towrzydlo, M, Lazinskia, I, Szydlowska, J, Lewinski, K.
登録日2017-04-30
公開日2018-04-04
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献The engineered beta-lactoglobulin with complementarity to the chlorpromazine chiral conformers.
Int. J. Biol. Macromol., 114, 2018
1CUL
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BU of 1cul by Molmil
COMPLEX OF GS-ALPHA WITH THE CATALYTIC DOMAINS OF MAMMALIAN ADENYLYL CYCLASE: COMPLEX WITH 2',5'-DIDEOXY-ADENOSINE 3'-TRIPHOSPHATE AND MG
分子名称: 2',5'-DIDEOXY-ADENOSINE 3'-MONOPHOSPHATE, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 5'-GUANOSINE-DIPHOSPHATE-MONOTHIOPHOSPHATE, ...
著者Tesmer, J.J.G, Dessauer, C.A, Sunahara, R.K, Johnson, R.A, Gilman, A.G, Sprang, S.R.
登録日1999-08-20
公開日2001-01-10
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Molecular basis for P-site inhibition of adenylyl cyclase.
Biochemistry, 39, 2000
4QYA
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BU of 4qya by Molmil
Crystal structure of human transthyretin variant V30M in complex with luteolin
分子名称: 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4-one, SODIUM ION, Transthyretin
著者Begum, A, Olofsson, A, Sauer-Eriksson, A.E.
登録日2014-07-24
公開日2015-06-03
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The flavonoid luteolin, but not luteolin-7-o-glucoside, prevents a transthyretin mediated toxic response.
Plos One, 10, 2015
5NUM
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BU of 5num by Molmil
Engineered beta-lactoglobulin: variant F105L-L39A in complex with chlorpromazine (LG-LA-CLP)
分子名称: 3-(2-chloro-10H-phenothiazin-10-yl)-N,N-dimethylpropan-1-amine, Beta-lactoglobulin, PHOSPHATE ION
著者Loch, J.I, Bonarek, P, Tworzydlo, M, Lazinska, I, Szydlowska, J, Lewinski, K.
登録日2017-04-30
公開日2018-04-04
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献The engineered beta-lactoglobulin with complementarity to the chlorpromazine chiral conformers.
Int. J. Biol. Macromol., 114, 2018
5NUJ
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BU of 5nuj by Molmil
Engineered beta-lactoglobulin: variant I56F-L39A in complex with chlorpromazine (LG-FA-CLP)
分子名称: 3-(2-chloro-10H-phenothiazin-10-yl)-N,N-dimethylpropan-1-amine, Beta-lactoglobulin
著者Loch, J.I, Bonarek, P, Tworzydlo, M, Lazinska, I, Szydlowska, J, Lewinski, K.
登録日2017-04-30
公開日2018-04-04
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献The engineered beta-lactoglobulin with complementarity to the chlorpromazine chiral conformers.
Int. J. Biol. Macromol., 114, 2018
5F86
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BU of 5f86 by Molmil
Crystal structure of Drosophila Poglut1 (Rumi) complexed with its substrate protein (EGF repeat)
分子名称: Coagulation factor IX, GLYCEROL, O-glucosyltransferase rumi, ...
著者Yu, H.J, Li, H.L.
登録日2015-12-09
公開日2016-07-20
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural analysis of Notch-regulating Rumi reveals basis for pathogenic mutations.
Nat. Chem. Biol., 12, 2016
6ZBX
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BU of 6zbx by Molmil
Structure of the catalytic domain of the Bacillus circulans alpha-1,6 Mannanase in complex with an alpha-1,6- alpha-manno-cyclophellitol carbasugar-stabilised trisaccharide inhibitor
分子名称: (1~{S},2~{R},3~{S},4~{R},5~{R})-5-(hydroxymethyl)cyclohexane-1,2,3,4-tetrol, (1~{S},4~{S},5~{R})-6-(hydroxymethyl)cyclohexane-1,2,3,4,5-pentol, 1,2-ETHANEDIOL, ...
著者Schroeder, S, Offen, W.A, Jin, Y, De Boer, C, Enoterpi, J, Marino, L, van der Marel, G.A, Codee, J.D.C, Overkleeft, H.S, Davies, G.J.
登録日2020-06-09
公開日2021-04-28
最終更新日2024-10-09
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Development of Non-Hydrolysable Oligosaccharide Activity-Based Inactivators for Endoglycanases: A Case Study on alpha-1,6 Mannanases.
Chemistry, 27, 2021
5F85
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BU of 5f85 by Molmil
Crystal structure of Drosophila Poglut1 (Rumi) complexed with its substrate protein (EGF repeat) and UDP
分子名称: Coagulation factor IX, GLYCEROL, O-glucosyltransferase rumi, ...
著者Yu, H.J, Li, H.L.
登録日2015-12-09
公開日2016-07-20
最終更新日2018-04-18
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Structural analysis of Notch-regulating Rumi reveals basis for pathogenic mutations.
Nat. Chem. Biol., 12, 2016
5NUK
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BU of 5nuk by Molmil
Engineered beta-lactoglobulin: variant I56F-L39A-M107F in complex with chlorpromazine (LG-FAF-CLP)
分子名称: 3-(2-chloro-10H-phenothiazin-10-yl)-N,N-dimethylpropan-1-amine, Beta-lactoglobulin, CHLORIDE ION, ...
著者Loch, J.I, Bonarek, P, Tworzydlo, M, Lazinska, I, Szydlowska, J, Lewinski, K.
登録日2017-04-30
公開日2018-04-04
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The engineered beta-lactoglobulin with complementarity to the chlorpromazine chiral conformers.
Int. J. Biol. Macromol., 114, 2018
4QXV
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BU of 4qxv by Molmil
CRYSTAL STRUCTURE of HUMAN TRANSTHYRETIN IN COMPLEX WITH LUTEOLIN AT 1.1 A RESOLUTION
分子名称: 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4-one, GLYCEROL, SODIUM ION, ...
著者Begum, A, Olofsson, A, Sauer-Eriksson, A.E.
登録日2014-07-22
公開日2015-06-03
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.12 Å)
主引用文献The flavonoid luteolin, but not luteolin-7-o-glucoside, prevents a transthyretin mediated toxic response.
Plos One, 10, 2015
6VII
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BU of 6vii by Molmil
Crystal structure of mouse RABL3 in complex with GTPgammaS
分子名称: 5'-GUANOSINE-DIPHOSPHATE-MONOTHIOPHOSPHATE, MAGNESIUM ION, Rab-like protein 3
著者Su, L, Tomchick, D.R, Beutler, B.
登録日2020-01-13
公開日2020-04-08
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Genetic and structural studies of RABL3 reveal an essential role in lymphoid development and function.
Proc.Natl.Acad.Sci.USA, 117, 2020
5GRT
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BU of 5grt by Molmil
HUMAN GLUTATHIONE REDUCTASE A34E, R37W MUTANT, GLUTATHIONYLSPERMIDINE COMPLEX
分子名称: FLAVIN-ADENINE DINUCLEOTIDE, GLUTATHIONE REDUCTASE, GLUTATHIONYLSPERMIDINE DISULFIDE
著者Stoll, V.S, Simpson, S.J, Krauth-Siegel, R.L, Walsh, C.T, Pai, E.F.
登録日1997-02-12
公開日1997-08-12
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Glutathione reductase turned into trypanothione reductase: structural analysis of an engineered change in substrate specificity.
Biochemistry, 36, 1997
6VIK
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BU of 6vik by Molmil
Crystal structure of mouse xm RABL3 in complex with GTPgammsS
分子名称: 5'-GUANOSINE-DIPHOSPHATE-MONOTHIOPHOSPHATE, MAGNESIUM ION, Rab-like protein 3
著者Su, L, Tomchick, D.R, Beutler, B.
登録日2020-01-13
公開日2020-04-08
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Genetic and structural studies of RABL3 reveal an essential role in lymphoid development and function.
Proc.Natl.Acad.Sci.USA, 117, 2020

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